Others

  • Inhibitory Selectivity
  • Solubility
Catalog No. Product Name Solubility(25°C)
Water DMSO Alcohol
S1097 BTZ043 Racemate <1 mg/mL 22 mg/mL <1 mg/mL
S6002 NXY-059 (Disufenton sodium) 76 mg/mL 76 mg/mL <1 mg/mL
S1751 Gadodiamide Hydrate 100 mg/mL <1 mg/mL <1 mg/mL
S1236 Leucovorin Calcium Pentahydrate 40 mg/mL <1 mg/mL <1 mg/mL
S1591 Bestatin <1 mg/mL 0.4 mg/mL <1 mg/mL
S8446 Importazole <1 mg/mL 63 mg/mL 31 mg/mL
S4742 Rebaudioside C 100 mg/mL 100 mg/mL 8 mg/mL
S4746 (20S)-Protopanaxadiol <1 mg/mL 92 mg/mL 33 mg/mL
S4739 Oxyresveratrol 1 mg/mL 48 mg/mL 48 mg/mL
S2301 Genistin (Genistoside) <1 mg/mL 86 mg/mL 34 mg/mL
S8368 LM10 <1 mg/mL 45 mg/mL 11 mg/mL
S8269 CFSE <1 mg/mL 100 mg/mL <1 mg/mL
S4701 2-Deoxy-D-glucose 32 mg/mL 32 mg/mL 1 mg/mL
S4703 Choline bitartrate 50 mg/mL <1 mg/mL <1 mg/mL
S8251 Necrosulfonamide <1 mg/mL 92 mg/mL <1 mg/mL
S8358 WNK463 <1 mg/mL 92 mg/mL 92 mg/mL
S4704 D-(+)-Cellobiose 68 mg/mL 3 mg/mL <1 mg/mL
S4728 3,3'-Diindolylmethane <1 mg/mL 49 mg/mL 18 mg/mL
S4721 L-Glutamic acid monosodium salt 33 mg/mL <1 mg/mL <1 mg/mL
S4667 Lidocaine hydrochloride 54 mg/mL 54 mg/mL 54 mg/mL
S4689 Deoxycholic acid <1 mg/mL 78 mg/mL 60 mg/mL
S8321 MLR-1023 <1 mg/mL 40 mg/mL 23 mg/mL
S8284 Fatostatin HBr <1 mg/mL 7 mg/mL 25 mg/mL
S8299 HA15 <1 mg/mL 93 mg/mL 45 mg/mL
S4562 Dehydrocholic acid <1 mg/mL 80 mg/mL 15 mg/mL
S4607 2,2′-Dihydroxy-4-methoxybenzophenone <1 mg/mL 48 mg/mL 48 mg/mL
S4691 Oxybenzone <1 mg/mL 45 mg/mL 45 mg/mL
S4659 Nandrolone <1 mg/mL 54 mg/mL 54 mg/mL
S4658 Hydroquinidine <1 mg/mL 65 mg/mL <1 mg/mL
S4646 Ciclesonide <1 mg/mL 100 mg/mL 100 mg/mL
S4664 Molsidomine 9 mg/mL 48 mg/mL 48 mg/mL
S4515 Ademetionine disulfate tosylate 79 mg/mL 79 mg/mL <1 mg/mL
S4670 Sucralfate <1 mg/mL 0.01 mg/mL <1 mg/mL
S4680 Protirelin 72 mg/mL 72 mg/mL 72 mg/mL
S4652 Sulisobenzone 61 mg/mL 61 mg/mL 61 mg/mL
S4657 Eslicarbazepine Acetate <1 mg/mL 59 mg/mL 11 mg/mL
S4608 L-Tyrosine <1 mg/mL 0.1 mg/mL <1 mg/mL
S4606 Glutathione 61 mg/mL <1 mg/mL <1 mg/mL
S8234 RS-1 <1 mg/mL 100 mg/mL <1 mg/mL
S4615 Modafinil <1 mg/mL 54 mg/mL <1 mg/mL
S4640 Lesinurad <1 mg/mL 80 mg/mL 54 mg/mL
S4633 Isosorbide Mononitrate 38 mg/mL 38 mg/mL 38 mg/mL
S4624 5,5-Dimethyloxazolidine-2,4-dione 84 mg/mL 84 mg/mL 84 mg/mL
S4653 L-Ornithine 26 mg/mL <1 mg/mL <1 mg/mL
S4583 Butamben 38 mg/mL 38 mg/mL 38 mg/mL
S4616 Nandrolone decanoate 85 mg/mL 85 mg/mL 85 mg/mL
S4566 DL-Panthenol 41 mg/mL 41 mg/mL 41 mg/mL
S4558 Citiolone 31 mg/mL 31 mg/mL 31 mg/mL
S4556 Carzenide <1 mg/mL 40 mg/mL 12 mg/mL
S4549 Antimonyl potassium tartrate trihydrate 100 mg/mL <1 mg/mL <1 mg/mL
S4577 Terpin hydrate <1 mg/mL 38 mg/mL 38 mg/mL
S4546 Xylitol 30 mg/mL 30 mg/mL <1 mg/mL
S4544 Urethane 17 mg/mL 17 mg/mL 17 mg/mL
S4535 Methylene Blue 63 mg/mL 63 mg/mL 10 mg/mL
S4514 Acetylleucine <1 mg/mL 34 mg/mL 34 mg/mL
S4512 Aceglutamide 37 mg/mL 37 mg/mL <1 mg/mL
S4548 Aminoguanidine hydrochloride 22 mg/mL 22 mg/mL <1 mg/mL
S4561 Danthron <1 mg/mL 4 mg/mL <1 mg/mL
S4551 Bisoctrizole <1 mg/mL 0.01 mg/mL <1 mg/mL
S4543 Trimetazidine dihydrochloride 67 mg/mL 67 mg/mL 67 mg/mL
S4567 Eprodisate disodium 49 mg/mL <1 mg/mL <1 mg/mL
S8181 SBI-0640756 <1 mg/mL 80 mg/mL <1 mg/mL
S8185 FPS-ZM1 <1 mg/mL 65 mg/mL 65 mg/mL
S1601 Reserpine <1 mg/mL 13 mg/mL <1 mg/mL
S1627 Nitazoxanide <1 mg/mL 62 mg/mL <1 mg/mL
S1137 Malotilate <1 mg/mL 58 mg/mL 58 mg/mL
S1934 Nystatin (Fungicidin) <1 mg/mL 19 mg/mL <1 mg/mL
S1428 Risedronate Sodium 2 mg/mL <1 mg/mL <1 mg/mL
S1271 Acarbose 100 mg/mL 100 mg/mL 8 mg/mL
S2757 TH-302 10 mg/mL 90 mg/mL 90 mg/mL
S1624 Alendronate sodium trihydrate <1 mg/mL <1 mg/mL <1 mg/mL
S1311 Pamidronate Disodium 56 mg/mL <1 mg/mL <1 mg/mL
S2553 5-Aminolevulinic acid HCl 34 mg/mL 34 mg/mL 6 mg/mL
S1201 Dimesna 65 mg/mL 65 mg/mL <1 mg/mL
S1732 Mitotane <1 mg/mL 64 mg/mL 64 mg/mL
S2417 20-Hydroxyecdysone <1 mg/mL 96 mg/mL 96 mg/mL
S1326 Edaravone <1 mg/mL 35 mg/mL 35 mg/mL
S1897 Potassium Iodide 33 mg/mL 33 mg/mL <1 mg/mL
S1988 Propylthiouracil <1 mg/mL 34 mg/mL 19 mg/mL
S2586 Dimethyl Fumarate <1 mg/mL 29 mg/mL 10 mg/mL
S1740 Guaifenesin 25 mg/mL 40 mg/mL 40 mg/mL
S3038 Fosaprepitant dimeglumine salt 135 mg/mL 201 mg/mL <1 mg/mL
S1698 Torsemide <1 mg/mL 3 mg/mL <1 mg/mL
S7372 PTC-209 <1 mg/mL 99 mg/mL <1 mg/mL
S7270 SRPIN340 <1 mg/mL 70 mg/mL 70 mg/mL
S4067 Deferiprone 1 mg/mL <1 mg/mL <1 mg/mL
S7272 4μ8C <1 mg/mL 19 mg/mL <1 mg/mL
S2129 Fudosteine 36 mg/mL <1 mg/mL <1 mg/mL
S1287 Bumetanide <1 mg/mL 73 mg/mL 36 mg/mL
S8077 RI-1 <1 mg/mL 50 mg/mL <1 mg/mL
S7217 OAC1 <1 mg/mL 47 mg/mL 21 mg/mL
S1849 Daidzein <1 mg/mL 51 mg/mL <1 mg/mL
S2408 Cephalomannine <1 mg/mL 100 mg/mL 100 mg/mL
S2610 Lonidamine <1 mg/mL 64 mg/mL <1 mg/mL
S7365 AdipoRon <1 mg/mL 86 mg/mL 50 mg/mL
S4059 Sodium Nitroprusside Dihydrate 60 mg/mL 60 mg/mL <1 mg/mL
S7450 FH1(BRD-K4477) <1 mg/mL 56 mg/mL <1 mg/mL
S2155 LY2608204 <1 mg/mL 112 mg/mL 35 mg/mL
S1749 L-Glutamine 29 mg/mL <1 mg/mL <1 mg/mL
S2901 CCG 50014 <1 mg/mL 63 mg/mL <1 mg/mL
S2035 Epalrestat <1 mg/mL 3 mg/mL <1 mg/mL
S1917 Crystal Violet 14 mg/mL 82 mg/mL 8 mg/mL
S1874 Risedronate <1 mg/mL <1 mg/mL <1 mg/mL
S2412 Genipin <1 mg/mL 45 mg/mL 45 mg/mL
S3199 Reboxetine mesylate 82 mg/mL 82 mg/mL <1 mg/mL
S2410 Paeoniflorin 96 mg/mL 96 mg/mL 96 mg/mL
S1609 Methimazole 23 mg/mL 23 mg/mL 23 mg/mL
S2594 Pramiracetam <1 mg/mL 54 mg/mL <1 mg/mL
S7369 4EGI-1 <1 mg/mL 90 mg/mL <1 mg/mL
S2388 L-carnitine 32 mg/mL 12 mg/mL 32 mg/mL
S1643 Ursodiol <1 mg/mL 79 mg/mL 79 mg/mL
S1647 Adenosine <1 mg/mL 12 mg/mL <1 mg/mL
S1671 (6-)ε-​Aminocaproic acid 26 mg/mL 6 mg/mL 1 mg/mL
S1853 Penicillamine 30 mg/mL <1 mg/mL <1 mg/mL
S2536 Miconazole <1 mg/mL 83 mg/mL 83 mg/mL
S2724 Heparin sodium 100 mg/mL <1 mg/mL <1 mg/mL
S1806 Acipimox <1 mg/mL 31 mg/mL <1 mg/mL
S4217 Liothyronine Sodium <1 mg/mL 100 mg/mL <1 mg/mL
S1985 ATP 100 mg/mL <1 mg/mL <1 mg/mL
S3148 Ibandronate sodium 72 mg/mL <1 mg/mL <1 mg/mL
S3150 Articaine HCl 64 mg/mL 64 mg/mL 64 mg/mL
S1875 Tranexamic Acid 31 mg/mL <1 mg/mL <1 mg/mL
S3000 Carbazochrome sodium sulfonate (AC-17) 3 mg/mL 64 mg/mL <1 mg/mL
S2599 L-Thyroxine <1 mg/mL 100 mg/mL <1 mg/mL
S1610 Metolazone <1 mg/mL 73 mg/mL 8 mg/mL
S4020 Sodium Picosulfate 96 mg/mL 96 mg/mL 3 mg/mL
S4129 Sevelamer HCl <1 mg/mL 0.005 mg/mL <1 mg/mL
S2381 D-Mannitol 36 mg/mL 36 mg/mL <1 mg/mL
S2393 Sorbitol 36 mg/mL 36 mg/mL <1 mg/mL
S1641 Chlorothiazide <1 mg/mL 59 mg/mL <1 mg/mL
S2293 DL-Carnitine HCl 40 mg/mL 40 mg/mL <1 mg/mL
S2305 Grape Seed Extract <1 mg/mL 94 mg/mL <1 mg/mL
S1715 Glipizide <1 mg/mL 89 mg/mL <1 mg/mL
S4095 Difluprednate <1 mg/mL 100 mg/mL 25 mg/mL
S2032 Rebamipide <1 mg/mL 74 mg/mL <1 mg/mL
S1928 Alibendol <1 mg/mL 50 mg/mL 50 mg/mL
S1735 Mesna 7 mg/mL 33 mg/mL <1 mg/mL
S2411 Geniposide 78 mg/mL 78 mg/mL <1 mg/mL
S2409 10-Deacetylbaccatin-III <1 mg/mL 109 mg/mL <1 mg/mL
S3209 Amidopyrine 10 mg/mL 46 mg/mL 46 mg/mL
S7382 Phosphoramidon Disodium Salt 100 mg/mL 100 mg/mL <1 mg/mL
S7589 N6022 <1 mg/mL 82 mg/mL 5 mg/mL
S7922 Tiplaxtinin (PAI-039) <1 mg/mL 72 mg/mL 18 mg/mL
S1511 Lactulose 68 mg/mL 68 mg/mL <1 mg/mL
S1708 Hydrochlorothiazide 0 mg/mL 0 mg/mL 0 mg/mL
S2596 Clindamycin palmitate HCl 140 mg/mL 140 mg/mL 140 mg/mL
S4298 Amifostine 42 mg/mL <1 mg/mL <1 mg/mL
S7909 Dp44mT <1 mg/mL 57 mg/mL 47 mg/mL
S7913 MCB-613 <1 mg/mL 60 mg/mL 60 mg/mL
S4299 Dicoumarol <1 mg/mL 67 mg/mL 67 mg/mL
S4017 Allylthiourea <1 mg/mL 23 mg/mL 23 mg/mL
S2830 Clindamycin <1 mg/mL 85 mg/mL 85 mg/mL
S7914 Isoxazole 9 (ISX-9) <1 mg/mL 46 mg/mL 13 mg/mL
S2589 Miglitol <1 mg/mL 3 mg/mL <1 mg/mL
S2518 NAD+ 100 mg/mL <1 mg/mL <1 mg/mL
S4015 Cyclamic acid 36 mg/mL 36 mg/mL 36 mg/mL
S7209 GSK650394 <1 mg/mL 76 mg/mL <1 mg/mL
S1730 Indapamide <1 mg/mL 73 mg/mL 73 mg/mL
S7363 BRD7552 <1 mg/mL 100 mg/mL 100 mg/mL
S4115 Hydroxypropyl Cellulose <1 mg/mL 4 mg/mL <1 mg/mL
S7976 SBC-115076 <1 mg/mL 33 mg/mL <1 mg/mL
S2052 Oxytetracycline Dihydrate <1 mg/mL 5 mg/mL <1 mg/mL
S2053 Cytidine 49 mg/mL 49 mg/mL <1 mg/mL
S4128 Troxipide <1 mg/mL 18 mg/mL 3 mg/mL
S4134 Sevelamer Carbonate <1 mg/mL 0.05 mg/mL <1 mg/mL
S7928 DASA-58 <1 mg/mL 91 mg/mL <1 mg/mL
S2008 Taurine 20 mg/mL <1 mg/mL <1 mg/mL
S4137 Eprazinone 2HCl 18 mg/mL 1 mg/mL <1 mg/mL
S2060 Bromhexine HCl <1 mg/mL 6 mg/mL 5 mg/mL
S4138 Dropropizine 11 mg/mL 47 mg/mL 47 mg/mL
S7370 4E1RCat <1 mg/mL 96 mg/mL <1 mg/mL
S2252 (+)-Usniacin <1 mg/mL 4 mg/mL <1 mg/mL
S2253 3-Indolebutyric acid (IBA) <1 mg/mL 41 mg/mL 41 mg/mL
S2424 Hypoxanthine <1 mg/mL 0.4 mg/mL <1 mg/mL
S2374 5-hydroxytryptophan (5-HTP) 4 mg/mL 44 mg/mL <1 mg/mL
S2442 Inosine 47 mg/mL 53 mg/mL <1 mg/mL
S2256 4-Methylumbelliferone (4-MU) <1 mg/mL 35 mg/mL 35 mg/mL
S2258 Esculin 2 mg/mL 68 mg/mL 13 mg/mL
S3071 Vanillin <1 mg/mL 30 mg/mL 30 mg/mL
S4040 Norethindrone <1 mg/mL 60 mg/mL 5 mg/mL
S2260 Amygdalin <1 mg/mL 91 mg/mL <1 mg/mL
S2379 Dioscin <1 mg/mL 100 mg/mL 22 mg/mL
S7771 STF-083010 <1 mg/mL 63 mg/mL <1 mg/mL
S4153 D-Phenylalanine 1 mg/mL <1 mg/mL <1 mg/mL
S7635 Lomitapide <1 mg/mL 100 mg/mL 100 mg/mL
S2383 Gastrodin <1 mg/mL 50 mg/mL <1 mg/mL
S4154 Cholesterol <1 mg/mL 0.03 mg/mL <1 mg/mL
S2384 Hematoxylin 61 mg/mL 61 mg/mL 61 mg/mL
S8128 BAY 41-2272 <1 mg/mL 35 mg/mL 4 mg/mL
S2267 Azomycin <1 mg/mL 22 mg/mL <1 mg/mL
S2387 Lappaconite HBr <1 mg/mL 28 mg/mL <1 mg/mL
S2883 4-Aminohippuric Acid 3 mg/mL 39 mg/mL 2 mg/mL
S2884 Acesulfame Potassium 40 mg/mL 40 mg/mL <1 mg/mL
S7594 Abscisic Acid (Dormin) <1 mg/mL 52 mg/mL 52 mg/mL
S8135 Riociguat (BAY 63-2521) <1 mg/mL 84 mg/mL <1 mg/mL
S2270 Bergenin <1 mg/mL 66 mg/mL <1 mg/mL
S4161 Benzoic Acid <1 mg/mL 24 mg/mL 24 mg/mL
S2273 β-Sitosterol <1 mg/mL <1 mg/mL <1 mg/mL
S2392 Sesamin <1 mg/mL 70 mg/mL <1 mg/mL
S2276 Bilobalide <1 mg/mL 65 mg/mL 65 mg/mL
S2277 Caffeic Acid <1 mg/mL 36 mg/mL <1 mg/mL
S4047 Bisacodyl <1 mg/mL 72 mg/mL <1 mg/mL
S2280 Chlorogenic Acid 18 mg/mL 71 mg/mL 71 mg/mL
S4048 Carbimazole <1 mg/mL 38 mg/mL 15 mg/mL
S2281 Chrysin <1 mg/mL 51 mg/mL <1 mg/mL
S2422 Ipriflavone (Osteofix) <1 mg/mL 56 mg/mL 2 mg/mL
S4166 Chlorpropamide <1 mg/mL 55 mg/mL 55 mg/mL
S7213 Thiamet G 50 mg/mL 50 mg/mL 12 mg/mL
S7633 Lomitapide Mesylate <1 mg/mL 100 mg/mL 100 mg/mL
S2290 Dihydroartemisinin (DHA) <1 mg/mL 56 mg/mL 11 mg/mL
S7763 D-Luciferin <1 mg/mL 56 mg/mL 1 mg/mL
S2292 Diosmin <1 mg/mL 6 mg/mL <1 mg/mL
S4173 1-Hexadecanol 68 mg/mL 68 mg/mL 68 mg/mL
S1974 Meglumine 39 mg/mL 39 mg/mL <1 mg/mL
S4174 Sodium Gluconate 44 mg/mL <1 mg/mL <1 mg/mL
S2396 Salidroside 60 mg/mL 60 mg/mL 4 mg/mL
S4057 Methyclothiazide <1 mg/mL 72 mg/mL 4 mg/mL
S4177 Uracil <1 mg/mL 22 mg/mL 22 mg/mL
S2397 Palmatine chloride 5 mg/mL 77 mg/mL 14 mg/mL
S2299 Formononetin <1 mg/mL 54 mg/mL <1 mg/mL
S2398 Coenzyme Q10 (CoQ10) <1 mg/mL <1 mg/mL 1 mg/mL
S2300 Ferulic Acid <1 mg/mL 39 mg/mL 39 mg/mL
S2402 Cyclovirobuxin D <1 mg/mL <1 mg/mL 20 mg/mL
S2304 Gramine <1 mg/mL 35 mg/mL 35 mg/mL
S7447 ZLN005 <1 mg/mL 37 mg/mL 2 mg/mL
S2306 Gynostemma Extract <1 mg/mL 189 mg/mL 189 mg/mL
S4185 Tiratricol <1 mg/mL 100 mg/mL 100 mg/mL
S7443 AP-III-a4 (ENOblock) 9 mg/mL 100 mg/mL 100 mg/mL
S2309 Hesperidin <1 mg/mL 100 mg/mL <1 mg/mL
S2404 Isoliquiritigenin <1 mg/mL 12 mg/mL 26 mg/mL
S4186 Domiphen Bromide 83 mg/mL 83 mg/mL 83 mg/mL
S2405 Sophocarpine 6 mg/mL 49 mg/mL 49 mg/mL
S2311 Hyodeoxycholic acid (HDCA) <1 mg/mL 78 mg/mL 78 mg/mL
S4189 Cyclandelate <1 mg/mL 55 mg/mL 55 mg/mL
S4190 Cinchophen <1 mg/mL 50 mg/mL 5 mg/mL
S4070 Guanidine HCl 19 mg/mL 19 mg/mL 6 mg/mL
S4077 Mequinol 25 mg/mL 25 mg/mL 25 mg/mL
S7451 FPH1 (BRD-6125) <1 mg/mL 78 mg/mL <1 mg/mL
S7929 BEC HCl 45 mg/mL 45、 mg/mL 45 mg/mL
S4263 Efaproxiral Sodium 73 mg/mL 73 mg/mL 73 mg/mL
S7339 AZD3965 <1 mg/mL 100 mg/mL 100 mg/mL
S4264 Etofibrate <1 mg/mL 73 mg/mL 73 mg/mL
S4265 Nicaraven 57 mg/mL 57 mg/mL 57 mg/mL
S7517 AZD7545 <1 mg/mL 95 mg/mL 95 mg/mL
S2021 Chlormezanone <1 mg/mL 55 mg/mL 26 mg/mL
S4194 Azaguanine-8 <1 mg/mL 6 mg/mL <1 mg/mL
S2316 Kinetin <1 mg/mL 8 mg/mL <1 mg/mL
S2317 L-(+)-Rhamnose Monohydrate 36 mg/mL 36 mg/mL 36 mg/mL
S7453 MSDC-0160 <1 mg/mL 0.01 mg/mL <1 mg/mL
S7383 (-)-p-Bromotetramisole Oxalate 30 mg/mL 74 mg/mL <1 mg/mL
S4092 Pramoxine HCl 66 mg/mL 66 mg/mL 66 mg/mL
S4204 Isosorbide 29 mg/mL 29 mg/mL 29 mg/mL
S2124 Xylose 30 mg/mL 30 mg/mL <1 mg/mL
S4205 Dibenzothiophene <1 mg/mL 37 mg/mL 1 mg/mL
S8199 LTX-315 100 mg/mL -1 mg/mL -1 mg/mL
S2323 Methyl-Hesperidin 100 mg/mL 100 mg/mL <1 mg/mL
S2538 Acetanilide <1 mg/mL 27 mg/mL 27 mg/mL
S4206 Cysteamine HCl 23 mg/mL 23 mg/mL 23 mg/mL
S4208 Chromocarb <1 mg/mL 38 mg/mL <1 mg/mL
S7606 RBC8 <1 mg/mL 84 mg/mL <1 mg/mL
S7534 BAPTA-AM <1 mg/mL 20 mg/mL <1 mg/mL
S2609 Inulin 104 mg/mL 10 mg/mL <1 mg/mL
S1904 Avobenzone <1 mg/mL 62 mg/mL 9 mg/mL
S4214 Sucralose 80 mg/mL 80 mg/mL <1 mg/mL
S2324 Sodium Monensin <1 mg/mL <1 mg/mL 100 mg/mL
S1825 Erdosteine <1 mg/mL 50 mg/mL 10 mg/mL
S4101 Voglibose 74 mg/mL 74 mg/mL <1 mg/mL
S7446 L-Mimosine <1 mg/mL 0.01 mg/mL <1 mg/mL
S2325 Morin Hydrate <1 mg/mL 64 mg/mL 2 mg/mL
S7539 PTC-209 HBr <1 mg/mL 100 mg/mL <1 mg/mL
S2439 Guanosine <1 mg/mL 56 mg/mL <1 mg/mL
S4104 Diminazene Aceturate 100 mg/mL 19 mg/mL <1 mg/mL
S8196 ML264 <1 mg/mL 76 mg/mL <1 mg/mL
S7852 Eliglustat Tartrate <1 mg/mL 80 mg/mL 80 mg/mL
S2331 Neohesperidin Dihydrochalcone (Nhdc) <1 mg/mL 100 mg/mL 100 mg/mL
S4108 Clodronate Disodium 72 mg/mL <1 mg/mL <1 mg/mL
S2335 Oridonin <1 mg/mL 72 mg/mL 28 mg/mL
S2336 Orotic acid (6-Carboxyuracil) <1 mg/mL 2 mg/mL <1 mg/mL
S2337 Osthole <1 mg/mL 49 mg/mL 49 mg/mL
S2338 Oxymatrine 53 mg/mL 53 mg/mL 53 mg/mL
S4224 Erythritol 24 mg/mL 24 mg/mL <1 mg/mL
S7452 FPH2 (BRD-9424) <1 mg/mL 70 mg/mL <1 mg/mL
S3100 2-Thiouracil <1 mg/mL 26 mg/mL <1 mg/mL
S3102 Creatinine 23 mg/mL <1 mg/mL <1 mg/mL
S2347 Quercetin Dihydrate <1 mg/mL 67 mg/mL 21 mg/mL
S4508 2,2,2-Tribromoethanol 56 mg/mL 56 mg/mL 56 mg/mL
S4233 Zoxazolamine <1 mg/mL 34 mg/mL 34 mg/mL
S4510 4-Aminobenzoic acid <1 mg/mL 27 mg/mL 27 mg/mL
S3106 Pidotimod 10 mg/mL 49 mg/mL <1 mg/mL
S3104 Moguisteine <1 mg/mL 68 mg/mL 68 mg/mL
S2066 Moxonidine <1 mg/mL 24 mg/mL 2 mg/mL
S4519 Citric acid trilithium salt tetrahydrate 56 mg/mL 56 mg/mL <1 mg/mL
S4530 i-Inositol 36 mg/mL 36 mg/mL <1 mg/mL
S2074 Mecarbinate <1 mg/mL 47 mg/mL <1 mg/mL
S3138 Methylthiouracil <1 mg/mL 28 mg/mL <1 mg/mL
S4532 Iopamidol 100 mg/mL 100 mg/mL <1 mg/mL
S2916 ML161 <1 mg/mL 72 mg/mL <1 mg/mL
S7498 DDR1-IN-1 <1 mg/mL 100 mg/mL 4 mg/mL
S3190 N6-methyladenosine (m6A) 14 mg/mL 47 mg/mL 2 mg/mL
S7548 Rilmenidine Phosphate 55 mg/mL 1 mg/mL <1 mg/mL
S2354 Sclareol <1 mg/mL 61 mg/mL 24 mg/mL
S2355 Sclareolide <1 mg/mL 50 mg/mL 50 mg/mL
S4509 4-Aminoantipyrine 40 mg/mL 40 mg/mL 40 mg/mL
S2356 Shikimic Acid 35 mg/mL 35 mg/mL <1 mg/mL
S2357 Silibinin <1 mg/mL 96 mg/mL <1 mg/mL
S1900 Talc <1 mg/mL 0.1 mg/mL <1 mg/mL
S2358 Silymarin <1 mg/mL 96 mg/mL 1 mg/mL
S2359 Sinomenine 65 mg/mL 65 mg/mL 7 mg/mL
S7814 AI-10-49 <1 mg/mL 100 mg/mL 100 mg/mL
S7777 Coelenterazine <1 mg/mL 84 mg/mL 1 mg/mL
S2036 Aspartame 4 mg/mL 33 mg/mL <1 mg/mL
S7685 SecinH3 <1 mg/mL 92 mg/mL 1 mg/mL
S2370 Ursolic Acid <1 mg/mL 91 mg/mL <1 mg/mL
S2371 Vanillylacetone 10 mg/mL 38 mg/mL 38 mg/mL
S2372 Xanthone <1 mg/mL 39 mg/mL 1 mg/mL
S7608 UM171 <1 mg/mL 45 mg/mL <1 mg/mL
S7873 Disodium (R)-2-Hydroxyglutarate 38 mg/mL <1 mg/mL <1 mg/mL
Catalog No. Information Product Use Citations Product Validations
S1097

BTZ043 Racemate

BTZ043 racemate is a decaprenylphosphoryl-β-D-ribose 2'-epimerase (DprE1) inhibitor acting as a new antimycobacterial agent that kill Mycobacterium tuberculosis.

S1591

Bestatin

Bestatin is a potent aminopeptidase-B and leukotriene (LT) A4 hydrolase inhibitor, used in the treatment of acute myelocytic leukemia.

S1601

Reserpine

Reserpine is an inhibitor of multidrug efflux pumps, used as an antipsychotic and antihypertensive drug.

S1428

Risedronate Sodium

Risedronate Sodium, a nitrogen-containing bisphosphonate, inhibits osteoclast-mediated bone resorption and modulates bone metabolism, used in the treatment of osteoporosis.

S1271

Acarbose

Acarbose is an inhibitor of intestinal alpha-glucosidase, used to treat type 2 diabetes mellitus.

S1624

Alendronate sodium trihydrate

Alendronate sodium trihydrate, a nitrogen-containing bisphosphonate, is a potent inhibitor of bone resorption used for the treatment and prevention of osteoporosis.

S1988

Propylthiouracil

Propylthiouracil is a thyroperoxidase and 5'-deiodinase inhibitor, used to treat hyperthyroidism.

S1698

Torsemide

Torsemide is a pyridyl sulfonylurea with a chemical structure between that of traditional loop diuretics and Cl- channel blockers, used to treat hypertension.

S7372

PTC-209

PTC-209 is a potent and selective BMI-1 inhibitor with IC50 of 0.5 μM in HEK293T cell line, and results in irreversible reduction of cancer-initiating cells (CICs).

S7270

SRPIN340

SRPIN340 is a selective SRPK inhibitor with Ki of 0.89 μM for SRPK1, showing no significant inhibitory activity against more than 140 other kinases..

S7272

4μ8C

4μ8C is a potent and selective IRE1 Rnase inhibitor with IC50 of 76 nM.

S2129

Fudosteine

Fudosteine is a cysteine derivative and a MUC5AC mucin hypersecretion inhibitor, used as a muco-active agent with indications for chronic respiratory diseases.

S8077

RI-1

RI-1 is a RAD51 inhibitor with IC50 ranging from 5 to 30 μM.

S2610

Lonidamine

Lonidamine is an orally administered small molecule hexokinase inactivator.

S2901

CCG 50014

CCG 50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM.

S2035

Epalrestat

Epalrestat is an aldose reductase inhibitor with IC50 of 72 nM.

S3199

Reboxetine mesylate

Reboxetine is a norepinephrine reuptake inhibitor with Ki of 8.2 nM.

S7369

4EGI-1

4EGI-1 is a competitive eIF4E/eIF4G interaction inhibitor by binding to eIF4E with KD of 25 μM.

S1875

Tranexamic Acid

Tranexamic Acid is an antifibrinolytic for blocking lysine-binding sites of plasmin and elastase-derived plasminogen fragments with IC50 of 5 mM.

S4020

Sodium Picosulfate

Sodium Picosulfate inhibits absorption of water and electrolytes, and increases their secretion.

S2032

Rebamipide

Rebamipide is a cholecystokinin type 1 (CCK1) receptor inhibitor for inhibiting [125I]BH-CCK-8S with IC50 of 37.7 μM.

S7382

Phosphoramidon Disodium Salt

Phosphoramidon Disodium Salt is a metalloendopeptidase inhibitor, widely used as a biochemical tool.

S7589

N6022

N6022 is a selective, and reversible inhibitor of S-nitrosoglutathione reductase (GSNOR) with IC50 of 8 nM and Ki of 2.5 nM. Phase 1/2.

S7922

Tiplaxtinin (PAI-039)

Tiplaxtinin(PAI-039) is an orally efficacious and selective plasminogen activator inhibitor-1 (PAI-1) inhibitor with IC50 of 2.7 μM.

S4299

Dicoumarol

Dicoumarol is a competitive NADH quinone oxidoreductase (NQO1) inhibitor,and used as an anticoagulant by interfering with the metabolism of vitamin K.

S4017

Allylthiourea

Allylthiourea is a metabolic inhibitor that selective inhibits ammonia oxidation.

S2830

Clindamycin

Clindamycin inhibits protein synthesis by acting on the 50S ribosomal, used for the treatment of bacterial infections.

S7209

GSK650394

GSK650394 is a serum- and glucocorticoid-regulated kinase-1 inhibitor with IC50 of 62 nM and 103 nM for SGK1 and SGK2, respectively.

S7370

4E1RCat

4E1RCat is a dual inhibitor of eIF4E:eIF4G and eIF4E:4E-BP1 interaction, and inhibits the binding of eIF4G to eIF4E with IC50 of 3.2 μM.

S2256

4-Methylumbelliferone (4-MU)

4-Methylumbelliferone is a hyaluronic acid (HA) synthesis inhibitor with an IC50 of 0.4 mM.

S7771

STF-083010

STF-083010 is a specific IRE1α endonuclease inhibitor without affecting its kinase activity.

S4153

D-Phenylalanine

D-Phenylalanine, a carboxypeptidase A, endorphinase and enkephalinase inhibitor, enhances endorphin production and diminishes pain.

S7635

Lomitapide

Lomitapide is a potent microsomal triglyceride transfer protein (MTP) inhibitor, used in the treatment of familial hypercholesterolemia.

S2422

Ipriflavone (Osteofix)

Ipriflavone (7-Isopropoxyisoflavon) is used to inhibit bone resorption.

S7213

Thiamet G

Thiamet G is a potent, selective O-GlcNAcase inhibitor with Kiof 21 nM, while exhibiting 37,000-fold selectivity over human lysosomal –hexosaminidase.

S7633

Lomitapide Mesylate

Lomitapide Mesylate is a potent microsomal triglyceride transfer protein (MTP) inhibitor, used in the treatment of familial hypercholesterolemia.

S7443

AP-III-a4 (ENOblock)

AP-III-a4 (ENOblock) is the first nonsubstrate analogue inhibitor of enolase with IC50 of 0.576 μM.

S2404

Isoliquiritigenin

Isoliquiritigenin, an anti-tumor flavonoid from the root of Glycyrrhiza glabra, inhibits aldose reductase with an IC50 of 320 nM.

S7929

BEC HCl

BEC HCl is a slow-binding, and competitive arginase inhibitor with Ki of 0.31 μM (pH7.5) and 0.4-0.6 μM for Arginase II and rat Arginase I, respectively.

S7339

AZD3965

AZD3965 is a potent, selective and orally available monocarboxylate transporter 1 (MCT1) inhibitor with a binding affinity of 1.6 nM, 6-fold selective over MCT2. Phase 1.

S7517

AZD7545

AZD7545 is a potent PDHK inhibitor with IC50 of 36.8 nM and 6.4 nM for PDHK1 and PDHK2, respectively. It failed to inhibit PDHK4 at higher concentrations(>10 nM), AZD7545 stimulates PDHK4 activity.

S7606

RBC8

RBC8 is a selective inhibitor of the GTPases RalA and RalB by inhibiting the binding of Ral to its effector RALBP1, no inhibition on the GTPases Ras and RhoA.

S7539

PTC-209 HBr

PTC-209 HBr is the hydrobromide salt of PTC-209, which is a potent and selective BMI-1 inhibitor with IC50 of 0.5 μM, and results in irreversible reduction of cancer-initiating cells (CICs).

S8196

ML264

ML264, a selectively inhibitor of kruppel-like factor 5 (KLF5),potently Inhibits Growth of Colorectal Cancer.

S7852

Eliglustat Tartrate

Eliglustat (Tartrate) inhibits glucosylceramide synthase(GCS),thus reducing the load of glucosylceramide influx into the lysosome.

S4108

Clodronate Disodium

Clodronate Disodium, a bisphosphonate, is a potent antiosteolytic agent which inhibits bone resorption.

S4233

Zoxazolamine

Zoxazolamine is a centrally acting myorelaxant, which is formerly used as an antispasmodic and uricosuric.

S2916

ML161

ML-161 is an allosteric inhibitor of PAR1 with IC50 of 0.26 μM.

S2063

Pamidronate

Pamidronate is bisphosphonate which binds to the hydroxyapatite in bone and act as an inhibitor of the resorption of bone for the treatment of osteitis deformans and postmenopausal osteoporosis.

S7498

DDR1-IN-1

DDR1-IN-1 is a potent and selective discoidin domain receptor 1 (DDR1) receptor tyrosine kinase inhibitor with IC50 of 105 nM, about 3-fold selectivity over DDR2.

S7814

AI-10-49

AI-10-49 is a selective inhibitor of the binding of CBFβ-SMMHC to RUNX1 with IC50 of 260 nM.

S7685

SecinH3

SecinH3 is a selective cytohesin inhibitor with IC50 of 2.4 μM, 5.4 μM, 5.4 μM, 5.6 μM, 5.6 μM, and 65 μM for hCyh2, hCyh1, mCyh3, hCyh3, drosophila steppke, and yGea2-S7, respectively.

S7873

Disodium (R)-2-Hydroxyglutarate

Disodium (R)-2-Hydroxyglutarate is a competitive inhibitor of α-ketoglutarate-dependent dioxygenases with Ki of 0.628 mM.

S7594

Abscisic Acid (Dormin)

Abscisic Acid is a plant hormone, which is involved in many plant developmental processes, modulates ion homeostasis and metabolism, and inhibits germination and seedling growth.

S6002

NXY-059 (Disufenton sodium)

NXY-059 is a novel nitrone, shows efficacious neuroprotective effects. Phase 3.

S1751

Gadodiamide Hydrate

Gadodiamide Hydrate, a nonionic Gd3+ chelate, is frequently injected i.v. into magnetic resonance imaging (MRI) to enhance contrast.

S1236

Leucovorin Calcium Pentahydrate

Leucovorin is a derivative of folic acid, which can be used to increase levels of folic acid under conditions favoring folic acid inhibition.

S4728New

3,3'-Diindolylmethane

3,3'-Diindolylmethane(DIM) is a major digestive product of indole-3-carbinol, a potential anticancer component of cruciferous vegetables.

S1627

Nitazoxanide

Nitazoxanide is a synthetic nitrothiazolyl-salicylamide derivative and an antiprotozoal agent. (IC50 for canine influenza virus ranges from 0.17 to 0.21 μM)

S1137

Malotilate

Malotilate, diisopropyl 1,3-dithiol-2-ylidenemalonate, is a drug used for the treatment of liver cirrhosis.

S1934

Nystatin (Fungicidin)

Nystatin, which belongs to the polyene group of antimycotics, is frequently used as a topical agent in the treatment of oro-pharyngeal candidosis.

S2757

TH-302

TH-302 is selective hypoxia-activated prodrug targeting hypoxic regions of solid tumors with IC50 of 19 nM, demonstrates 270-fold enhanced cytotoxicity under hypoxia versus their potency under aerobic conditions, stable to cytochrome P450 metabolism.

S1311

Pamidronate Disodium

Pamidronate Disodium is a nitrogen containing bisphosphonate, used to prevent osteoporosis.

S2553

5-Aminolevulinic acid HCl

5-Aminolevulinic Acid HCl is an intermediate in the porphyrin synthesis pathway, used as a photosensitizing agent and a antineoplastic agent.

S1201

Dimesna

Dimesna is an uroprotective agent used to decrease urotoxicity.

S1732

Mitotane

Mitotane, is an antineoplastic medication used in the treatment of adrenocortical carcinoma.

S2417

20-Hydroxyecdysone

20-Hydroxyecdysone (Ecdysterone, 20E) is a naturally occurring ecdysteroid hormone which controls the ecdysis (moulting) and metamorphosis of arthropods.

S1326

Edaravone

Edaravone is a novel potent free radical scavenger that has been clinically used to reduce the neuronal damage following ischemic stroke.

S1897

Potassium Iodide

Potassium Iodide is used to treat overactive thyroid and to protect the thyroid gland from the effects of radiation from inhaled or swallowed radioactive iodine.

S2586

Dimethyl Fumarate

Dimethyl fumarate (DMF)is the methyl ester of fumaric acid, used to treat people with relapsing forms of multiple sclerosis.

S1740

Guaifenesin

Guaifenesin is an expectorant used to relieve chest congestion.

S4067

Deferiprone

Deferiprone is a chelating agent with an affinity for ferric ion (iron III),binds with ferric ions to form neutral 3:1 (deferiprone:iron) complexes that are stable over a wide range of pH values.

S1287

Bumetanide

Bumetanide (Bumex) is a loop diuretic of the sulfamyl category to treat heart failure.

S7217

OAC1

OAC1 (Oct4-activating compound 1) can enhance the efficiency of reprogramming.

S1849

Daidzein

Daidzein is a natural isoflavone phytoestrogen found in Leguminosae, used as a component of foods and dietary supplements.

S2408

Cephalomannine

Cephalomannine is an active anti-cancer agent obtained from Taxus yunnanensis and has an antineoplastic effect on tumors found in mice.

S4059

Sodium Nitroprusside Dihydrate

Sodium Nitroprusside Dihydrate is a potent vasodilator working through releasing NO spontaneously in blood.

S7450

FH1(BRD-K4477)

FH1 (BRD-K4477) is a small molecule, which promotes differentiation of iPS-derived hepatocytes.

S1749

L-Glutamine

L-Glutamine (Gln) is one of the 20 amino acids encoded by the standard genetic code and also a major respiratory fuel and substrate for nucleic acid synthesis in mammalian intestinal cells.

S1917

Crystal Violet

Crystal violet is a triarylmethane dye.

S1874

Risedronate

Risedronate is a bisphosphonate used to strengthen bone, treat or prevent osteoporosis, and treat Paget's disease of bone.

S2412

Genipin

Genipin is an active aglycone derived from an iridoid glycoside called geniposide, which is found in the fruit of Gardenia jasminoides Ellis.

S2410

Paeoniflorin

Paeoniflorin is a herbal constituent extracted from the root of Paeonia albiflora Pall.

S1609

Methimazole

Methimazole is an antithyroid medicine.

S2594

Pramiracetam

Pramiracetam is a more potent nootropic drug derived from piracetam.

S2388

L-carnitine

L-carnitine is constituent of striated muscle and liver. It is used therapeutically to stimulate gastric and pancreatic secretions and in the treatment of hyperlipoproteinemias.

S1643

Ursodiol

Ursodiol reduces cholesterol absorption and is used to dissolve (cholesterol) gallstones. (IC50=0.22 μM)

S1647

Adenosine

Adenosine is a nucleoside composed of a molecule of adenine attached to a ribose sugar molecule (ribofuranose) moiety via a β-N9-glycosidic bond.

S1671

(6-)ε-​Aminocaproic acid

(6-)ε-​Aminocaproic acid is a derivative and analogue of the amino acid lysine.

S1853

Penicillamine

Penicillamine is used as an antirheumatic and as a chelating agent in Wilson’s disease.

S2536

Miconazole

Miconazole (Monistat) is an imidazole antifungal agent.

S2724

Heparin sodium

Heparin sodium is a sodium salt of heparin which is a naturally-occurring anticoagulant used for anticoagulation for cardiovascular disease.

S1806

Acipimox

Acipimox is a niacin derivative used as a hypolipidemic agent.

S4217

Liothyronine Sodium

Liothyronine Sodium is the most potent form of thyroid hormone acting on the body to increase the basal metabolic rate, affect protein synthesis.

S1985

ATP

ATP Disodium is a disodium salt form of adenosine-triphosphate that is used in cells as a coenzyme.

S3148

Ibandronate sodium

Ibandronate is a highly potent nitrogen-containing bisphosphonate used for the treatment of osteoporosis.

S3150

Articaine HCl

Articaine is a dental local anesthetic which contains an additional ester group that is metabolized by estearases in blood and tissue.

S3000

Carbazochrome sodium sulfonate (AC-17)

Carbazochrome sodium sulfonate (AC-17) is an antihemorrhagic for use in the treatment of hemorrhoids.

S2599

L-Thyroxine

L-Thyroxine is a synthetic form of thyroxine and a hormone replacement drug.

S1610

Metolazone

Metolazone is a diuretic that primarily used to treat congestive heart failure and high blood pressure.

S4129

Sevelamer HCl

Sevelamer HCl is a phosphate binding drug used to treat hyperphosphatemia via binding to dietary phosphate and prevents its absorption.

S2381

D-Mannitol

D-Mannitol is an osmotic diuretic agent and a weak renal vasodilator.

S2393

Sorbitol

Sorbitol is a sugar alcohol and a sugar substitute.

S1641

Chlorothiazide

Chlorothiazide is a diuretic and antihypertensive. (IC50=3.8 mM)

S2293

DL-Carnitine HCl

DL-Carnitine HCl is a quaternary ammonium compound biosynthesized from the amino acids lysine and methionine.

S2305

Grape Seed Extract

Grape Seed Extract are industrial derivatives from whole grape seeds that have a great concentration of vitamin E, flavonoids, linoleic acid, and OPCs.

S1715

Glipizide

Glipizide is used to treat high blood sugar levels caused by a type of diabetes mellitus called type 2 diabetes.

S4095

Difluprednate

Difluprednate (difluoroprednisolone butyrate acetate, or DFBA) is a synthetic difluorinated prednisolone derivative, it is originally developed for dermatologic applications.

S1928

Alibendol

Alibendol is an antispasmodic,choleretic, and cholekinetic.

S1735

Mesna

Mesna, a sulfhydryl compound that is used to reduce the incidence of hemorrhagic cystitis associated with certain chemotherapeutic agents.

S2411

Geniposide

Geniposide is an iridoid glycoside isolated from the fruit of Gardenia jasminoides Ellis.

S2409

10-Deacetylbaccatin-III

10-Deacetylbaccatin-III is an antineoplastic agent and an anti-cancer intermediate.

S3209

Amidopyrine

Amidopyrine is a white crystalline substance used as an analgesic and antipyretic.

S1708

Hydrochlorothiazide

Hydrochlorothiazide is a first line diuretic compound of the thiazide class.

S2596

Clindamycin palmitate HCl

Clindamycin palmitate HCl is a water soluble hydrochloride salt of the ester of clindamycin and palmitic acid and a lincosamide antibiotic.

S4298

Amifostine

Amifostine is the first approved radioprotective drug, used to decrease the risk of kidney problems caused by treatment with cisplatin.

S7909

Dp44mT

Dp44mT is a potent iron chelator, which shows selective antitumor activity.

S7913

MCB-613

MCB-613 is a potent steroid receptor coactivator (SRC) stimulator.

S7914

Isoxazole 9 (ISX-9)

Isoxazole 9 (Isx-9) is a synthetic promotor of adult neurogenesis by triggering neuronal differentiation of adult neural stem/precursor cells (NSPCs).

S2589

Miglitol

Miglitol is an oral anti-diabetic drug.

S2518

NAD+

NAD+ is a coenzyme composed of ribosylnicotinamide 5'-diphosphate coupled to adenosine 5'-phosphate by pyrophosphate linkage.

S4015

Cyclamic acid

Cyclamic acid in the form of its sodium or calcium salt is one of the most widely used artificial sweeteners.

S1730

Indapamide

Indapamide is a non-thiazide sulphonamide diuretic compound, generally used in the treatment of hypertension, as well as decompensated cardiac failure.

S7363

BRD7552

BRD7552 is an inducer of transcription factor PDX1, which increases insulin expression.

S4115

Hydroxypropyl Cellulose

Hydroxypropyl cellulose (HPC) is a derivative of cellulose with both water solubility and organic solubility, it is used as food additive and sieving matrix for DNA separations.

S2052

Oxytetracycline Dihydrate

Oxytetracycline Dihydrate is a prescription antibiotic, interfering with the ability of bacteria to produce essential proteins.

S2053

Cytidine

Cytidine is a nucleoside molecule that is formed when cytosine is attached to a ribose ring, cytidine is a component of RNA.

S4128

Troxipide

Troxipide is a novel systemic non-antisecretory gastric cytoprotective agent with anti-ulcer, anti-inflammatory and mucus secreting properties irrespective of pH of stomach or duodenum.

S4134

Sevelamer Carbonate

Sevelamer carbonate is a non-absorbed phosphate binding crosslinked polymer, with the same polymeric structure as sevelamer hydrochloride, in which carbonate replaces chloride as the counterion.

S2008

Taurine

Taurine is an organic acid widely distributed in animal tissues.

S4137

Eprazinone 2HCl

Eprazinone is a mucolytic.

S2060

Bromhexine HCl

Bromhexine HCl is a medication prescribed for coughs which works by dissolving hard phlegm.

S4138

Dropropizine

Dropropizine is a racemic non-opiate antitussive agent, it is used as a cough suppressant.

S2252

(+)-Usniacin

(+)-Usniacin is a naturally occurring dibenzofuran derivative found in several lichen species.

S3068

Guanosine Hydrate

Guanosine hydrate plays important roles in various biochemical processes such as synthesis of nucleic acids and proteins, photosynthesis, muscle contraction and intracellular signal transduction (cGMP).

S2253

3-Indolebutyric acid (IBA)

3-Indolebutyric acid(IBA) is a plant hormone in the auxin family and is an ingredient in many commercial plant rooting horticultural products.

S2424

Hypoxanthine

Hypoxanthine, a naturally occurring purine derivative, an intermediate product of uric acid synthesis, formed from adenylic acid and itself a precursor of xanthine.

S2374

5-hydroxytryptophan (5-HTP)

5-Hydroxytryptophan (5-HTP), also known as oxitriptan (INN), is a naturally occurring amino acid and chemical precursor for the treatment of depression.

S2442

Inosine

Inosine is a nucleoside that is formed when hypoxanthine is attached to a ribose ring via a β-N9-glycosidic bond.

S2258

Esculin

Esculin is a glucoside found in horse chestnuts.

S3071

Vanillin

Vanillin, 4-hydroxy-3-methoxybenzaldehyde, is a food additive.

S4040

Norethindrone

Norethindrone is a synthetic progestin, which mimic the actions of the endogenous ovarian hormone progesterone.

S2260

Amygdalin

Amygdalin is a glycoside initially isolated from the seeds of the tree Prunus dulcis, also known as bitter almonds.

S2379

Dioscin

Dioscin is a saponin extracted and isolated from Polygonatum Zanlanscianense Pamp, showing antitumor activities.

S2383

Gastrodin

Gastrodin, an anti-inflammatory polyphenol extracted from Chinese natural herbal Gastrodia elata Blume., benefits neurodegenerative diseases.

S4154

Cholesterol

Cholesterol is the principal sterol of all higher animals required to build and maintain membranes.

S2384

Hematoxylin

Hematoxylin (Hydroxybrazilin) is a compound that forms strongly colored complexes with certain metal ions, notably Fe(III) and Al(III) salts and a kind of stain in histology.

S8128

BAY 41-2272

BAY 41-2272 is a direct and NO-independent soluble guanylate cyclase (sGC) stimulator.

S2267

Azomycin

Azomycin is an antimicrobial antibiotic produced by a strain of Nocardia mesenterica.

S2387

Lappaconite HBr

Lappaconite Hydrobromide is a kind of alkaloid extracted from Aconitum sinomontanum Nakai and has anti-inflammatory effects.

S2883

4-Aminohippuric Acid

4-Aminohippuric acid is a typical substrate of organic anion transport systems.

S2884

Acesulfame Potassium

Acesulfame potassium is a non-nutritive sweetener.

S8135

Riociguat (BAY 63-2521)

Riociguat (BAY 63-2521) is an oral soluble guanylate cyclase (GC) stimulator, used in the treatment of ipulmonary hypertension.

S2270

Bergenin

Bergenin is trihydroxybenzoic acid glycoside and the C-glycoside of 4-O-methyl gallic acid.

S4161

Benzoic Acid

Benzoic acid is a colorless crystalline solid and a simple aromatic carboxylic acid, used as a food preservative.

S2273

β-Sitosterol

β-Sitosterol is one of several phytosterols (plant sterols) with chemical structures similar to that of cholesterol.

S2392

Sesamin

Sesamin, a lignan isolated from the bark of Fagara plants and from sesame oil, exhibits various health benefits.

S2276

Bilobalide

Bilobalide is a biologically active terpenic trilactone present in Ginkgo biloba.

S2277

Caffeic Acid

Caffeic acid is a hydroxycinnamic acid, a naturally occurring organic compound.

S4047

Bisacodyl

Bisacodyl (INN) is a stimulant laxative drug that works directly on the colon to produce a bowel movement.

S2280

Chlorogenic Acid

Chlorogenic acid is a hydroxycinnamic acid and a member of a family of naturally occurring organic compounds.

S4048

Carbimazole

Carbimazole is an imidazole antithyroid agent.

S2281

Chrysin

Chrysin is a naturally occurring flavone chemically extracted from the blue passion flower (Passiflora caerulea).

S4166

Chlorpropamide

Chlorpropamide is a sulfonylurea class drug for type 2 diabetes mellitus.

S2290

Dihydroartemisinin (DHA)

Dihydroartemisinin (DHA) is a semi-synthetic derivative of artemisinin and isolated from the traditional Chinese herb Artemisia annua.

S7763

D-Luciferin

D-Luciferin is a popular bioluminescent substrate of luciferase in the presence of ATP, used in luciferase-based bioluminescence imaging and cell-based high-throughput screening applications.

S2292

Diosmin

Diosmin is a semisynthetic phlebotropic agent and a member of the flavonoid family.

S4173

1-Hexadecanol

1-Hexadecanol is a fatty alcohol used to make other chemicals.

S1974

Meglumine

Meglumine is an amino sugar derived from sorbitol for THP-1 cells with IC50 of 22 μg/mL.

S4174

Sodium Gluconate

Sodium gluconate is the sodium salt of gluconic acid widely used in food and pharmaceutical industry.

S2396

Salidroside

Salidroside, a phenylpropanoid glycoside isolated from Rhodiola rosea, has been reported to have a broad spectrum of pharmacological properties.

S4057

Methyclothiazide

Methyclothiazide is a substituted benzothiadiazide, used to treat high blood pressure and fluid retention caused by various conditions including heart disease.

S4177

Uracil

Uracil is one of the four nucleobases in the nucleic acid of RNA can be used for drug delivery and as a pharmaceutical.

S2397

Palmatine chloride

Palmatine hydrochloride (Palmatine chloride (6CI,7CI); Fibrauretin) is a hydrochloride salt of palmatine which is a protoberberine alkaloid.

S2299

Formononetin

Formononetin is a phytoestrogen from the root of Astragalus membranaceus and an O-methylated isoflavone.

S2398

Coenzyme Q10 (CoQ10)

Coenzyme Q10 (ubiquinone, ubidecarenone, coenzyme Q) is a component of the electron transport chain and participates in aerobic cellular respiration.

S2300

Ferulic Acid

Ferulic Acid is a hydroxycinnamic acid and a type of organic compound found in the Ferula assafoetida L. or Ligusticum chuanxiong.

S2402

Cyclovirobuxin D

Cyclovirobuxine D is an active compound extracted from Buxus microphylla, which has been used for treating acute myocardial ischemia.

S2304

Gramine

Gramine is a naturally occurring indole alkaloid present in several plant species.

S2306

Gynostemma Extract

Gynostemma Extract is a saponins extract derived from the Gynostemma pentaphyllum.

S4185

Tiratricol

Tiratricol (also known as TRIAC or triiodothyroacetic acid) is a thyroid hormone analogue.

S2309

Hesperidin

Hesperidin is a flavanone glycoside found abundantly in citrus fruits.

S4186

Domiphen Bromide

Domiphen bromide is a quaternary ammonium antiseptic with actions as a cationic surfactant.

S2405

Sophocarpine

Sophocarpine, a major ingredient of Sophora alopecuroides, has a wide range of pharmacological effects.

S2311

Hyodeoxycholic acid (HDCA)

Hyodeoxycholic(HDCA) acid is a secondary bile acid, one of the metabolic byproducts of intestinal bacteria.

S4189

Cyclandelate

Cyclandelate is an effective inhibitor of rat hepatic acycloenzyme A: cholesterol acyltransferase (ACAT) with IC50 of 80 μM.

S4190

Cinchophen

Cinchophen is an analgesic drug that is frequently used to treat gout.

S4070

Guanidine HCl

Guanidine HCl, the crystalline compound of strong alkalinity formed by the oxidation of guanine, is a normal product of protein metabolism and a protein denaturant.

S4077

Mequinol

Mequinol (4-Methoxyphenol) is a depigmentation agent.

S7451

FPH1 (BRD-6125)

FPH1 (BRD-6125) is a small molecule, which promotes expansion of iPS-derived hepatocytes.

S4263

Efaproxiral Sodium

Efaproxiral Sodium is a synthetic allosteric modifier of hemoglobin, used for brain metastases originating from breast cancer.

S4264

Etofibrate

Etofibrate is a combination of clofibrate and niacin, used to treat hyperlipemia.

S4265

Nicaraven

Nicaraven is a hydroxyl radical scavenger with antivasospastic and neuroprotective effects.

S2021

Chlormezanone

Chlormezanone,a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.

S4194

Azaguanine-8

Azaguanine-8 is a purine analogs showing antineoplastic activity by competing with guanine in the metabolism.

S2316

Kinetin

Kinetin is a type of cytokinin, a class of plant hormone that promotes cell division.

S2317

L-(+)-Rhamnose Monohydrate

L(+)-Rhamnose (Rham) is a naturally-occurring deoxy sugar that is found primarily in plants and some bacteria.

S7453

MSDC-0160

MSDC-0160 is a prototype mTOT-modulating insulin sensitizer being studied to treat diabetes and Alzheimer's disease. Phase 2.

S4092

Pramoxine HCl

Pramoxine is a topical local anesthetic that has been shown to have antipruritic properties.

S4204

Isosorbide

Isosorbide is a heterocyclic compound that is derived from glucose, used as a diuretic.

S2124

Xylose

Xylose is a sugar first isolated from wood.

S4205

Dibenzothiophene

Dibenzothiophene (DBT) is a model compound for organic sulfur in fossil fuels.

S8199

LTX-315

LTX-315 is the oncolytic peptide that kills cancer cells through Bax/Bak-regulated mitochondrial membrane permeabilization.

S2323

Methyl-Hesperidin

Methyl Hesperidin is a flavanone glycoside (flavonoid) (C28H34O15) found abundantly in citrus fruits. Its aglycone form is called hesperetin.

S2538

Acetanilide

Acetanilide is an aniline derivative and has possess analgesic.

S4206

Cysteamine HCl

Cysteamine is an agent for the treatment of nephropathic cystinosis and an antioxidant.

S4208

Chromocarb

Chromocarb is a vasoprotectant.

S7534

BAPTA-AM

BAPTA-AM is a selective, membrane-permeable calcium chelator.

S2609

Inulin

Inulin(Inulin and sodium chloride), a starch found in the tubers and roots of many plants. Since it is hydrolyzable to fructose, it is classified as a fructosan.

S1904

Avobenzone

Avobenzone is an oil soluble ingredient used in sunscreen products to absorb the full spectrum of UVA rays and a dibenzoylmethane derivative.

S4214

Sucralose

Sucralose is an artificial and noncaloric sweetener, not broken down by the body.

S2324

Sodium Monensin

Sodium Monensin, isolated from Streptomyces cinnamonensis, is a well-known representative of naturally polyether ionophore antibiotics.

S1825

Erdosteine

Erdosteine is a mucolytic which is used in treatment of excessive viscous mucus.

S4101

Voglibose

Voglibose is an N-substituted derivative of valiolamine, excellent inhibitory activity against α-glucosidases and its action against hyperglycemia and various disorders caused by hyperglycemia.

S7446

L-Mimosine

L-Mimosine is a non-protein amino acid, and acts as an iron chelator.

S2325

Morin Hydrate

Morin hydrate(Aurantica) is a flavonoid isolated from Maclura pomifera (Osage orange), Maclura tinctoria (old fustic) and from leaves of Psidium guajava (common guava).

S2439

Guanosine

Guanosine is a purine nucleoside comprising guanine attached to a ribose (ribofuranose) ring via a β-N9-glycosidic bond.

S4104

Diminazene Aceturate

Diminazene is a di-amidine also known as 4,4-(1-Triazene–1,3–diyl)bis(benzenecarboximidamide), used as an effective trypanocidal agent.

S2331

Neohesperidin Dihydrochalcone (Nhdc)

Neohesperidin dihydrochalcone(Nhdc), sometimes abbreviated to neohesperidin DC or simply NHDC, is an artificial sweetener derived from citrus.

S2335

Oridonin

Oridonin, a diterpenoid purified from Rabdosia rubescens, is an antitumor agent.

S2336

Orotic acid (6-Carboxyuracil)

Orotic acid(6-Carboxyuracil) is a heterocyclic compound and an acid.

S2337

Osthole

Osthol is an O-methylated coumarin, which is found in the plants such as Cnidium monnieri, Angelica archangelica and Angelica pubescens.

S2338

Oxymatrine

Oxymatrine is a quinolizidine alkaloid extracted from the root of Sophora flavescens with anti-inflammatory, antifibrosis, and antitumor effects, inhibits the iNOS expression and TGF-β/Smad pathway. It is used for the treatment of viral hepatitis, cancer, viral myocarditis, gastrointestinal hemorrhage and skin diseases.

S4224

Erythritol

Erythritol is a sugar alcohol used as low-calorie sweetener.

S7452

FPH2 (BRD-9424)

FPH2 (BRD-9424) is a small molecule, which promotes differentiation of iPS-derived hepatocytes.

S3100

2-Thiouracil

2-Thiouracil is a thiolated uracil derivative that is a known antihyperthyroid agent.

S3102

Creatinine

Creatinine is a break-down product of creatine phosphate in muscle, and is usually produced at a fairly constant rate by the body.

S2347

Quercetin Dihydrate

Quercetin, a polyphenolic flavonoid found in a wide variety of plant-based foods, such as apples, onions, berries, and red wine, is utilized in many different cultures for their nervous system and anticancer effects.

S4508

2,2,2-Tribromoethanol

2,2,2-Tribromoethanol is an organic compound used to anesthetize mice.

S4510

4-Aminobenzoic acid

4-Aminobenzoic acid is an intermediate in the synthesis of tetrahydrofolic acid in many non-mammalian organisms, including bacteria and fungi.

S3106

Pidotimod

Pidotimod is an immunostimulant.

S3104

Moguisteine

Moguisteine is a novel peripheral non-narcotic antitussive drug.

S4519

Citric acid trilithium salt tetrahydrate

Citric acid trilithium salt tetrahydrate is a pharmaceutical and construction material. It is commonly used in HPLC gradient elution for quantification of amino acids.

S4530

i-Inositol

i-Inositol, also known as myo-inositol, is a chemical compound which is sugar alcohol. i-Inositol is involved in a number of biological processes including insulin signal transduction, cytoskeleton transduction and so on.

S2074

Mecarbinate

Mecarbinate is a chemical intermediate of arbidol hydrochloride.

S3138

Methylthiouracil

Methylthiouracil is an antithyroid preparation.

S4532

Iopamidol

Iopamidol is a non-ionic, water-soluble radiographic contrast agent.

S2353

Sapogenins Glycosides

Sapogenins glycosides are a mixture of triterpene and steroid saponins isolated from medicinal plants such as Aesculus hippocastanum L., Hedera helix L. and Ruscus aculeatus L., which are claimed to be effective for the treatment/prevention of venous insufficiency.

S3190

N6-methyladenosine (m6A)

N6-methyladenosine (m6A) is a base modified analog of adenosine and is found as a minor nucleoside in natural RNAs.

S2354

Sclareol

Sclareol, a labdane-type diterpene isolated from clary sage (Salvia sclarea), exerts growth inhibition and cytotoxic activity against a variety of human cancer cell lines.

S2355

Sclareolide

Sclareolide(Norambreinolide) is a sesquiterpene lactone natural product derived from various plant sources including Salvia sclarea, Salvia yosgadensis, and cigar tobacco.

S4509

4-Aminoantipyrine

4-Aminoantipyrine(Ampyrone) is a metabolite of aminopyrine with analgesic, anti-inflammatory, and antipyretic properties. It is used as a reagent for biochemical reactions producing peroxides or phenols.

S2356

Shikimic Acid

Shikimic acid(Shikimate), more commonly known as its anionic form shikimate, is an important biochemical intermediate in plants and microorganisms.

S2357

Silibinin

Silibinin, the main flavonoid extracted from the milk thistle Silybum marianum, displays hepatoprotective properties in acute and chronic liver injury.

S1900

Talc

Talc is a mineral composed of hydrated magnesium silicate with the chemical formula H2Mg3(SiO3)4 or Mg3Si4O10(OH)2.

S2358

Silymarin

Silymarin (Silybin B), a polyphenolic flavonoid extracted from the seeds of Silybum marianum or milk thistle, is used in the prevention and treatment of liver diseases and primary liver cancer.

S2359

Sinomenine

Sinomenine, a pure alkaloid extracted from the chinese medical plant Sinomenium acutum, is used for the treatment of rheumatism and arthritis.

S7777

Coelenterazine

Coelenterazine is a luminescent enzyme substrate, used for monitoring reporter genes in BRET, ELISA and HTS techniques.

S2036

Aspartame

Aspartame is an artificial, non-saccharide sweetener used as a sugar substitute in some foods and beverages.

S2370

Ursolic Acid

Ursolic acid (Malol) is a pentacyclic triterpene acid, used in cosmetics.

S2371

Vanillylacetone

Vanillylacetone is similar in chemical structure to other flavor chemicals such as vanillin and eugenol and is used as a flavor additive in spice oils and in perfumery to introduce spicy aromas.

S2372

Xanthone

Xanthone is an organic compound, which can be prepared by the heating of phenyl salicylate.

S7365

AdipoRon

AdipoRon is a novel, and orally bioavailable adiponectin receptor agonist with KD of 1.8 and 3.1 μM for AdipoR1 and AdipoR2, respectively.

S2066

Moxonidine

Moxonidine is a selective agonist at the imidazoline receptor subtype 1, used as antihypertensive agent.

S7548

Rilmenidine Phosphate

Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist, used for the treatment of hypertension.

S7608

UM171

UM171 is a potent agonist of human hematopoietic stem cell renewal, independently of AhR suppression.

S2155

LY2608204

LY2608204 activates glucokinase (GK) with EC50 of 42 nM. Phase 2.

S1511

Lactulose

Lactulose, a disaccharide composed of galactose and fructose, is a stimulator of health-promoting bacterium growth in the gastrointestinal tract, used to treat chronic constipation and hepatic encephalopathy.

S7928

DASA-58

DASA-58 is a specific and potent Pyruvate kinase M2 (PKM2) activator.

S7447

ZLN005

ZLN005 is a potent and tissue-specific PGC-1α transcriptional activator.

S3038

Fosaprepitant dimeglumine salt

Fosaprepitant is a water-soluble phosphoryl prodrug for Aprepitant which is a NK1 antagonist.

S7976

SBC-115076

SBC-115076 is a potent extracellular proprotein convertase subtilisin kexin type 9 (PCSK9) antagonist.

Catalog No. Information Product Use Citations Product Validations
S1097

BTZ043 Racemate

BTZ043 racemate is a decaprenylphosphoryl-β-D-ribose 2'-epimerase (DprE1) inhibitor acting as a new antimycobacterial agent that kill Mycobacterium tuberculosis.

S1591

Bestatin

Bestatin is a potent aminopeptidase-B and leukotriene (LT) A4 hydrolase inhibitor, used in the treatment of acute myelocytic leukemia.

S1601

Reserpine

Reserpine is an inhibitor of multidrug efflux pumps, used as an antipsychotic and antihypertensive drug.

S1428

Risedronate Sodium

Risedronate Sodium, a nitrogen-containing bisphosphonate, inhibits osteoclast-mediated bone resorption and modulates bone metabolism, used in the treatment of osteoporosis.

S1271

Acarbose

Acarbose is an inhibitor of intestinal alpha-glucosidase, used to treat type 2 diabetes mellitus.

S1624

Alendronate sodium trihydrate

Alendronate sodium trihydrate, a nitrogen-containing bisphosphonate, is a potent inhibitor of bone resorption used for the treatment and prevention of osteoporosis.

S1988

Propylthiouracil

Propylthiouracil is a thyroperoxidase and 5'-deiodinase inhibitor, used to treat hyperthyroidism.

S1698

Torsemide

Torsemide is a pyridyl sulfonylurea with a chemical structure between that of traditional loop diuretics and Cl- channel blockers, used to treat hypertension.

S7372

PTC-209

PTC-209 is a potent and selective BMI-1 inhibitor with IC50 of 0.5 μM in HEK293T cell line, and results in irreversible reduction of cancer-initiating cells (CICs).

S7270

SRPIN340

SRPIN340 is a selective SRPK inhibitor with Ki of 0.89 μM for SRPK1, showing no significant inhibitory activity against more than 140 other kinases..

S7272

4μ8C

4μ8C is a potent and selective IRE1 Rnase inhibitor with IC50 of 76 nM.

S2129

Fudosteine

Fudosteine is a cysteine derivative and a MUC5AC mucin hypersecretion inhibitor, used as a muco-active agent with indications for chronic respiratory diseases.

S8077

RI-1

RI-1 is a RAD51 inhibitor with IC50 ranging from 5 to 30 μM.

S2610

Lonidamine

Lonidamine is an orally administered small molecule hexokinase inactivator.

S2901

CCG 50014

CCG 50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM.

S2035

Epalrestat

Epalrestat is an aldose reductase inhibitor with IC50 of 72 nM.

S3199

Reboxetine mesylate

Reboxetine is a norepinephrine reuptake inhibitor with Ki of 8.2 nM.

S7369

4EGI-1

4EGI-1 is a competitive eIF4E/eIF4G interaction inhibitor by binding to eIF4E with KD of 25 μM.

S1875

Tranexamic Acid

Tranexamic Acid is an antifibrinolytic for blocking lysine-binding sites of plasmin and elastase-derived plasminogen fragments with IC50 of 5 mM.

S4020

Sodium Picosulfate

Sodium Picosulfate inhibits absorption of water and electrolytes, and increases their secretion.

S2032

Rebamipide

Rebamipide is a cholecystokinin type 1 (CCK1) receptor inhibitor for inhibiting [125I]BH-CCK-8S with IC50 of 37.7 μM.

S7382

Phosphoramidon Disodium Salt

Phosphoramidon Disodium Salt is a metalloendopeptidase inhibitor, widely used as a biochemical tool.

S7589

N6022

N6022 is a selective, and reversible inhibitor of S-nitrosoglutathione reductase (GSNOR) with IC50 of 8 nM and Ki of 2.5 nM. Phase 1/2.

S7922

Tiplaxtinin (PAI-039)

Tiplaxtinin(PAI-039) is an orally efficacious and selective plasminogen activator inhibitor-1 (PAI-1) inhibitor with IC50 of 2.7 μM.

S4299

Dicoumarol

Dicoumarol is a competitive NADH quinone oxidoreductase (NQO1) inhibitor,and used as an anticoagulant by interfering with the metabolism of vitamin K.

S4017

Allylthiourea

Allylthiourea is a metabolic inhibitor that selective inhibits ammonia oxidation.

S2830

Clindamycin

Clindamycin inhibits protein synthesis by acting on the 50S ribosomal, used for the treatment of bacterial infections.

S7209

GSK650394

GSK650394 is a serum- and glucocorticoid-regulated kinase-1 inhibitor with IC50 of 62 nM and 103 nM for SGK1 and SGK2, respectively.

S7370

4E1RCat

4E1RCat is a dual inhibitor of eIF4E:eIF4G and eIF4E:4E-BP1 interaction, and inhibits the binding of eIF4G to eIF4E with IC50 of 3.2 μM.

S2256

4-Methylumbelliferone (4-MU)

4-Methylumbelliferone is a hyaluronic acid (HA) synthesis inhibitor with an IC50 of 0.4 mM.

S7771

STF-083010

STF-083010 is a specific IRE1α endonuclease inhibitor without affecting its kinase activity.

S4153

D-Phenylalanine

D-Phenylalanine, a carboxypeptidase A, endorphinase and enkephalinase inhibitor, enhances endorphin production and diminishes pain.

S7635

Lomitapide

Lomitapide is a potent microsomal triglyceride transfer protein (MTP) inhibitor, used in the treatment of familial hypercholesterolemia.

S2422

Ipriflavone (Osteofix)

Ipriflavone (7-Isopropoxyisoflavon) is used to inhibit bone resorption.

S7213

Thiamet G

Thiamet G is a potent, selective O-GlcNAcase inhibitor with Kiof 21 nM, while exhibiting 37,000-fold selectivity over human lysosomal –hexosaminidase.

S7633

Lomitapide Mesylate

Lomitapide Mesylate is a potent microsomal triglyceride transfer protein (MTP) inhibitor, used in the treatment of familial hypercholesterolemia.

S7443

AP-III-a4 (ENOblock)

AP-III-a4 (ENOblock) is the first nonsubstrate analogue inhibitor of enolase with IC50 of 0.576 μM.

S2404

Isoliquiritigenin

Isoliquiritigenin, an anti-tumor flavonoid from the root of Glycyrrhiza glabra, inhibits aldose reductase with an IC50 of 320 nM.

S7929

BEC HCl

BEC HCl is a slow-binding, and competitive arginase inhibitor with Ki of 0.31 μM (pH7.5) and 0.4-0.6 μM for Arginase II and rat Arginase I, respectively.

S7339

AZD3965

AZD3965 is a potent, selective and orally available monocarboxylate transporter 1 (MCT1) inhibitor with a binding affinity of 1.6 nM, 6-fold selective over MCT2. Phase 1.

S7517

AZD7545

AZD7545 is a potent PDHK inhibitor with IC50 of 36.8 nM and 6.4 nM for PDHK1 and PDHK2, respectively. It failed to inhibit PDHK4 at higher concentrations(>10 nM), AZD7545 stimulates PDHK4 activity.

S7606

RBC8

RBC8 is a selective inhibitor of the GTPases RalA and RalB by inhibiting the binding of Ral to its effector RALBP1, no inhibition on the GTPases Ras and RhoA.

S7539

PTC-209 HBr

PTC-209 HBr is the hydrobromide salt of PTC-209, which is a potent and selective BMI-1 inhibitor with IC50 of 0.5 μM, and results in irreversible reduction of cancer-initiating cells (CICs).

S8196

ML264

ML264, a selectively inhibitor of kruppel-like factor 5 (KLF5),potently Inhibits Growth of Colorectal Cancer.

S7852

Eliglustat Tartrate

Eliglustat (Tartrate) inhibits glucosylceramide synthase(GCS),thus reducing the load of glucosylceramide influx into the lysosome.

S4108

Clodronate Disodium

Clodronate Disodium, a bisphosphonate, is a potent antiosteolytic agent which inhibits bone resorption.

S4233

Zoxazolamine

Zoxazolamine is a centrally acting myorelaxant, which is formerly used as an antispasmodic and uricosuric.

S2916

ML161

ML-161 is an allosteric inhibitor of PAR1 with IC50 of 0.26 μM.

S2063

Pamidronate

Pamidronate is bisphosphonate which binds to the hydroxyapatite in bone and act as an inhibitor of the resorption of bone for the treatment of osteitis deformans and postmenopausal osteoporosis.

S7498

DDR1-IN-1

DDR1-IN-1 is a potent and selective discoidin domain receptor 1 (DDR1) receptor tyrosine kinase inhibitor with IC50 of 105 nM, about 3-fold selectivity over DDR2.

S7814

AI-10-49

AI-10-49 is a selective inhibitor of the binding of CBFβ-SMMHC to RUNX1 with IC50 of 260 nM.

S7685

SecinH3

SecinH3 is a selective cytohesin inhibitor with IC50 of 2.4 μM, 5.4 μM, 5.4 μM, 5.6 μM, 5.6 μM, and 65 μM for hCyh2, hCyh1, mCyh3, hCyh3, drosophila steppke, and yGea2-S7, respectively.

S7873

Disodium (R)-2-Hydroxyglutarate

Disodium (R)-2-Hydroxyglutarate is a competitive inhibitor of α-ketoglutarate-dependent dioxygenases with Ki of 0.628 mM.

Catalog No. Information Product Use Citations Product Validations
S2155

LY2608204

LY2608204 activates glucokinase (GK) with EC50 of 42 nM. Phase 2.

S1511

Lactulose

Lactulose, a disaccharide composed of galactose and fructose, is a stimulator of health-promoting bacterium growth in the gastrointestinal tract, used to treat chronic constipation and hepatic encephalopathy.

S7928

DASA-58

DASA-58 is a specific and potent Pyruvate kinase M2 (PKM2) activator.

S7447

ZLN005

ZLN005 is a potent and tissue-specific PGC-1α transcriptional activator.

2016, 345(1):25-36

Catalog No. Information Product Use Citations Product Validations
S3038

Fosaprepitant dimeglumine salt

Fosaprepitant is a water-soluble phosphoryl prodrug for Aprepitant which is a NK1 antagonist.

S7976

SBC-115076

SBC-115076 is a potent extracellular proprotein convertase subtilisin kexin type 9 (PCSK9) antagonist.

Catalog No. Information Product Use Citations Product Validations
S7365

AdipoRon

AdipoRon is a novel, and orally bioavailable adiponectin receptor agonist with KD of 1.8 and 3.1 μM for AdipoR1 and AdipoR2, respectively.

S2066

Moxonidine

Moxonidine is a selective agonist at the imidazoline receptor subtype 1, used as antihypertensive agent.

S7548

Rilmenidine Phosphate

Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist, used for the treatment of hypertension.

S7608

UM171

UM171 is a potent agonist of human hematopoietic stem cell renewal, independently of AhR suppression.

Catalog No. Information Product Use Citations Product Validations
S7594

Abscisic Acid (Dormin)

Abscisic Acid is a plant hormone, which is involved in many plant developmental processes, modulates ion homeostasis and metabolism, and inhibits germination and seedling growth.

Catalog No. Information Product Use Citations Product Validations
S6002

NXY-059 (Disufenton sodium)

NXY-059 is a novel nitrone, shows efficacious neuroprotective effects. Phase 3.

2015, 86:308-21

S1751

Gadodiamide Hydrate

Gadodiamide Hydrate, a nonionic Gd3+ chelate, is frequently injected i.v. into magnetic resonance imaging (MRI) to enhance contrast.

2014, 22(9):1311-21

2015, 427(4):966-81

S1236

Leucovorin Calcium Pentahydrate

Leucovorin is a derivative of folic acid, which can be used to increase levels of folic acid under conditions favoring folic acid inhibition.

S4728New

3,3'-Diindolylmethane

3,3'-Diindolylmethane(DIM) is a major digestive product of indole-3-carbinol, a potential anticancer component of cruciferous vegetables.

S1627

Nitazoxanide

Nitazoxanide is a synthetic nitrothiazolyl-salicylamide derivative and an antiprotozoal agent. (IC50 for canine influenza virus ranges from 0.17 to 0.21 μM)

S1137

Malotilate

Malotilate, diisopropyl 1,3-dithiol-2-ylidenemalonate, is a drug used for the treatment of liver cirrhosis.

S1934

Nystatin (Fungicidin)

Nystatin, which belongs to the polyene group of antimycotics, is frequently used as a topical agent in the treatment of oro-pharyngeal candidosis.

S2757

TH-302

TH-302 is selective hypoxia-activated prodrug targeting hypoxic regions of solid tumors with IC50 of 19 nM, demonstrates 270-fold enhanced cytotoxicity under hypoxia versus their potency under aerobic conditions, stable to cytochrome P450 metabolism.

S1311

Pamidronate Disodium

Pamidronate Disodium is a nitrogen containing bisphosphonate, used to prevent osteoporosis.

S2553

5-Aminolevulinic acid HCl

5-Aminolevulinic Acid HCl is an intermediate in the porphyrin synthesis pathway, used as a photosensitizing agent and a antineoplastic agent.

S1201

Dimesna

Dimesna is an uroprotective agent used to decrease urotoxicity.

S1732

Mitotane

Mitotane, is an antineoplastic medication used in the treatment of adrenocortical carcinoma.

2016, 10.1007/s10637-016-0358-3

S2417

20-Hydroxyecdysone

20-Hydroxyecdysone (Ecdysterone, 20E) is a naturally occurring ecdysteroid hormone which controls the ecdysis (moulting) and metamorphosis of arthropods.

S1326

Edaravone

Edaravone is a novel potent free radical scavenger that has been clinically used to reduce the neuronal damage following ischemic stroke.

S1897

Potassium Iodide

Potassium Iodide is used to treat overactive thyroid and to protect the thyroid gland from the effects of radiation from inhaled or swallowed radioactive iodine.

S2586

Dimethyl Fumarate

Dimethyl fumarate (DMF)is the methyl ester of fumaric acid, used to treat people with relapsing forms of multiple sclerosis.

2014, 15(12):1646-57

S1740

Guaifenesin

Guaifenesin is an expectorant used to relieve chest congestion.

S4067

Deferiprone

Deferiprone is a chelating agent with an affinity for ferric ion (iron III),binds with ferric ions to form neutral 3:1 (deferiprone:iron) complexes that are stable over a wide range of pH values.

S1287

Bumetanide

Bumetanide (Bumex) is a loop diuretic of the sulfamyl category to treat heart failure.

S7217

OAC1

OAC1 (Oct4-activating compound 1) can enhance the efficiency of reprogramming.

S1849

Daidzein

Daidzein is a natural isoflavone phytoestrogen found in Leguminosae, used as a component of foods and dietary supplements.

S2408

Cephalomannine

Cephalomannine is an active anti-cancer agent obtained from Taxus yunnanensis and has an antineoplastic effect on tumors found in mice.

S4059

Sodium Nitroprusside Dihydrate

Sodium Nitroprusside Dihydrate is a potent vasodilator working through releasing NO spontaneously in blood.

S7450

FH1(BRD-K4477)

FH1 (BRD-K4477) is a small molecule, which promotes differentiation of iPS-derived hepatocytes.

S1749

L-Glutamine

L-Glutamine (Gln) is one of the 20 amino acids encoded by the standard genetic code and also a major respiratory fuel and substrate for nucleic acid synthesis in mammalian intestinal cells.

S1917

Crystal Violet

Crystal violet is a triarylmethane dye.

S1874

Risedronate

Risedronate is a bisphosphonate used to strengthen bone, treat or prevent osteoporosis, and treat Paget's disease of bone.

S2412

Genipin

Genipin is an active aglycone derived from an iridoid glycoside called geniposide, which is found in the fruit of Gardenia jasminoides Ellis.

S2410

Paeoniflorin

Paeoniflorin is a herbal constituent extracted from the root of Paeonia albiflora Pall.

S1609

Methimazole

Methimazole is an antithyroid medicine.

S2594

Pramiracetam

Pramiracetam is a more potent nootropic drug derived from piracetam.

S2388

L-carnitine

L-carnitine is constituent of striated muscle and liver. It is used therapeutically to stimulate gastric and pancreatic secretions and in the treatment of hyperlipoproteinemias.

S1643

Ursodiol

Ursodiol reduces cholesterol absorption and is used to dissolve (cholesterol) gallstones. (IC50=0.22 μM)

S1647

Adenosine

Adenosine is a nucleoside composed of a molecule of adenine attached to a ribose sugar molecule (ribofuranose) moiety via a β-N9-glycosidic bond.

S1671

(6-)ε-​Aminocaproic acid

(6-)ε-​Aminocaproic acid is a derivative and analogue of the amino acid lysine.

S1853

Penicillamine

Penicillamine is used as an antirheumatic and as a chelating agent in Wilson’s disease.

S2536

Miconazole

Miconazole (Monistat) is an imidazole antifungal agent.

S2724

Heparin sodium

Heparin sodium is a sodium salt of heparin which is a naturally-occurring anticoagulant used for anticoagulation for cardiovascular disease.

S1806

Acipimox

Acipimox is a niacin derivative used as a hypolipidemic agent.

S4217

Liothyronine Sodium

Liothyronine Sodium is the most potent form of thyroid hormone acting on the body to increase the basal metabolic rate, affect protein synthesis.

S1985

ATP

ATP Disodium is a disodium salt form of adenosine-triphosphate that is used in cells as a coenzyme.

S3148

Ibandronate sodium

Ibandronate is a highly potent nitrogen-containing bisphosphonate used for the treatment of osteoporosis.

S3150

Articaine HCl

Articaine is a dental local anesthetic which contains an additional ester group that is metabolized by estearases in blood and tissue.

S3000

Carbazochrome sodium sulfonate (AC-17)

Carbazochrome sodium sulfonate (AC-17) is an antihemorrhagic for use in the treatment of hemorrhoids.

S2599

L-Thyroxine

L-Thyroxine is a synthetic form of thyroxine and a hormone replacement drug.

S1610

Metolazone

Metolazone is a diuretic that primarily used to treat congestive heart failure and high blood pressure.

S4129

Sevelamer HCl

Sevelamer HCl is a phosphate binding drug used to treat hyperphosphatemia via binding to dietary phosphate and prevents its absorption.

S2381

D-Mannitol

D-Mannitol is an osmotic diuretic agent and a weak renal vasodilator.

S2393

Sorbitol

Sorbitol is a sugar alcohol and a sugar substitute.

S1641

Chlorothiazide

Chlorothiazide is a diuretic and antihypertensive. (IC50=3.8 mM)

S2293

DL-Carnitine HCl

DL-Carnitine HCl is a quaternary ammonium compound biosynthesized from the amino acids lysine and methionine.

S2305

Grape Seed Extract

Grape Seed Extract are industrial derivatives from whole grape seeds that have a great concentration of vitamin E, flavonoids, linoleic acid, and OPCs.

S1715

Glipizide

Glipizide is used to treat high blood sugar levels caused by a type of diabetes mellitus called type 2 diabetes.

S4095

Difluprednate

Difluprednate (difluoroprednisolone butyrate acetate, or DFBA) is a synthetic difluorinated prednisolone derivative, it is originally developed for dermatologic applications.

S1928

Alibendol

Alibendol is an antispasmodic,choleretic, and cholekinetic.

S1735

Mesna

Mesna, a sulfhydryl compound that is used to reduce the incidence of hemorrhagic cystitis associated with certain chemotherapeutic agents.

S2411

Geniposide

Geniposide is an iridoid glycoside isolated from the fruit of Gardenia jasminoides Ellis.

S2409

10-Deacetylbaccatin-III

10-Deacetylbaccatin-III is an antineoplastic agent and an anti-cancer intermediate.

S3209

Amidopyrine

Amidopyrine is a white crystalline substance used as an analgesic and antipyretic.

S1708

Hydrochlorothiazide

Hydrochlorothiazide is a first line diuretic compound of the thiazide class.

S2596

Clindamycin palmitate HCl

Clindamycin palmitate HCl is a water soluble hydrochloride salt of the ester of clindamycin and palmitic acid and a lincosamide antibiotic.

S4298

Amifostine

Amifostine is the first approved radioprotective drug, used to decrease the risk of kidney problems caused by treatment with cisplatin.

S7909

Dp44mT

Dp44mT is a potent iron chelator, which shows selective antitumor activity.

S7913

MCB-613

MCB-613 is a potent steroid receptor coactivator (SRC) stimulator.

S7914

Isoxazole 9 (ISX-9)

Isoxazole 9 (Isx-9) is a synthetic promotor of adult neurogenesis by triggering neuronal differentiation of adult neural stem/precursor cells (NSPCs).

S2589

Miglitol

Miglitol is an oral anti-diabetic drug.

S2518

NAD+

NAD+ is a coenzyme composed of ribosylnicotinamide 5'-diphosphate coupled to adenosine 5'-phosphate by pyrophosphate linkage.

S4015

Cyclamic acid

Cyclamic acid in the form of its sodium or calcium salt is one of the most widely used artificial sweeteners.

S1730

Indapamide

Indapamide is a non-thiazide sulphonamide diuretic compound, generally used in the treatment of hypertension, as well as decompensated cardiac failure.

S7363

BRD7552

BRD7552 is an inducer of transcription factor PDX1, which increases insulin expression.

S4115

Hydroxypropyl Cellulose

Hydroxypropyl cellulose (HPC) is a derivative of cellulose with both water solubility and organic solubility, it is used as food additive and sieving matrix for DNA separations.

S2052

Oxytetracycline Dihydrate

Oxytetracycline Dihydrate is a prescription antibiotic, interfering with the ability of bacteria to produce essential proteins.

S2053

Cytidine

Cytidine is a nucleoside molecule that is formed when cytosine is attached to a ribose ring, cytidine is a component of RNA.

S4128

Troxipide

Troxipide is a novel systemic non-antisecretory gastric cytoprotective agent with anti-ulcer, anti-inflammatory and mucus secreting properties irrespective of pH of stomach or duodenum.

S4134

Sevelamer Carbonate

Sevelamer carbonate is a non-absorbed phosphate binding crosslinked polymer, with the same polymeric structure as sevelamer hydrochloride, in which carbonate replaces chloride as the counterion.

S2008

Taurine

Taurine is an organic acid widely distributed in animal tissues.

S4137

Eprazinone 2HCl

Eprazinone is a mucolytic.

S2060

Bromhexine HCl

Bromhexine HCl is a medication prescribed for coughs which works by dissolving hard phlegm.

S4138

Dropropizine

Dropropizine is a racemic non-opiate antitussive agent, it is used as a cough suppressant.

S2252

(+)-Usniacin

(+)-Usniacin is a naturally occurring dibenzofuran derivative found in several lichen species.

S3068

Guanosine Hydrate

Guanosine hydrate plays important roles in various biochemical processes such as synthesis of nucleic acids and proteins, photosynthesis, muscle contraction and intracellular signal transduction (cGMP).

S2253

3-Indolebutyric acid (IBA)

3-Indolebutyric acid(IBA) is a plant hormone in the auxin family and is an ingredient in many commercial plant rooting horticultural products.

S2424

Hypoxanthine

Hypoxanthine, a naturally occurring purine derivative, an intermediate product of uric acid synthesis, formed from adenylic acid and itself a precursor of xanthine.

S2374

5-hydroxytryptophan (5-HTP)

5-Hydroxytryptophan (5-HTP), also known as oxitriptan (INN), is a naturally occurring amino acid and chemical precursor for the treatment of depression.

S2442

Inosine

Inosine is a nucleoside that is formed when hypoxanthine is attached to a ribose ring via a β-N9-glycosidic bond.

S2258

Esculin

Esculin is a glucoside found in horse chestnuts.

S3071

Vanillin

Vanillin, 4-hydroxy-3-methoxybenzaldehyde, is a food additive.

S4040

Norethindrone

Norethindrone is a synthetic progestin, which mimic the actions of the endogenous ovarian hormone progesterone.

S2260

Amygdalin

Amygdalin is a glycoside initially isolated from the seeds of the tree Prunus dulcis, also known as bitter almonds.

S2379

Dioscin

Dioscin is a saponin extracted and isolated from Polygonatum Zanlanscianense Pamp, showing antitumor activities.

S2383

Gastrodin

Gastrodin, an anti-inflammatory polyphenol extracted from Chinese natural herbal Gastrodia elata Blume., benefits neurodegenerative diseases.

S4154

Cholesterol

Cholesterol is the principal sterol of all higher animals required to build and maintain membranes.

S2384

Hematoxylin

Hematoxylin (Hydroxybrazilin) is a compound that forms strongly colored complexes with certain metal ions, notably Fe(III) and Al(III) salts and a kind of stain in histology.

S8128

BAY 41-2272

BAY 41-2272 is a direct and NO-independent soluble guanylate cyclase (sGC) stimulator.

S2267

Azomycin

Azomycin is an antimicrobial antibiotic produced by a strain of Nocardia mesenterica.

S2387

Lappaconite HBr

Lappaconite Hydrobromide is a kind of alkaloid extracted from Aconitum sinomontanum Nakai and has anti-inflammatory effects.

S2883

4-Aminohippuric Acid

4-Aminohippuric acid is a typical substrate of organic anion transport systems.

S2884

Acesulfame Potassium

Acesulfame potassium is a non-nutritive sweetener.

S8135

Riociguat (BAY 63-2521)

Riociguat (BAY 63-2521) is an oral soluble guanylate cyclase (GC) stimulator, used in the treatment of ipulmonary hypertension.

S2270

Bergenin

Bergenin is trihydroxybenzoic acid glycoside and the C-glycoside of 4-O-methyl gallic acid.

S4161

Benzoic Acid

Benzoic acid is a colorless crystalline solid and a simple aromatic carboxylic acid, used as a food preservative.

S2273

β-Sitosterol

β-Sitosterol is one of several phytosterols (plant sterols) with chemical structures similar to that of cholesterol.

S2392

Sesamin

Sesamin, a lignan isolated from the bark of Fagara plants and from sesame oil, exhibits various health benefits.

S2276

Bilobalide

Bilobalide is a biologically active terpenic trilactone present in Ginkgo biloba.

S2277

Caffeic Acid

Caffeic acid is a hydroxycinnamic acid, a naturally occurring organic compound.

2015, 5:12580

S4047

Bisacodyl

Bisacodyl (INN) is a stimulant laxative drug that works directly on the colon to produce a bowel movement.

S2280

Chlorogenic Acid

Chlorogenic acid is a hydroxycinnamic acid and a member of a family of naturally occurring organic compounds.

S4048

Carbimazole

Carbimazole is an imidazole antithyroid agent.

S2281

Chrysin

Chrysin is a naturally occurring flavone chemically extracted from the blue passion flower (Passiflora caerulea).

S4166

Chlorpropamide

Chlorpropamide is a sulfonylurea class drug for type 2 diabetes mellitus.

S2290

Dihydroartemisinin (DHA)

Dihydroartemisinin (DHA) is a semi-synthetic derivative of artemisinin and isolated from the traditional Chinese herb Artemisia annua.

2015, 6(7):5275-91

2015, 10(3):e0120426

2017, 10.1186/s13046-017-0531-3

S7763

D-Luciferin

D-Luciferin is a popular bioluminescent substrate of luciferase in the presence of ATP, used in luciferase-based bioluminescence imaging and cell-based high-throughput screening applications.

S2292

Diosmin

Diosmin is a semisynthetic phlebotropic agent and a member of the flavonoid family.

S4173

1-Hexadecanol

1-Hexadecanol is a fatty alcohol used to make other chemicals.

S1974

Meglumine

Meglumine is an amino sugar derived from sorbitol for THP-1 cells with IC50 of 22 μg/mL.

S4174

Sodium Gluconate

Sodium gluconate is the sodium salt of gluconic acid widely used in food and pharmaceutical industry.

S2396

Salidroside

Salidroside, a phenylpropanoid glycoside isolated from Rhodiola rosea, has been reported to have a broad spectrum of pharmacological properties.

S4057

Methyclothiazide

Methyclothiazide is a substituted benzothiadiazide, used to treat high blood pressure and fluid retention caused by various conditions including heart disease.

S4177

Uracil

Uracil is one of the four nucleobases in the nucleic acid of RNA can be used for drug delivery and as a pharmaceutical.

S2397

Palmatine chloride

Palmatine hydrochloride (Palmatine chloride (6CI,7CI); Fibrauretin) is a hydrochloride salt of palmatine which is a protoberberine alkaloid.

S2299

Formononetin

Formononetin is a phytoestrogen from the root of Astragalus membranaceus and an O-methylated isoflavone.

S2398

Coenzyme Q10 (CoQ10)

Coenzyme Q10 (ubiquinone, ubidecarenone, coenzyme Q) is a component of the electron transport chain and participates in aerobic cellular respiration.

S2300

Ferulic Acid

Ferulic Acid is a hydroxycinnamic acid and a type of organic compound found in the Ferula assafoetida L. or Ligusticum chuanxiong.

S2402

Cyclovirobuxin D

Cyclovirobuxine D is an active compound extracted from Buxus microphylla, which has been used for treating acute myocardial ischemia.

S2304

Gramine

Gramine is a naturally occurring indole alkaloid present in several plant species.

S2306

Gynostemma Extract

Gynostemma Extract is a saponins extract derived from the Gynostemma pentaphyllum.

S4185

Tiratricol

Tiratricol (also known as TRIAC or triiodothyroacetic acid) is a thyroid hormone analogue.

S2309

Hesperidin

Hesperidin is a flavanone glycoside found abundantly in citrus fruits.

S4186

Domiphen Bromide

Domiphen bromide is a quaternary ammonium antiseptic with actions as a cationic surfactant.

S2405

Sophocarpine

Sophocarpine, a major ingredient of Sophora alopecuroides, has a wide range of pharmacological effects.

S2311

Hyodeoxycholic acid (HDCA)

Hyodeoxycholic(HDCA) acid is a secondary bile acid, one of the metabolic byproducts of intestinal bacteria.

S4189

Cyclandelate

Cyclandelate is an effective inhibitor of rat hepatic acycloenzyme A: cholesterol acyltransferase (ACAT) with IC50 of 80 μM.

S4190

Cinchophen

Cinchophen is an analgesic drug that is frequently used to treat gout.

S4070

Guanidine HCl

Guanidine HCl, the crystalline compound of strong alkalinity formed by the oxidation of guanine, is a normal product of protein metabolism and a protein denaturant.

S4077

Mequinol

Mequinol (4-Methoxyphenol) is a depigmentation agent.

S7451

FPH1 (BRD-6125)

FPH1 (BRD-6125) is a small molecule, which promotes expansion of iPS-derived hepatocytes.

S4263

Efaproxiral Sodium

Efaproxiral Sodium is a synthetic allosteric modifier of hemoglobin, used for brain metastases originating from breast cancer.

S4264

Etofibrate

Etofibrate is a combination of clofibrate and niacin, used to treat hyperlipemia.

S4265

Nicaraven

Nicaraven is a hydroxyl radical scavenger with antivasospastic and neuroprotective effects.

S2021

Chlormezanone

Chlormezanone,a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.

S4194

Azaguanine-8

Azaguanine-8 is a purine analogs showing antineoplastic activity by competing with guanine in the metabolism.

S2316

Kinetin

Kinetin is a type of cytokinin, a class of plant hormone that promotes cell division.

S2317

L-(+)-Rhamnose Monohydrate

L(+)-Rhamnose (Rham) is a naturally-occurring deoxy sugar that is found primarily in plants and some bacteria.

S7453

MSDC-0160

MSDC-0160 is a prototype mTOT-modulating insulin sensitizer being studied to treat diabetes and Alzheimer's disease. Phase 2.

S4092

Pramoxine HCl

Pramoxine is a topical local anesthetic that has been shown to have antipruritic properties.

S4204

Isosorbide

Isosorbide is a heterocyclic compound that is derived from glucose, used as a diuretic.

S2124

Xylose

Xylose is a sugar first isolated from wood.

S4205

Dibenzothiophene

Dibenzothiophene (DBT) is a model compound for organic sulfur in fossil fuels.

S8199

LTX-315

LTX-315 is the oncolytic peptide that kills cancer cells through Bax/Bak-regulated mitochondrial membrane permeabilization.

S2323

Methyl-Hesperidin

Methyl Hesperidin is a flavanone glycoside (flavonoid) (C28H34O15) found abundantly in citrus fruits. Its aglycone form is called hesperetin.

S2538

Acetanilide

Acetanilide is an aniline derivative and has possess analgesic.

S4206

Cysteamine HCl

Cysteamine is an agent for the treatment of nephropathic cystinosis and an antioxidant.

S4208

Chromocarb

Chromocarb is a vasoprotectant.

S7534

BAPTA-AM

BAPTA-AM is a selective, membrane-permeable calcium chelator.

2016, 11(7):e0159089

2017, 10.1111/jcmm.13067

S2609

Inulin

Inulin(Inulin and sodium chloride), a starch found in the tubers and roots of many plants. Since it is hydrolyzable to fructose, it is classified as a fructosan.

S1904

Avobenzone

Avobenzone is an oil soluble ingredient used in sunscreen products to absorb the full spectrum of UVA rays and a dibenzoylmethane derivative.

S4214

Sucralose

Sucralose is an artificial and noncaloric sweetener, not broken down by the body.

S2324

Sodium Monensin

Sodium Monensin, isolated from Streptomyces cinnamonensis, is a well-known representative of naturally polyether ionophore antibiotics.

2013, 75(1):9-17

S1825

Erdosteine

Erdosteine is a mucolytic which is used in treatment of excessive viscous mucus.

S4101

Voglibose

Voglibose is an N-substituted derivative of valiolamine, excellent inhibitory activity against α-glucosidases and its action against hyperglycemia and various disorders caused by hyperglycemia.

S7446

L-Mimosine

L-Mimosine is a non-protein amino acid, and acts as an iron chelator.

S2325

Morin Hydrate

Morin hydrate(Aurantica) is a flavonoid isolated from Maclura pomifera (Osage orange), Maclura tinctoria (old fustic) and from leaves of Psidium guajava (common guava).

S2439

Guanosine

Guanosine is a purine nucleoside comprising guanine attached to a ribose (ribofuranose) ring via a β-N9-glycosidic bond.

S4104

Diminazene Aceturate

Diminazene is a di-amidine also known as 4,4-(1-Triazene–1,3–diyl)bis(benzenecarboximidamide), used as an effective trypanocidal agent.

S2331

Neohesperidin Dihydrochalcone (Nhdc)

Neohesperidin dihydrochalcone(Nhdc), sometimes abbreviated to neohesperidin DC or simply NHDC, is an artificial sweetener derived from citrus.

S2335

Oridonin

Oridonin, a diterpenoid purified from Rabdosia rubescens, is an antitumor agent.

S2336

Orotic acid (6-Carboxyuracil)

Orotic acid(6-Carboxyuracil) is a heterocyclic compound and an acid.

S2337

Osthole

Osthol is an O-methylated coumarin, which is found in the plants such as Cnidium monnieri, Angelica archangelica and Angelica pubescens.

2014, 73:260-9

2015, 22:63

2014, Haoran Cui

S2338

Oxymatrine

Oxymatrine is a quinolizidine alkaloid extracted from the root of Sophora flavescens with anti-inflammatory, antifibrosis, and antitumor effects, inhibits the iNOS expression and TGF-β/Smad pathway. It is used for the treatment of viral hepatitis, cancer, viral myocarditis, gastrointestinal hemorrhage and skin diseases.

S4224

Erythritol

Erythritol is a sugar alcohol used as low-calorie sweetener.

S7452

FPH2 (BRD-9424)

FPH2 (BRD-9424) is a small molecule, which promotes differentiation of iPS-derived hepatocytes.

S3100

2-Thiouracil

2-Thiouracil is a thiolated uracil derivative that is a known antihyperthyroid agent.

S3102

Creatinine

Creatinine is a break-down product of creatine phosphate in muscle, and is usually produced at a fairly constant rate by the body.

S2347

Quercetin Dihydrate

Quercetin, a polyphenolic flavonoid found in a wide variety of plant-based foods, such as apples, onions, berries, and red wine, is utilized in many different cultures for their nervous system and anticancer effects.

S4508

2,2,2-Tribromoethanol

2,2,2-Tribromoethanol is an organic compound used to anesthetize mice.

S4510

4-Aminobenzoic acid

4-Aminobenzoic acid is an intermediate in the synthesis of tetrahydrofolic acid in many non-mammalian organisms, including bacteria and fungi.

S3106

Pidotimod

Pidotimod is an immunostimulant.

S3104

Moguisteine

Moguisteine is a novel peripheral non-narcotic antitussive drug.

S4519

Citric acid trilithium salt tetrahydrate

Citric acid trilithium salt tetrahydrate is a pharmaceutical and construction material. It is commonly used in HPLC gradient elution for quantification of amino acids.

S4530

i-Inositol

i-Inositol, also known as myo-inositol, is a chemical compound which is sugar alcohol. i-Inositol is involved in a number of biological processes including insulin signal transduction, cytoskeleton transduction and so on.

S2074

Mecarbinate

Mecarbinate is a chemical intermediate of arbidol hydrochloride.

S3138

Methylthiouracil

Methylthiouracil is an antithyroid preparation.

S4532

Iopamidol

Iopamidol is a non-ionic, water-soluble radiographic contrast agent.

S2353

Sapogenins Glycosides

Sapogenins glycosides are a mixture of triterpene and steroid saponins isolated from medicinal plants such as Aesculus hippocastanum L., Hedera helix L. and Ruscus aculeatus L., which are claimed to be effective for the treatment/prevention of venous insufficiency.

S3190

N6-methyladenosine (m6A)

N6-methyladenosine (m6A) is a base modified analog of adenosine and is found as a minor nucleoside in natural RNAs.

2016, 476(4):340-5

S2354

Sclareol

Sclareol, a labdane-type diterpene isolated from clary sage (Salvia sclarea), exerts growth inhibition and cytotoxic activity against a variety of human cancer cell lines.

S2355

Sclareolide

Sclareolide(Norambreinolide) is a sesquiterpene lactone natural product derived from various plant sources including Salvia sclarea, Salvia yosgadensis, and cigar tobacco.

S4509

4-Aminoantipyrine

4-Aminoantipyrine(Ampyrone) is a metabolite of aminopyrine with analgesic, anti-inflammatory, and antipyretic properties. It is used as a reagent for biochemical reactions producing peroxides or phenols.

S2356

Shikimic Acid

Shikimic acid(Shikimate), more commonly known as its anionic form shikimate, is an important biochemical intermediate in plants and microorganisms.

S2357

Silibinin

Silibinin, the main flavonoid extracted from the milk thistle Silybum marianum, displays hepatoprotective properties in acute and chronic liver injury.

2015, 10.1021/cb5009487

2015, 21(1):49-59

S1900

Talc

Talc is a mineral composed of hydrated magnesium silicate with the chemical formula H2Mg3(SiO3)4 or Mg3Si4O10(OH)2.

S2358

Silymarin

Silymarin (Silybin B), a polyphenolic flavonoid extracted from the seeds of Silybum marianum or milk thistle, is used in the prevention and treatment of liver diseases and primary liver cancer.

2016, 10.1080/13880209.2016.1199042

S2359

Sinomenine

Sinomenine, a pure alkaloid extracted from the chinese medical plant Sinomenium acutum, is used for the treatment of rheumatism and arthritis.

2016, 40:492-500

S7777

Coelenterazine

Coelenterazine is a luminescent enzyme substrate, used for monitoring reporter genes in BRET, ELISA and HTS techniques.

S2036

Aspartame

Aspartame is an artificial, non-saccharide sweetener used as a sugar substitute in some foods and beverages.

S2370

Ursolic Acid

Ursolic acid (Malol) is a pentacyclic triterpene acid, used in cosmetics.

S2371

Vanillylacetone

Vanillylacetone is similar in chemical structure to other flavor chemicals such as vanillin and eugenol and is used as a flavor additive in spice oils and in perfumery to introduce spicy aromas.

S2372

Xanthone

Xanthone is an organic compound, which can be prepared by the heating of phenyl salicylate.