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UGT

Other Metabolism Related Inhibitors

Dehydrogenase Transferase DPP Aminopeptidase Procollagen C Proteinase P450 (e.g. CYP17) Phospholipase (e.g. PLA) Factor Xa PDE DHFR
Cat.No. Product Name Information Product Use Citations Product Validations
S4067 Deferiprone Deferiprone (CP20) is a chelating agent with an affinity for ferric ion (iron III)，binds with ferric ions to form neutral 3:1 (deferiprone:iron) complexes that are stable over a wide range of pH values.
Redox Biol, 2025, 85:103739
bioRxiv, 2025, 2025.07.10.663832
Cancer Lett, 2024, 592:216898
S6828 Cremophor EL Cremophor EL, a polyethoxylated surfactant, is a formulation vehicle used for various poorly-water soluble drugs, including the anticancer agent paclitaxel (Taxol). This compound is used in severe anaphylactoid hypersensitivity reactions, hyperlipidaemia, abnormal lipoprotein patterns, aggregation of erythrocytes and peripheral neuropathy.
Aging Dis, 2024, 16(2):1120-1140
Front Oncol, 2022, 12:936145
S2487 Mycophenolic acid Mycophenolic acid (Mycophenolate, RS-61443) is a potent IMPDH inhibitor and the active metabolite of an immunosuppressive drug, used to prevent rejection in organ transplantation.
EMBO Mol Med, 2025, 10.1038/s44321-025-00278-4
Cancer Cell, 2023, 41(1):124-138.e6
Cells, 2023, 12(5)743
S7828 Licochalcone A Licochalcone A is an estrogenic flavanoid extracted from licorice root, showing antimalarial, anticancer, antibacterial and antiviral activities. Phase 3.
Br J Pharmacol, 2023, 180(8):1114-1131
Eur J Pharmacol, 2023, 957:176031
Front Oncol, 2022, 12:1006131
S3608 Demethylzeylasteral (T-96) An active component isolated from Tripterygium wilfordii Hook F., Demethylzeylasteral (T-96) inhibits UDP-glucuronosyltransferase (UGT) isoforms UGT1A6 and UGT2B7 with immunosuppressive effects.
J Cancer, 2025, 16(1):227-240
J Cancer, 2021, 12(13):3967-3975
Front Biosci (Landmark Ed), 2020, 25:498-512
S3018 Niflumic acid Niflumic acid (Nifluril) is an inhibitor of cyclooxygenase-2 used for joint and muscular pain.
Oncol Lett, 2020, 20(4):39
S0931 Jaceosidin Jaceosidin, a flavonoid isolated from Artemisia vestita, possesses anti-tumor and anti-proliferative activities in many cancer cells. This compound induces apoptosis, activates Bax and down-regulates Mcl-1 and c-FLIP expression. It also inhibits COX-2 expression and NF-κB activation.