Doxorubicin (Adriamycin) HCl

Licensed by Pfizer Catalog No.S1208 Synonyms: NSC 123127

Doxorubicin (Adriamycin) HCl Chemical Structure

Molecular Weight(MW): 579.98

Doxorubicin (Adriamycin) HCl is an antibiotic agent that inhibits DNA topoisomerase II and induces DNA damage and apoptosis in tumor cells.

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Cited by 150 Publications

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Choose Selective Topoisomerase Inhibitors

Biological Activity

Description Doxorubicin (Adriamycin) HCl is an antibiotic agent that inhibits DNA topoisomerase II and induces DNA damage and apoptosis in tumor cells.
Targets
Topo II [1]
(Tumor cells)
In vitro

Doxorubicin, an antibiotic anthracycline, is commonly considered to exert its anti-tumor activity at two fundamental levels, altering DNA and producing free radicals to trigger apoptosis of cancer cells through DNA damage. Doxorubicin can block the synthesis of DNA by intercalating into the DNA strand, and inhibits DNA topoisomerase II (TOP2). Doxorubicin is most effective when cells are rapidly proliferating and expressing high levels of TOP2. Additionally, Doxorubicin can trigger apoptosis by producing ceramide (which prompts apoptosis by activating p53 or other downstream pathways such as JNK), the degradation of Akt by serine threonine proteases, the mitochondrial release of cytochrome c, increased FasL (death receptor Fas/CD95 ligand) mRNA production, and a greater production of free radicals. [2] Pre-treatment with GSNO (nitrosoglutathione) suppresses the resistance in the doxorubicin-resistant breast cancer cell line MCF7/Dx, accompanied by enhanced protein glutathionylation and accumulation of doxorubicin in the nucleus. [3] Doxorubicin induced G2/M checkpoint arrest are attributed to elevated cyclin G2 (CycG2) expression and phospho-modification of proteins in the ataxia telangiectasia mutated (ATM) and ATM and Rad3-related (ATR) signaling pathways. [5] Doxorubicin inhibits AMP-activated protein kinase (AMPK), resulting in SIRT1 dysfunction, p53 accumulation, and increased cell death in mouse embryonic fibroblasts (MEFs) and cardiomyocytes, which can be further sensitized by pre-inhibition of AMPK. [6] Doxorubicin elicits a marked heat shock response, and that either inhibition or silencing of heat shock proteins enhance the Doxorubicin apoptotic effect in neuroblastoma cells. Nanomolar Doxorubicin treatment of neuroblastoma cells causes dose-dependent over-ubiquitination of a specific set of proteins in the absence of measurable inhibition of proteasome, and loss of activity of ubiquitinated enzymes such as lactate dehydrogenase and α-enolase, the protein ubiquination patterns of which is similar to those with proteasome inhibitor Bortezomib, indicating that Doxorubicin may also exert its effect by damaging proteins. [8]

Cell Data
Cell Lines Assay Type Concentration Incubation Time Formulation Activity Description PMID
L1210 M3rjW2Z2dmO2aX;uJGF{e2G7 MYPJcohq[mm2aX;uJI9nKFKQQTDzfY51cGW|aYOge4l1cCCHREWwJI9nKDBwNUig{txO M1XsW|Q6ODV|Nh?=
Yoshida sarcoma MlSwSpVv[3Srb36gRZN{[Xl? MmjwTY5pcWKrdHnvckBw\iCdM1jdWIRTKGmwY3;ydI9z[XSrb36ge4l1cCCLQ{WwJI9nKDBwMEKg{txO NWTMVXFqOTN{Mkm4Oi=>
CHO MX\Hdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? M2XzOmlEPTB;MD6wOkDPxE1? MljvNVM2PDd3MB?=
8226 NF6wTZhIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NIPQN2RKSzVyPUCuNFM{KM7:TR?= NGDvNHkyPDR5N{Ow
8226/ADR M3zBOmdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 MkPuTWM2OD1yLkW2JO69VQ>? MX6xOFQ4PzNy
MCF7/ADR NGrJcm5Iem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NX3kVGs4UUN3ME2zMlEh|ryP MVexOFQ4PzNy
H69 M3H3[2dzd3e2aDDJcohq[mm2aX;uJGF{e2G7 M33nd2lEPTB;MD64O{DPxE1? NVOxV25rOTR5OUW4OS=>
N417 NEHuXIxIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= Ml21TWM2OD1yLkKzJO69VQ>? NH73VI8yPDd7NUi1
H9 Mni1S5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MmfyTY5pcWKrdHnvckBw\iCKOTDj[YxteyClaILvcolk[WyueTDpcoZm[3SnZDD3bZRpKHSqZTDITXYuOSBqSEmvTWlKSilid3n0bEBKTDVyIH;mJFAvODFizszN NU\OWoxOOTV2OE[4NS=>
T-C8166 NELCenRIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= MkjoTWQ2OD1yLkCxJO69VQ>? MV6xOVQ5Pjhz
T-H9 MnPBS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MW\JSFUxRTBwMEGg{txO MnjINVU1QDZ6MR?=
T-MT4 NV2wWmJ{T3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NXrXOlh6UUR3ME2wMlAyKM7:TR?= NUnudHFWOTV2OE[4NS=>
SKMEL-5 MYrHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? NH7TepBGTDVyPUOuNkDPxE1? NIrL[Y0yPjF|N{Wz
MLM MWrDfZRwfG:6aXOgRZN{[Xl? M124eGVFPTB;MD6xN{DPxE1? MnqwNVg4PTN3MB?=
KBM-3 MlTFS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MW\JR|UxRTBwMEK2JO69VQ>? NXTvbIg3OTl7NUi3Oy=>
HT-29 MmHUS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? NHm0UGgxNjBzIN88[y=> NVvEWHdMPDhiaB?= MWjBcpRqeHKxbHnm[ZJifGm4ZTDhZ5Rqfmm2eR?= NHf0cFYzPzd6NES5
EMT6 NEmxWI1Iem:5dHigTY5pcWKrdHnvckBCe3OjeR?= M4C3WlAvPSEQvF2= MlXDNUBp NUPuNHo6UW6qaXLpeIlwdiCxZjDwdo9tcW[ncnH0bY9vKGK7IH3lZZN2emmwZzDmc5Ihe3W{dnn2bY5oKG[{YXP0bY9veyC5aYToJGVFPTBib3[gNE4xODBzIN88US=> NXLkPZk6PzR3Mk[3OC=>
H2981 MmLmR5l1d3SxeHnjJGF{e2G7 MojKTWM2OD1yLkWg{txO MXe3O|MyODJ|
LOX Ml\4R5l1d3SxeHnjJGF{e2G7 NGixSYxKSzVyPUCuNFQzKM7:TR?= NF;Nbo84QDV|M{Ox
C38 M4K4Z2N6fG:2b4jpZ{BCe3OjeR?= Mm\pTWM2OD1yLkCxJO69VQ>? NXmzUpoyQDB3N{K5NS=>
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A2780-DX5 M{S5ZWN6fG:2b4jpZ{BCe3OjeR?= Mm\uR5l1d3SxeHnjbZR6KGGpYXnud5Qh\G:6b4L1ZolkcW5vcnXzbZN1[W62IFGyO|gxNUS[NTD3bZRpKEmFNUCgc4YhOC5|NUeg{txO M3S1UVg5OzF5NUW=
MXF7 M{[5OGN6fG:2b4jpZ{BCe3OjeR?= NWC2cI9mSW62aYT1cY9zKGGldHn2bZR6KGGpYXnud5Qhe2Wwc3n0bZZmKE2[Rkege4l1cCCLQ{WwJI9nKDBwMEK4JO69VQ>? NGLaZ4k5QTZyNUW4
MXF7 NYDDe|dZS3m2b4TvfIlkKEG|c3H5 M4DY[GFvfGm2dX3vdkBi[3Srdnn0fUBi\2GrboP0JI1qfG:6YX70do9v\S2{ZYPpd5RidnRiTWjGO{B4cXSqIFnDOVAhd2ZiMD6wNlgh|ryP MXq4PVYxPTV6
MXF7 MVXDfZRwfG:6aXOgRZN{[Xl? MkPpRY51cXS3bX;yJIFkfGm4aYT5JIFo[Wmwc4Sg[I95d3K3YnnjbY4uemW|aYP0ZY51KE2[Rkege4l1cCCLQ{WwJI9nKDFwMUeyJO69VQ>? MUO4PVYxPTV6
WiDr NInLcnlEgXSxdH;4bYMhSXO|YYm= MmXkRYN1cX[rdImgZYdicW6|dDDz[Y5{cXSrdnWgW4lFeiClZXzsJJdqfGhiSVO1NEBw\iByLkC1N{DPxE1? NFXrNpc5QTZyNUW4
MCF NGT4SohHfW6ldHnvckBCe3OjeR?= NF\JVZpT\X[ncoPhcEBw\iCSLXfwMY1m\GmjdHXkJI12dHSrZIL1[{Bz\XOrc4ThcoNmKGG|c3Xzd4VlKGG|IHXubIFv[2WvZX70JIlvKGO7dH;0c5hq[2m2eTDv[kBi\HKrYX35Z4lv NWXnNlhmQDl6NEG1NS=>
C6 NW\aOHFMS3m2b4TvfIlkKEG|c3H5 NV70[GY3Oi53IH3nM41N NWPuPHVmPzJiaB?= NE\2OmJFVVOR NFrtXFBEgXSxdH;4bYNqfHliYXfhbY5{fCC{YYSgR|Yh[2WubIOgZZQhPTBidXevcWwhfG9iMj61JI1oN22O NVjPfoh[QDl6OE[wOC=>
C6 NF7EZWRHfW6ldHnvckBCe3OjeR?= MWWyMlUhdWdxbVy= MYm0JIg> M4nBSGROW09? M1HW[GlvcGmkaYTpc44hd2ZidIXieYxqdiCyb3z5cYVzcXqjdHnvci=> MWS4PVg5PjB2
C6 MYTDfZRwfG:6aXOgRZN{[Xl? NUSzW3BQOi53IH3nM41N NELxRlM2KGh? NXrESIF2TE2VTx?= M3yzOGN6fG:2b4jpZ4l1gSCjc4Pld5Nm\CCjczDj[YxtKHKnbHXhd4U> M4TOWlg6QDh4MES=
SKVLB MmfTR5l1d3SxeHnjJGF{e2G7 MlHBO|IhcA>? MUPJR|UxRTZwNUSg{txO NIDQUoc6ODB|NUKw
MCF7/VP16 NUXNcnBMS3m2b4TvfIlkKEG|c3H5 NULhe3RnPTBizsznM41N NEH5e2w4OiCq MojoTWM2OD1zND6yJO69VQ>? MljyPVAzOjd7Mh?=
CA755 NXrJRpB4T3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NFi3fmoyOCEQvF2= NVryc2JWPiCm NWXPe4x{UUN3ME2wMlAyPCEQvF2= NHXPdZg6PTJ4NUew
CHO M2jIR2dzd3e2aDDJcohq[mm2aX;uJGF{e2G7 M4rZRlExKM7:TR?= M3m5bVYh\A>? M4D0XGlEPTB;MD6wOkDPxE1? NInRWWM6PTJ4NUew
Panc02 M4nvS2dzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NF2zPGwyOCEQvF2= NW\ESpJyPiCm NHy5OZlKSzVyPUCuNFY2KM7:TR?= Ml[0PVUzPjV5MB?=
PC14 NVPVOYhwS3m2b4TvfIlkKEG|c3H5 M4Dsc|Qh\A>? MVXEUXNQ MlziTWM2OD1yLkK5JO69VQ>? MV65PFIzPTR{
HOP62 MWLDfZRwfG:6aXOgRZN{[Xl? M{H4W|czKGh? NYrOWIhPUUN3ME2wMlAxPCEQvF2= NWTE[5lTQTh5M{[2NS=>
SF-295 MV7DfZRwfG:6aXOgRZN{[Xl? Ml3UO|IhcA>? NUfne5AxUUN3ME2wMlA{PSEQvF2= MWS5PFc{PjZz
MDA-MB-361 MoCwR5l1d3SxeHnjJGF{e2G7 NYTxU2dDOSCq M{XFeWROW09? MnTTR5l1d3SxeHnjbZR6KGGpYXnud5QhVUSDLV3CMVM3OSCneIDy[ZN{cW6pIFzhZ3ohf2m2aDDJR|UxKG:oIECuNFEzKM7:TR?= M2DpUFExOzl3NEmw
MDA-MB-361 MoPIR5l1d3SxeHnjJGF{e2G7 NVf1bG1sOSCq NGPjTIhFVVOR NVn3fYxPS3m2b4TvfIlkcXS7IHHnZYlve3RiTVTBJG1DKDN4MTDlfJBz\XO|aX7nJINiemKxeInw[ZB1cWSjc3Wgd5REWEd{IIfpeIghUUN3MDDv[kAxNjBzODFOwG0> MWmxNFM6PTR7MB?=
CCRF-SB NFrWe2pIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= MXy0JIQ> MU\EUXNQ NYHNVW5YUUN3ME2wMlAyKM7:TR?= NI\sWXMyODRzMUS3Oi=>
CHO-K1 NYrlRVh1T3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NUfTUIhQPCCm MVfEUXNQ M4DVfGlEPTB;MD60JO69VQ>? MUCxNFQyOTR5Nh?=
KB NV\LUYRrT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= M1nUNlQh\A>? NXjU[|lMTE2VTx?= M4PuemFvfGmycn;sbYZmemG2aY\lJIFkfGm4aYT5JIFo[Wmwc4Sg[JJ2\y2{ZYPpd5RidnRiS1K3SEB4cXSqIFnDOVAhd2ZiMD62OUDPxE1? MWWxNFQyOTR5Nh?=
KB MmWxS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? NX\idVhjPCCm NXKxSVBkTE2VTx?= MlPoRY51cXC{b3zp[oVz[XSrdnWgZYN1cX[rdImgZYdicW6|dDDkdpVoNXKnc3nzeIFvfCCNQlPhcZB4cXSqIFnDOVAhd2ZiMD6wOkDPxE1? M3H3b|ExPDFzNEe2
KB NUj1[mJoT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= MVe0JIQ> MVfEUXNQ NXPOeY9ISW62aYDyc4xq\mW{YYTpeoUh[WO2aY\peJkh[WejaX7zeEBlenWpLYLld4l{fGGwdDDLRm1FWiC5aYToJGlEPTBib3[gNE42KM7:TR?= MoHlNVA1OTF2N{[=
KB MXzHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? NUjy[XJSPCCm M3n5NGROW09? M4fy[2FvfGmycn;sbYZmemG2aY\lJIFkfGm4aYT5JIFo[Wmwc4Sg[JJ2\y2{ZYPpd5RidnRiS1LWNlBEKHerdHigTWM2OCCxZjCwMlQh|ryP MmS0NVA1OTF2N{[=
HTB-54 NF7xNpFEgXSxdH;4bYMhSXO|YYm= MnXJNVAxKM7:TR?= NVTtcJdDUUN3ME2xMlEh|ryP NVvPeIdOOTB2N{[4OlE>
MEL-AC M4XpXGN6fG:2b4jpZ{BCe3OjeR?= MkfiNVAxKM7:TR?= NFXKdYRKSzVyPUGuNkDPxE1? NGj2eZAyODR5Nki2NS=>
DU145 NYCyN40xS3m2b4TvfIlkKEG|c3H5 NYXGVXhtPzJiaB?= MWHJR|UxRTBwMEWyPEDPxE1? NVHJcWk1OTB2N{myPFI>
K562R MWDDfZRwfG:6aXOgRZN{[Xl? Moi4O|IhcA>? M4fB[GlEPTB;MD6wNVU3KM7:TR?= MUixNFQ4QTJ6Mh?=
PACA-2 NHPGXWpEgXSxdH;4bYMhSXO|YYm= M3HkTVYh\A>? NVTTclZOTUR3ME2wMlAxPjNizszN M{LmWVExPDl6MkG0
3Y1 NWG2SFNMS3m2b4TvfIlkKEG|c3H5 M4H0SlczKGh? NH20c5hIUTVyPUCuNFA{QCEQvF2= MkXsNVA3QTF5MUC=
P388 Mm\5R5l1d3SxeHnjJGF{e2G7 MUC3NkBp MX;HTVUxRTBwMEGyJO69VQ>? NWe4fG5iOTB4OUG3NVA>
HMV-1 NXrtOZBUT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NIHzUotKSzVyPUCuNlgh|ryP MYCxNFY6QDR|Nh?=
MKN-1 NGe4d29Iem:5dHigTY5pcWKrdHnvckBCe3OjeR?= MXnJR|UxRTBwNkSg{txO Mn71NVA3QTh2M{[=
PC14 MVnHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? MniwTWM2OD1zLkmg{txO NWnlR25zOTB4OUi0N|Y>
T24 M172e2dzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NWnJdoFtUUN3ME2wMlY1KM7:TR?= MoHrNVA3QTh2M{[=
U937 M2[1ZWZ2dmO2aX;uJGF{e2G7 M2TaRVI1KGh? M2rJXGROW09? NVmxUm9SUW6qaXLpeJMhcW6lb4Lwc5JifGmxbjDv[kBcO0ifdHj5cYllcW6nIIfpeIghUUN3MDDv[kAxNjFizszN MlzHNVA4QDB7MUG=
H460pv8/eto Mo\pR5l1d3SxeHnjJGF{e2G7 MUWxNFAh|ryP M{W4blQ5KGh? MmLSV4FtcW6n M1O3U2lEPTB;MD6wNkDPxE1? MV:xNFc5ODlzMx?=
H460pv8 M1z5eGN6fG:2b4jpZ{BCe3OjeR?= MnzZNVAxKM7:TR?= NF\pS2E1QCCq NGTmPYFU[WyrbnW= M{HYWWlEPTB;MD6wNFQh|ryP MmnqNVA4QDB7MUO=
MDA-231 MWLDfZRwfG:6aXOgRZN{[Xl? NHnaWZMyODBizszN NEW0fmI1QCCq MXHTZYxqdmV? NEPMRoNEgXSxdH;4bYNqfHliYXfhbY5{fCCPRFGtNlMyKGOnbHygLGVTNSyHR1\SL{xufXSjboSgdFU{MSC5aYToJGlEPTBib3[gNE4xODZizszN MnLRNVA4QDB7MUO=
MDA-468 NHm1OXVEgXSxdH;4bYMhSXO|YYm= MYKxNFAh|ryP MWi0PEBp NVrGT|djW2GuaX7l Mlf2R5l1d3SxeHnjbZR6KGGpYXnud5QhVUSDLUS2PEBk\WyuIDjFVk0tKGGvcHzp[olm\CCHR1\SMEBufXSjboSgdFU{MSC5aYToJGlEPTBib3[gNE4xODVizszN MlXxNVA4QDB7MUO=
NCI-H226 MXHDfZRwfG:6aXOgRZN{[Xl? MoHSNVAxKM7:TR?= MorjOFghcA>? M3zx[nNidGmwZR?= NIHwNZlEgXSxdH;4bYNqfHliYXfhbY5{fCCQQ1mtTFIzPiClZXzsJEhufXSjboSgdFU{MSC5aYToJGlEPTBib3[gNE4xODhizszN NFHUOFgyODd6MEmxNy=>
NCI-H322 MULDfZRwfG:6aXOgRZN{[Xl? MlO4NVAxKM7:TR?= NHHzOIU1QCCq NYPl[GVyW2GuaX7l MmWyR5l1d3SxeHnjbZR6KGGpYXnud5QhVkOLLVizNlIh[2WubDCocZV1[W62IIC1N{khf2m2aDDJR|UxKG:oIECuNFMh|ryP MoC2NVA4QDB7MUO=
NCI-H358 NVnM[Y9bS3m2b4TvfIlkKEG|c3H5 MYqxNFAh|ryP NGH4d201QCCq MoP6V4FtcW6n NVvBTY1GS3m2b4TvfIlkcXS7IHHnZYlve3RiTlPJMWg{PThiY3XscEApdXW2YX70JJA2Oylid3n0bEBKSzVyIH;mJFAvOTNizszN MlWzNVA4QDB7MUO=
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SKBR-3 NWqzVIx7S3m2b4TvfIlkKEG|c3H5 MYGxNFAh|ryP MmLPOFghcA>? M4TzPXNidGmwZR?= Ml;HR5l1d3SxeHnjbZR6KGGpYXnud5QhW0uEUj2zJINmdGxiKFXSMYFueGyrZnnl[EBmekJ{LH31eIFvfCCyNUOpJJdqfGhiSVO1NEBw\iByLkCyJO69VQ>? NEnrUVkyODd6MEmxNy=>
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L1210 M1zrbmN6fG:2b4jpZ{BCe3OjeR?= NWfDOZVJUUN3ME2wMlAzPSEQvF2= NF7DZ5AyODh7MEG2Oy=>
D40 NYnFO3dtS3m2b4TvfIlkKEG|c3H5 MUSyOEBp NGno[|hFVVOR NX;TV45IUUN3ME2xMlE4OiEQvF2= NVLlVVh{OTB7NU[yNVQ>
OVCAR-3 MUDDfZRwfG:6aXOgRZN{[Xl? MVeyOEBp M3:2TmROW09? NWDtVlJVUUN3ME2wMlA{PSEQvF2= NYn3SVNxOTB7NU[yNVQ>
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RT-112 Mn64S5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? M1zBWWlEPTB;M{KuPVIhdk1? MWDTRW5ITVJ?
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NCI-H719 MX\Hdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? MUPJR|UxRTN7Lk[1JI5O M1HhcXNCVkeHUh?=
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PA-1 NFHYU3dIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= M3LQVWlEPTB;NESuOFghdk1? M4LXfnNCVkeHUh?=
CAL-85-1 MX\Hdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? M2HlfmlEPTB;NESuOVIhdk1? NGjJUZVUSU6JRWK=
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NUGC-3 MVLHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? NVHScGo5UUN3ME20OU4zKG6P MVfTRW5ITVJ?
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NCI-H209 MVLHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? M33TbGlEPTB;NEiuO|Mhdk1? MljZV2FPT0WU
MC-CAR NXnu[FJ2T3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= Mk\STWM2OD12OD63OEBvVQ>? MVnTRW5ITVJ?
NCI-H661 MYXHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? M2K2fGlEPTB;NEmuNFMhdk1? NXX3cmVCW0GQR1XS
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GP5d NIH6dHFIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= M3KyWGlEPTB;NEmuNVIhdk1? MlrVV2FPT0WU
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ACHN Mn;YS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MWjJR|UxRTR7LkO0JI5O NYn1W2s6W0GQR1XS
NCI-H2087 MoPJS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? NV\tTm5kUUN3ME20PU41OiCwTR?= M1nIUXNCVkeHUh?=
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NCI-H526 MYfHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? NVnNWm5wUUN3ME20PU46PiCwTR?= NX3Tbo0yW0GQR1XS
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KYSE-140 NF\rVVRIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NI\D[FhKSzVyPUWwMlQzKG6P MVPTRW5ITVJ?
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CAPAN-1 NVfqeHNoT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= M2PlbmlEPTB;NUGuO|Yhdk1? MV;TRW5ITVJ?
NCI-H2009 Mo[4S5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? NH;XU|NKSzVyPUWxMlc3KG6P NFfkV3BUSU6JRWK=
NCI-H522 MVLHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? MV7JR|UxRTVzLkmzJI5O M{XGVXNCVkeHUh?=
HuP-T4 MULHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? MoHlTWM2OD13Mj6yNkBvVQ>? NVvC[GY{W0GQR1XS
BCPAP NEXkbpRIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NGq0Z2VKSzVyPUWyMlUhdk1? MWPTRW5ITVJ?
NCI-H1734 MofhS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MUPJR|UxRTV|IH7N NEnvb4JUSU6JRWK=
SK-LMS-1 M3HiT2dzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NFyxcYhKSzVyPUWzMlIzKG6P M4e1c3NCVkeHUh?=
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RPMI-8402 Mom1S5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? NV3qcFB4UUN3ME21N{45PiCwTR?= M4nRWnNCVkeHUh?=
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CHP-126 NI[0NlNIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= M4T5cGlEPTB;NUmuNlQhdk1? MYDTRW5ITVJ?
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CAMG MlW3S5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MVnJR|UxRTV7Lkm2JI5O MoOyV2FPT0WU
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OVCAR-8 MkS4S5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? M17kOmlEPTB;NkGuPVIhdk1? MlvqV2FPT0WU
HL-60 NVTafY1ST3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NIK2OlBKSzVyPU[yMlU3KG6P NYDLbVFKW0GQR1XS
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HCC2157 NHH6TJNIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NVPOV5cxUUN3ME22N{46PSCwTR?= NI\relNUSU6JRWK=
CTB-1 NF;JNWxIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NVfLSm04UUN3ME22OFAyQSCwTR?= NF60T3hUSU6JRWK=
NCI-H1437 NV\YcoFKT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= MVjJR|UxRTZ2Lk[0JI5O MYjTRW5ITVJ?
U251 NYTDZXJVT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= MYfJR|UxRTZ2Lki5JI5O MnXnV2FPT0WU
ALL-PO NVrjWolyT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= MkXkTWM2OD14NT6wN{BvVQ>? M{DNU3NCVkeHUh?=
NCI-SNU-1 NWX0SG5kT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= MojmTWM2OD14NT64OkBvVQ>? Ml;tV2FPT0WU
RPMI-6666 MUPHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? MmPKTWM2OD14NT65PUBvVQ>? MYDTRW5ITVJ?
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PF-382 MlrwS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? M33qXGlEPTB;NkeuNVchdk1? MXTTRW5ITVJ?
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LU-134-A M2PWe2dzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NVT6dHdTUUN3ME22O{43QCCwTR?= MlriV2FPT0WU
CAL-33 M4S5N2dzd3e2aDDJcohq[mm2aX;uJGF{e2G7 M4XsOmlEPTB;NkeuPFchdk1? NX\wWJlXW0GQR1XS
MC-IXC M{nofWdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NIjuRVhKSzVyPU[3Mlkhdk1? NX;kXHQzW0GQR1XS
CPC-N MWTHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? NXvqdGF1UUN3ME22PE41KG6P NX3kWFlqW0GQR1XS
A2780 NWPpOoxST3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= M{\rOmlEPTB;NkiuO|khdk1? NU\ORY0yW0GQR1XS
Daudi MojPS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? NHvsflZKSzVyPU[4Mlk3KG6P MkTTV2FPT0WU
GI-1 MXHHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? MkO0TWM2OD14OT62OUBvVQ>? NYjhRXB5W0GQR1XS
SW962 M1\tXGdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 MUHJR|UxRTZ7Lkm1JI5O MVnTRW5ITVJ?
MFE-296 M3\Je2dzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NUnUXJdTUUN3ME23NE41QSCwTR?= Mmn3V2FPT0WU
H4 M1jkeWdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NWToeY9RUUN3ME23NU42PiCwTR?= MWLTRW5ITVJ?
AN3-CA MkXVS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? Mn7rTWM2OD15Mj6zNkBvVQ>? M3L1bXNCVkeHUh?=
HCC1599 MUTHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? NH7YZ4JKSzVyPUeyMlU1KG6P MUTTRW5ITVJ?
HuCCT1 NYLwN416T3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= M3\pVmlEPTB;N{KuPVMhdk1? MW\TRW5ITVJ?
Calu-1 NHv0dWNIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= M4S4Z2lEPTB;N{OuOkBvVQ>? MYLTRW5ITVJ?
DU-145 M3vKTWdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 M{TMTGlEPTB;N{OuO|Mhdk1? MUPTRW5ITVJ?
IST-SL2 MoPqS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? M3\rWWlEPTB;N{OuPFEhdk1? MYXTRW5ITVJ?
HSC-3 M{PEeGdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NFXiZVVKSzVyPUe0MlU{KG6P M4rxR3NCVkeHUh?=
HCC1806 M4f0dmdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 MWHJR|UxRTd2Lkm2JI5O MojPV2FPT0WU
VM-CUB-1 NXO5b4o1T3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= MYPJR|UxRTd3LkO2JI5O NYi1VmVpW0GQR1XS
HSC-4 M17rV2dzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NFjBeWFKSzVyPUe1Mlc3KG6P MXnTRW5ITVJ?
NH-12 MW\Hdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? MoW5TWM2OD15NjDuUS=> NGTBTFZUSU6JRWK=
MDA-MB-468 MVHHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? MlTwTWM2OD15Nj6xPEBvVQ>? NVzpOodtW0GQR1XS
TUR NH\yZ|hIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NEC5N2dKSzVyPUe2MlMzKG6P M1\xSnNCVkeHUh?=
TE-1 MlXFS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MYnJR|UxRTd4LkO1JI5O NIPXeldUSU6JRWK=
CMK NXXUVZBvT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NFP5dVNKSzVyPUe3MlQzKG6P MVrTRW5ITVJ?
LB996-RCC NU\oSY1uT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NFPGNJFKSzVyPUe4MlQ2KG6P MkXtV2FPT0WU
NCI-H1650 M3TBOmdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NVPLSFA3UUN3ME23PE43OiCwTR?= M2Pxd3NCVkeHUh?=
DMS-273 NUn5RlhPT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= MVrJR|UxRTd6Lkmgcm0> M2nsO3NCVkeHUh?=
NOS-1 NWLUc4RQT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= M3TLO2lEPTB;N{muNVQhdk1? M3LCeHNCVkeHUh?=
NB69 M3nLTWdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NH7XZllKSzVyPUe5MlIhdk1? NUTtT5JpW0GQR1XS
SUP-T1 Mm\hS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? NHOxWYlKSzVyPUe5MlczKG6P NV3FOFJ3W0GQR1XS
A172 NXfHe2pyT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NYXJcHM1UUN3ME24NE42PSCwTR?= NGHSS|VUSU6JRWK=
TE-12 MkGyS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? M4jlbGlEPTB;OEGuNFYhdk1? NVX6[oFmW0GQR1XS
MKN45 M3rOdWdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 M2PaVWlEPTB;OEGuOVEhdk1? M{K4fnNCVkeHUh?=
LoVo MYLHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? M2T1U2lEPTB;OEGuPFIhdk1? Mn\rV2FPT0WU
SW1573 M3;6Smdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 MoLUTWM2OD16Mj64NUBvVQ>? MlL6V2FPT0WU
ETK-1 MYfHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? NXrYTpVSUUN3ME24N{4xOSCwTR?= M1z5UHNCVkeHUh?=
ABC-1 MmexS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? M3m4XmlEPTB;OEOuOFUhdk1? M3fpeHNCVkeHUh?=
COLO-668 NHnWNFFIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= M4DI[WlEPTB;OESuOFchdk1? NF3a[o1USU6JRWK=
UM-UC-3 M3vlNWdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 MYTJR|UxRTh4LkCyJI5O NU\HdIpJW0GQR1XS
BC-1 M{TSZWdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 M1vmZWlEPTB;OE[uO|Yhdk1? MWPTRW5ITVJ?
PANC-10-05 NIHYcZNIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NVzkc5UyUUN3ME24PE41PSCwTR?= NVu0SGI{W0GQR1XS
ES3 NGn1elJIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= MWXJR|UxRTh7LkS4JI5O MlLRV2FPT0WU
TE-441-T M{\VWGdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 M{fY[mlEPTB;OEmuPFIhdk1? M1faTHNCVkeHUh?=
KM-H2 MXrHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? M4K4SGlEPTB;OUCuOlghdk1? M32zXHNCVkeHUh?=
SH-4 Ml\HS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? NWPNR2VXUUN3ME25Nk4yOSCwTR?= NV7pW2V[W0GQR1XS
SF268 MY\Hdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? M2PDb2lEPTB;OUKuOFIhdk1? MX;TRW5ITVJ?
VMRC-RCZ NH;GNHdIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NEeweXNKSzVyPUmzMlI3KG6P MUTTRW5ITVJ?
GI-ME-N NGnp[ItIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= MXzJR|UxRTl|LkOzJI5O M3WxNXNCVkeHUh?=
JEG-3 M1XyU2dzd3e2aDDJcohq[mm2aX;uJGF{e2G7 MXHJR|UxRTl3LkGyJI5O NV3aem1tW0GQR1XS
J-RT3-T3-5 NXrEcJhDT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NHvjUIpKSzVyPUm2MlMyKG6P NEGx[GtUSU6JRWK=
K5 MUPHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? MonKTWM2OD17Nj65JI5O MWnTRW5ITVJ?
EFO-27 MljlS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? NXi3OXZQUUN3ME25O{41PCCwTR?= M1:xSnNCVkeHUh?=
SW1783 NEHjcnBIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= MlTVTWM2OD17Nz65PUBvVQ>? MmHIV2FPT0WU
CAL-39 M{LMWWdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 MmqyTWM2OD17OD6yOEBvVQ>? MUHTRW5ITVJ?
LS-441N NFixV|BIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= M2D3Z2lEPTB;OUmuNFYhdk1? MnL2V2FPT0WU
G-402 NUjOeWlHT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NW[wenNNUUN3ME25PU4xQSCwTR?= NXX4eZJJW0GQR1XS
MES-SA M3XkWWdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 MX\JR|UxRTl7LkWzJI5O M1fXR3NCVkeHUh?=
FADU M4DzRmdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NH3QS|dKSzVyPUGwNk4yQCCwTR?= NYKwc|YzW0GQR1XS
DJM-1 MY\Hdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? MWjJR|UxRTFyMj6yOUBvVQ>? MUTTRW5ITVJ?
SU-DHL-1 MmfaS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MnPXTWM2OD1zMEKuOUBvVQ>? MWTTRW5ITVJ?
KYSE-410 NGTHPVhIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NHvDVYNKSzVyPUGwN{41PiCwTR?= MWfTRW5ITVJ?
NCI-H1618 NVHFXJI6T3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NHfFTGtKSzVyPUGwOE4{PSCwTR?= M2jz[XNCVkeHUh?=
AU565 NG\3UVBIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= MmPZTWM2OD1zMESuOVEhdk1? NIDYPHdUSU6JRWK=
SF126 MV\Hdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? MW\JR|UxRTFyND61PEBvVQ>? NI\NUFhUSU6JRWK=
MMAC-SF MmLES5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? M1e1TWlEPTB;MUC2MlQ5KG6P NHOyT5lUSU6JRWK=
ChaGo-K-1 MWXHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? NYDh[lFNUUN3ME2xNFcvQTVibl2= NI\yeGdUSU6JRWK=
NCI-H596 NUjPdG44T3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= MlHmTWM2OD1zMEiuNFEhdk1? NHzaUYtUSU6JRWK=
LXF-289 Mmi3S5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? NE\u[JNKSzVyPUGwPU4zPCCwTR?= NXz5bI54W0GQR1XS
HCC1569 NFrXN4dIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= MnTSTWM2OD1zMEmuN|Qhdk1? MlHsV2FPT0WU
NCI-H2170 MljWS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MVjJR|UxRTFyOT65NkBvVQ>? MoTJV2FPT0WU
ARH-77 M{C3cmdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NF\ncJRKSzVyPUGwPU46QSCwTR?= NGDseI9USU6JRWK=
BOKU NW\OOXQ1T3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= M{DwNWlEPTB;MUGwMlg4KG6P MnLEV2FPT0WU
SJSA-1 NHL0dlRIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= M{DpWWlEPTB;MUGxMlA2KG6P NEKxbWxUSU6JRWK=
SW626 MUHHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? MnTyTWM2OD1zMUGuO|Ehdk1? MXTTRW5ITVJ?
EHEB MXHHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? NFTwN25KSzVyPUGxNk42QSCwTR?= NHLkclNUSU6JRWK=
TE-10 NF3xRXFIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NH[1bVJKSzVyPUGxNk43QCCwTR?= NYS1Um01W0GQR1XS
MZ7-mel NH[zPIZIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NWjBVnk4UUN3ME2xNVIvQDRibl2= NGTwUHJUSU6JRWK=
SAS MWXHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? NXjMV3RvUUN3ME2xNVQvPDVibl2= MYHTRW5ITVJ?
TK10 M4\qW2dzd3e2aDDJcohq[mm2aX;uJGF{e2G7 M3nVUmlEPTB;MUG0MlYhdk1? NWf4S3ZRW0GQR1XS
SW13 NEfVbItIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= MWjJR|UxRTFzNT6yOkBvVQ>? MVrTRW5ITVJ?
HCC1937 Mn3pS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? Mn;yTWM2OD1zMUWuPFQhdk1? NGLjS45USU6JRWK=
SK-NEP-1 MmTYS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MmfnTWM2OD1zMU[uNlYhdk1? Mom2V2FPT0WU
OVCAR-5 MV\Hdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? M2rtVGlEPTB;MUG2MlgyKG6P M37zbHNCVkeHUh?=
SW837 NF\hOJlIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= M4DvNWlEPTB;MUG3Mlk2KG6P M3rEcXNCVkeHUh?=
BFTC-909 NHzLb|BIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= MkGyTWM2OD1zMUiuOFghdk1? NF7jOXNUSU6JRWK=
SW872 MkS1S5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? NVfZPIVZUUN3ME2xNlAvQDFibl2= NYLKNW1[W0GQR1XS
SF539 NUH6O25mT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= MofQTWM2OD1zMkGuO|Ihdk1? MmD6V2FPT0WU
MLMA MknWS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? M{f4UmlEPTB;MUKyMlA5KG6P MV3TRW5ITVJ?
BL-41 M4DSWGdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 MoHrTWM2OD1zMkKuNlIhdk1? NHTJPHpUSU6JRWK=
LB647-SCLC NVXpc45vT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NIPPeHJKSzVyPUGyN{4{PSCwTR?= NFfRbYZUSU6JRWK=
NCI-H1703 NFm0cItIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= M4XLZmlEPTB;MUK2MlQzKG6P NXHzXY1DW0GQR1XS
KURAMOCHI MYPHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? MX3JR|UxRTF{Nj63OkBvVQ>? NWO5WIIzW0GQR1XS
ATN-1 NHj3R3FIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NY\tSHVsUUN3ME2xNlcvPyCwTR?= Ml;OV2FPT0WU
SK-CO-1 NYnndnlZT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= MlqwTWM2OD1zMkmuNlEhdk1? NWn0U5JHW0GQR1XS
RPMI-7951 NWTGS4h6T3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NHThOI9KSzVyPUGzNE4yPCCwTR?= MYLTRW5ITVJ?
NCI-H1648 NH7CdYxIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NVnQZ3V2UUN3ME2xN|EvQTRibl2= NXS2dHQ2W0GQR1XS
NCI-H64 NV7uU4J3T3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NIPNXZdKSzVyPUGzNk43PSCwTR?= NGrmW4lUSU6JRWK=
HT-3 NFr5WZJIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= MV7JR|UxRTF|Mz6wOEBvVQ>? M1TKPXNCVkeHUh?=
NCI-H1770 NVHFOW1rT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= MWTJR|UxRTF|Mz6yNUBvVQ>? MV;TRW5ITVJ?
NB13 Mn:0S5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MVnJR|UxRTF|ND61OUBvVQ>? MXrTRW5ITVJ?
NCI-H747 NI[5R2pIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NGTMOJRKSzVyPUGzOU4xOiCwTR?= MkL2V2FPT0WU
ML-2 Mn;GS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? Mmf1TWM2OD1zM{WuNVYhdk1? NFnS[HRUSU6JRWK=
CA46 NWDwXo9NT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NWPsRYJGUUN3ME2xN|YvQDhibl2= MWrTRW5ITVJ?
ES6 M{nDRWdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NUjP[GtiUUN3ME2xN|cvOTJibl2= MofxV2FPT0WU
JiyoyeP-2003 M2KzUmdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NF;vfHRKSzVyPUGzO{45KG6P NVXrWpRwW0GQR1XS
NMC-G1 MoHFS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MUfJR|UxRTF|OT6xN{BvVQ>? NWiyOnRLW0GQR1XS
U-698-M MYnHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? MoSyTWM2OD1zM{muOUBvVQ>? NED6[|ZUSU6JRWK=
LU-99A M3\ZO2dzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NIrDOmZKSzVyPUG0Ok42PSCwTR?= NEH6No9USU6JRWK=
NCI-H748 MWTHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? M2TVfWlEPTB;MUS3MlMyKG6P M17lbXNCVkeHUh?=
SK-MEL-3 MmnJS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? NHi4fI9KSzVyPUG0O{43OSCwTR?= MVjTRW5ITVJ?
SNB75 NE\DTZpIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= MVHJR|UxRTF2OD62OUBvVQ>? NVLnR4lzW0GQR1XS
BB65-RCC NXjxVIQ2T3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NHzqRolKSzVyPUG0PU4{OSCwTR?= MXXTRW5ITVJ?
NCI-H1355 MXzHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? M1iwbWlEPTB;MUWyMlI1KG6P NH7xUlRUSU6JRWK=
SCC-25 MmP3S5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? NVvseJlnUUN3ME2xOVMvPzNibl2= M2rZWHNCVkeHUh?=
OAW-42 MXfHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? Ml;NTWM2OD1zNUOuPFQhdk1? M1X4c3NCVkeHUh?=
MONO-MAC-6 MVPHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? M3HvWmlEPTB;MUW0MlM3KG6P NH;QfHNUSU6JRWK=
WSU-NHL NHzGfnBIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= MUjJR|UxRTF3ND61PEBvVQ>? NFXjbGZUSU6JRWK=
SNU-423 Mnz6S5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? M{\KZmlEPTB;MUW1MlM1KG6P MVHTRW5ITVJ?
SBC-1 MWrHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? M4nKPGlEPTB;MUW2MlQhdk1? MlPZV2FPT0WU
OVCAR-4 NWXScIl7T3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NHXzZoVKSzVyPUG1Ok44QCCwTR?= MX\TRW5ITVJ?
NCI-H2347 MVLHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? NEjSUXNKSzVyPUG1PE4{PCCwTR?= NEC3WFRUSU6JRWK=
CAMA-1 MnLXS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? NFfReXNKSzVyPUG1PU4{OyCwTR?= NFPSNldUSU6JRWK=
GDM-1 NHnXXmdIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NEDSW|VKSzVyPUG1PU44KG6P M{TiV3NCVkeHUh?=
KNS-81-FD NV7RfI1DT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NWm0elg5UUN3ME2xOlAvOzJibl2= NVP5UVJiW0GQR1XS
no-10 MlnPS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MlzCTWM2OD1zNkCuN|ghdk1? NHn0flRUSU6JRWK=
NCI-H2052 Ml\jS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MVTJR|UxRTF4MD60O{BvVQ>? Mo\4V2FPT0WU
DB Ml7zS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? M3rBdmlEPTB;MU[xMlcyKG6P MXLTRW5ITVJ?
A4-Fuk Mm\ES5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? NXrUNXc2UUN3ME2xOlIvPDhibl2= M3nzb3NCVkeHUh?=
HCE-T MnjoS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MnzlTWM2OD1zNkSuPFchdk1? M2TGUHNCVkeHUh?=
HuP-T3 MoO2S5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? M3XwUWlEPTB;MU[1MlU2KG6P NGr4NWpUSU6JRWK=
BC-3 NGHjZnNIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= M1HCO2lEPTB;MU[1Mlg3KG6P MVzTRW5ITVJ?
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A704 NEfqRlJIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= MU\JR|UxRTJwMkmxN|Uh|ryP NWP5O4Z7W0GQR1XS
EVSA-T NH;G[pJIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= M1:1bGlEPTB;Mj6zNFA5QSEQvF2= MljZV2FPT0WU
HCT-15 M4PPWWdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NWXYc3J4UUN3ME2yMlM2PDZ4IN88US=> NWq3fot7W0GQR1XS
HuO-3N1 MnXIS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? NFzodZRKSzVyPUKuN|Y2QDNizszN MWDTRW5ITVJ?
GMS-10 NV7EWodjT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= M4DOUGlEPTB;Mj6zPVc{QCEQvF2= M1Xk[3NCVkeHUh?=
TGBC24TKB MUnHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? NWPZPYp3UUN3ME2yMlQyPDJ7IN88US=> NF7VclVUSU6JRWK=
C2BBe1 MojZS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MV;JR|UxRTJwNUGzNlgh|ryP M4Dkc3NCVkeHUh?=
SK-N-DZ NWXXbItDT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= MofsTWM2OD1{LkW2OVkzKM7:TR?= MofoV2FPT0WU
SK-N-AS NHizSGRIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= M1zKb2lEPTB;Mj63N|AyPSEQvF2= NF\sWmRUSU6JRWK=
T98G MlPDS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? M4TtdWlEPTB;Mj64NFQxOSEQvF2= NUjLXmdxW0GQR1XS
DMS-79 NHq2bFRIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= M4TPPGlEPTB;Mj65NFk5QCEQvF2= Ml31V2FPT0WU
SNU-475 Mnj5S5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MVPJR|UxRTJwOUK1O|Ih|ryP NVHaNmxzW0GQR1XS
COLO-792 M{m4dWdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 M2\LS2lEPTB;Mz6wNlg4KM7:TR?= MYjTRW5ITVJ?
YAPC NGe0d3pIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NH7oOolKSzVyPUOuN|I5OzJizszN NHrFfFZUSU6JRWK=
UACC-812 MXrHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? MVTJR|UxRTNwM{O3N|gh|ryP NIXBUmpUSU6JRWK=
Mewo M2fLXmdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NGS2Om9KSzVyPUOuOFYxQDZizszN NYqzS5BnW0GQR1XS
COLO-824 NEfO[3BIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NVOxbIFiUUN3ME2zMlU4Ozd6IN88US=> NYXKO205W0GQR1XS
SCC-9 NV7GWlluT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NVHtW5F6UUN3ME2zMlkyOzB7IN88US=> NGfuO5dUSU6JRWK=
CP50-MEL-B Ml\nS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? M4S2bGlEPTB;Mz65PFcxOyEQvF2= M2Lx[XNCVkeHUh?=
NCI-H345 NEHZSpdIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NWG4fWJnUUN3ME20MlAyOTd2IN88US=> NX[xdpJ4W0GQR1XS
COR-L88 MUDHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? NWjNOZRnUUN3ME20MlM6PThizszN MmT5V2FPT0WU
RCM-1 M3;mS2dzd3e2aDDJcohq[mm2aX;uJGF{e2G7 MmDMTWM2OD12LkS5NlczKM7:TR?= MV3TRW5ITVJ?
JVM-3 MmrES5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? M{jPSmlEPTB;ND62NFYyQCEQvF2= MXnTRW5ITVJ?
ECC4 MmruS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? NH;CW4ZKSzVyPUSuO|Y2PDFizszN M2nS[XNCVkeHUh?=
MDA-MB-453 MkToS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MYrJR|UxRTRwOEWxN|Qh|ryP Mmm4V2FPT0WU
SK-N-FI M4fNd2dzd3e2aDDJcohq[mm2aX;uJGF{e2G7 M3i2TGlEPTB;NT6yNlg4PyEQvF2= NWDobI9QW0GQR1XS
D-502MG NFX4dm9Iem:5dHigTY5pcWKrdHnvckBCe3OjeR?= M4\obGlEPTB;NT6yOFI3OiEQvF2= NWjwOodJW0GQR1XS
NCI-H2227 MVjHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? MlrmTWM2OD13LkO2NlMyKM7:TR?= M37NdnNCVkeHUh?=
DMS-53 NWG1d2lOT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NVy1OIVVUUN3ME22MlE4OTB4IN88US=> NHznZXVUSU6JRWK=
LB771-HNC NYq2TYpQT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= MUfJR|UxRTZwNE[4NFYh|ryP M1\lUXNCVkeHUh?=
BB49-HNC Mm\CS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? Mn7rTWM2OD15LkSxO|kyKM7:TR?= NXnyW2ppW0GQR1XS
MDA-MB-415 MULHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? Mme4TWM2OD15LkW3N|A{KM7:TR?= M4LhcXNCVkeHUh?=
TALL-1 MmD6S5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MmjMTWM2OD15Lkm2PFgh|ryP M4LWTnNCVkeHUh?=
HCC1395 NXf4WmtiT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NXjofWRUUUN3ME24MlE2OTJ{IN88US=> MofrV2FPT0WU
EFE-184 MWrHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? MULJR|UxRThwM{eyNVYh|ryP MnvEV2FPT0WU
EC-GI-10 NE[1XmtIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= MXPJR|UxRThwNki2PFYh|ryP NXP3S3czW0GQR1XS
TT MYnHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? M37ucWlEPTB;OT6wOlk3PiEQvF2= M{\jZ3NCVkeHUh?=
U-2-OS NX;VT4ZTT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= M1W3OWlEPTB;OT64NVM6OyEQvF2= NFW0enVUSU6JRWK=
SHP-77 MkCzS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? NILxZo1KSzVyPUmuPVAzQSEQvF2= MojFV2FPT0WU
HCC1143 M{T6T2dzd3e2aDDJcohq[mm2aX;uJGF{e2G7 Mn7MTWM2OD1zMD60O|k4KM7:TR?= NYTPbJd1W0GQR1XS
A498 NGXXSJBIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= MkLDTWM2OD1zOD6yPVc3KM7:TR?= M2\ncnNCVkeHUh?=
LS-513 Mn3jS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MUDJR|UxRTF6Lk[wPVMh|ryP NUjMdY01W0GQR1XS
K052 NUj3[FV2T3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NGDXW4ZKSzVyPUKxMlQ1OThizszN MVvTRW5ITVJ?
SiHa Mk\BS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MYHJR|UxRTJ|LkOzO|Eh|ryP MV3TRW5ITVJ?
RCC10RGB M2mybmdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 MUjJR|UxRTNyLkC2NVEh|ryP NUnXNmQyW0GQR1XS
NCI-SNU-16 MmixS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? NVXQW2FbUUN3ME2zNU4yQDN4IN88US=> MYnTRW5ITVJ?
SNU-C1 NEXQZo9Iem:5dHigTY5pcWKrdHnvckBCe3OjeR?= Ml\QTWM2OD1|Mj60NVc2KM7:TR?= MVjTRW5ITVJ?
C32 M1rRdWdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 MYDJR|UxRTN{Lki3NkDPxE1? M3LhOXNCVkeHUh?=
SW684 NYOwXG93T3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NIH4[mpKSzVyPUO0MlE2PjFizszN MXvTRW5ITVJ?
SK-MEL-28 NVzKb|dYT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= Mm\FTWM2OD1|NT61N|c4KM7:TR?= M4jqbnNCVkeHUh?=
SK-MEL-1 NGrXNmJIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NX7MNmlRUUN3ME2zOk44PTR5IN88US=> NYP5WYw3W0GQR1XS
NCI-H720 MVLHdo94fGhiSX7obYJqfGmxbjDBd5NigQ>? Mle4TWM2OD12MT65O|I3KM7:TR?= M{jRNnNCVkeHUh?=
P31-FUJ MlTxS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MVnJR|UxRTR2LkOyPFQh|ryP MlLxV2FPT0WU
NCI-H524 MmjJS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? M4T0fmlEPTB;NEiuPFI1QCEQvF2= M2\JUHNCVkeHUh?=

... Click to View More Cell Line Experimental Data

Assay
Methods Test Index PMID
Western blot
POU5F1 / SOX2 / NANOG; 

PubMed: 27929731     


NT2/D1 cells treated with 10 nM of doxorubicin were subjected to WB analysis for pluripotency factors (POU5F1, NANOG, SOX2) and differentiation markers (TUBB3).

ATG5 / ATG7 / SQSTM1 / LC3A-II / LC3B-II / p-mTOR; 

PubMed: 27929731     


NT2/D1 cells treated with 10 nM of doxorubicin were subjected to WB analysis for autophagy markers (ATG5, ATG7, SQSTM1, LC3A-II, LC3B-II and p-MTOR). 

P62 / LC3II; 

PubMed: 28208617     


(A,B) Doxorubicin induces autophagy in pancreatic cancer cells. Western blot analysis of LC3-II and p62 protein levels in Mia PaCa-2 and Panc-1 cell lines treated with indicated concentrations of doxorubicin for 24 h, or treated with 2.5 μM doxorubicin for indicated times.

p-AKT(T308) / p-Akt(S473) / Akt / p-PRAS40(T246) / PRAS40 / p-H2A.X(S139); 

PubMed: 26027929     


MCF10A cells were serum-starved and treated with (A) 2 μM doxorubicin over a 10 hour time course.

27929731 28208617 26027929
Growth inhibition assay
Cell viability; 

PubMed: 25871400     


Salinomycin enhances the cytotoxicity of doxorubicin in HCC cellsRelative cell viability (mean ± SD) for salinomycin (black), doxorubicin (blue) and doxorubicin plus salinomycin (red) in HuH-7, HepG2, SNU-449 and SNU-387 cells.

25871400
Immunofluorescence
LC3; 

PubMed: 24970805     


Doxorubicin induces GFP-LC3 puncta formation in hepatocellular carcinoma cells. SK-Hep1 cells were treated with doxorubicin (2.5 μM) or CQ (10 μM) plus doxorubicin for 7 h and cells were examined with a confocal microscope for GFP-LC3 punctuation/aggregation.

24970805
ELISA
OPN; 

PubMed: 24963635     


A549 were exposed to 50 nM doxorubicin or PBS for 48 h. OPN concentrations in cell culture media were determined by ELISA.

24963635
In vivo In vivo, Doxorubicin in combination with adenoviral MnSOD (AdMnSOD) plus 1,3-bis(2-chloroethyl)-1-nitrosourea (BCNU) has the greatest effect in decreasing the volumes of MB231 tumors and prolonging survival of mice. [1] Although its use is limited by the chronic and acute toxic side effects it produces, Doxorubicin is essential in treating breast and oesophageal carcinomas, solid tumours in childhood, osteosarcomas, Kaposi's sarcoma, soft tissue sarcomas, and Hodgkin and non-Hodgkin lymphomas. [2]

Protocol

Animal Research:[1]
- Collapse
  • Animal Models: Female athymic nude mice injected s.c. with MB231 cells
  • Formulation: Dissolved in DMSO, and diluted in saline
  • Dosages: 3 mg/kg/day
  • Administration: Delivered intratumorly
    (Only for Reference)

Solubility (25°C)

In vitro DMSO 100 mg/mL warmed (172.41 mM)
Water 20 mg/mL (34.48 mM)
Ethanol Insoluble

* Please note that Selleck tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Chemical Information

Molecular Weight 579.98
Formula

C27H29NO11.HCl

CAS No. 25316-40-9
Storage powder
in solvent
Synonyms NSC 123127

Bio Calculators

Molarity Calculator

Molarity Calculator

Calculate the mass, volume or concentration required for a solution. The Selleck molarity calculator is based on the following equation:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

  • Mass
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*When preparing stock solutions, please always use the batch-specific molecular weight of the product found on the via label and MSDS / COA (available on product pages).

Dilution Calculator

Dilution Calculator

Calculate the dilution required to prepare a stock solution. The Selleck dilution calculator is based on the following equation:

Concentration (start) x Volume (start) = Concentration (final) x Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2 ( Input Output )

  • C1
    V1
    C2
    V2

* When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and MSDS / COA (available online).

The Serial Dilution Calculator Equation

  • Serial Dilutions

  • Computed Result

  • C1=C0/X C1: LOG(C1):
    C2=C1/X C2: LOG(C2):
    C3=C2/X C3: LOG(C3):
    C4=C3/X C4: LOG(C4):
    C5=C4/X C5: LOG(C5):
    C6=C5/X C6: LOG(C6):
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    C8=C7/X C8: LOG(C8):
Molecular Weight Calculator

Molecular Weight Calculator

Enter the chemical formula of a compound to calculate its molar mass and elemental composition:

Total Molecular Weight: g/mol

Tip: Chemical formula is case sensitive. C10H16N2O2 c10h16n2o2

Instructions to calculate molar mass (molecular weight) of a chemical compound:

To calculate molar mass of a chemical compound, please enter its chemical formula and click 'Calculate'.

Definitions of molecular mass, molecular weight, molar mass and molar weight:

Molecular mass (molecular weight) is the mass of one molecule of a substance and is expressed in the unified atomic mass units (u). (1 u is equal to 1/12 the mass of one atom of carbon-12)
Molar mass (molar weight) is the mass of one mole of a substance and is expressed in g/mol.

Molarity Calculator

Mass Concentration Volume Molecular Weight

Clinical Trial Information

NCT Number Recruitment interventions Conditions Sponsor/Collaborators Start Date Phases
NCT04032964 Not yet recruiting Drug: L19TNF|Drug: DOXORUBICIN Soft Tissue Sarcoma Philogen S.p.A. September 2019 Phase 1
NCT03975205 Not yet recruiting Drug: Doxorubicin Lymphoma Leukemia Sutphin Drugs|Bharath Charitable Cancer Hospital and Institute July 1 2019 Early Phase 1
NCT03591276 Recruiting Drug: Chemotherapy Drugs Cancer Metastatic Breast Cancer Shaare Zedek Medical Center April 18 2019 Phase 1|Phase 2
NCT03719430 Recruiting Drug: Doxorubicin|Drug: APX005M Soft Tissue Sarcoma Columbia University|Apexigen Inc. March 20 2019 Phase 2
NCT03059615 Recruiting Drug: Nerofe|Drug: Doxorubicin Acute Myelogenous Leukemia|Myelodysplastic Syndromes Immune System Key Ltd October 25 2018 Phase 2

Tech Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store inhibitors, and issues that need special attention for cell-based assays and animal experiments.

Handling Instructions

Tel: +1-832-582-8158 Ext:3

If you have any other enquiries, please leave a message.

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Frequently Asked Questions

  • Question 1:

    Why the IC50 of the compound varied over time in our measurement?

  • Answer:

    Sometimes the IC50 value might vary between different batch of compounds due to the slight differences in purity. If different IC50 was seen in the same batch of compound, the problem may lies in the process of dissolvement. Make sure that you see no particles and the solution is clear with your stock solution.

Topoisomerase Signaling Pathway Map

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Cell Lines Assay Type Concentration Incubation Time Formulation Activity Description PMID