ACK

  • Inhibitory Selectivity
  • Solubility
Catalog No. Product Name Solubility(25°C)
Water DMSO Alcohol
S8272 XMD8-87 <1 mg/mL 65 mg/mL 5 mg/mL
S8273 XMD16-5 <1 mg/mL 83 mg/mL 5 mg/mL
Catalog No. Information Product Use Citations Product Validations
S8272New

XMD8-87

XMD8-87 is a novel tyrosine kinase nonreceptor 2(TNK2) inhibitor with IC50s of 38 nmol/L and 113 nmol/L for the D163E and R806Q mutations.

S8273New

XMD16-5

XMD16-5 is a novel tyrosine kinase nonreceptor 2(TNK2) inhibitor with IC50s of 16 nmol/L and 77 nmol/L for the D163E and R806Q mutations.

Tags: ACK activty | ACK phosphorylation | ACK inhibitor review