CGRP Receptor

  • Inhibitory Selectivity
  • Solubility
Catalog No. Product Name Solubility(25°C)
Water DMSO Alcohol
S1542 MK-3207 HCl 5 mg/mL 119 mg/mL 119 mg/mL

Isoform-specific Inhibitors

Catalog No. Information Product Use Citations Product Validations
S1542

MK-3207 HCl

MK-3207 is a potent CGRP receptor antagonist with IC50 and Kiof 0.12 nM and 0.022 nM, highly selective versus human AM1, AM2, CTR, and AMY3. Phase 2.

Catalog No. Information Product Use Citations Product Validations
S1542

MK-3207 HCl

MK-3207 is a potent CGRP receptor antagonist with IC50 and Kiof 0.12 nM and 0.022 nM, highly selective versus human AM1, AM2, CTR, and AMY3. Phase 2.

2016, 143(12):2103-10

2015, 10.1186/s13075-014-0513-1