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CPT

Isoform-selective Products

CPT Products

All (4)
CPT Inhibitors (2)
CPT Activator (1)
CPT Agonist (1)
New CPT Products

Catalog No.	Product Name	Information	Product Use Citations	Product Validations
S8244	Etomoxir sodium salt	Etomoxir sodium salt ((R)-(+)-Etomoxir sodium salt) is an irreversible inhibitor of carnitine palmitoyltransferase-1 (CPT-1) on the outer face of the inner mitochondrial membrane. Etomoxir enhances palmitate-induced cell apoptosis.	Bioact Mater, 2024, 35:549-563 Oncogene, 2024, 43(6):406-419 Biochem Pharmacol, 2024, S0006-2952(24)00144-8
S9819	C75	C75 (4-Methylene-2-octyl-5-oxotetrahydrofuran-3-carboxylic acid) , a more stable synthetic mimic of cerulenin, inhibits fatty-acid synthase (FAS/FASN) with an IC50 of 15.53 μM and has potential therapeutic effects in several cancer models. C75 is also a potent CPT1A activator.	Theranostics, 2023, 13(13):4482-4496 Theranostics, 2023, 10.7150/thno.84921 Front Microbiol, 2022, 13:961942
S6959	Perhexiline maleate	Perhexiline maleate is a potent inhibitor of carnitine palmitoyltransferase 1 (CPT1) with IC50s of 77 μM and 148 μM for rat heart CPT1 and liver CPT1, respectively, and also inhibits carnitine palmitoyltransferase 2 (CPT2).	Cancer Cell, 2022, S1535-6108(22)00312-9
S2269	Baicalin	Baicalin is an inhibitor of prolyl oligopeptidase and also is an allosteric activator of carnitine palmityl transferase 1 (CPT1). Baicalin reduces the expression of NF-κB.	Chem Biol Interact, 2024, 387:110820 Int J Mol Sci, 2023, 24(11)9435 Molecules, 2021, 26(5)1210
S8244	Etomoxir sodium salt	Etomoxir sodium salt ((R)-(+)-Etomoxir sodium salt) is an irreversible inhibitor of carnitine palmitoyltransferase-1 (CPT-1) on the outer face of the inner mitochondrial membrane. Etomoxir enhances palmitate-induced cell apoptosis.	Bioact Mater, 2024, 35:549-563 Oncogene, 2024, 43(6):406-419 Biochem Pharmacol, 2024, S0006-2952(24)00144-8
S6959	Perhexiline maleate	Perhexiline maleate is a potent inhibitor of carnitine palmitoyltransferase 1 (CPT1) with IC50s of 77 μM and 148 μM for rat heart CPT1 and liver CPT1, respectively, and also inhibits carnitine palmitoyltransferase 2 (CPT2).	Cancer Cell, 2022, S1535-6108(22)00312-9
S2269	Baicalin	Baicalin is an inhibitor of prolyl oligopeptidase and also is an allosteric activator of carnitine palmityl transferase 1 (CPT1). Baicalin reduces the expression of NF-κB.	Chem Biol Interact, 2024, 387:110820 Int J Mol Sci, 2023, 24(11)9435 Molecules, 2021, 26(5)1210
S9819	C75	C75 (4-Methylene-2-octyl-5-oxotetrahydrofuran-3-carboxylic acid) , a more stable synthetic mimic of cerulenin, inhibits fatty-acid synthase (FAS/FASN) with an IC50 of 15.53 μM and has potential therapeutic effects in several cancer models. C75 is also a potent CPT1A activator.	Theranostics, 2023, 13(13):4482-4496 Theranostics, 2023, 10.7150/thno.84921 Front Microbiol, 2022, 13:961942

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