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Catalog No. Product Name Information Product Use Citations Product Validations
E0805New KL-11743 KL-11743 is a potent glucose-competitive inhibitor of the class I glucose transporters with IC50s of 115, 137 and 90 nM for GLUT1, GLUT2, and GLUT3.
S0235 Lavendustin B Lavendustin B inhibits HIV-1 integrase (IN) interaction with its cognate cellular cofactor lens epithelium-derived growth factor (LEDGF/p75). Lavendustin B is an inhibitor of Tyrosine Kinase and also a competitive inhibitor of glucose transporter 1 (Glut1).
S5748 4′-Deoxyphlorizin 4'-Deoxyphlorizin is an inhibitor of the glucose transport system.
S7927 WZB117 WZB117 is an inhibitor of Glucose Transporter 1 (GLUT1). It inhibited cell proliferation in lung cancer A549 cells and breast cancer MCF7 cells with an IC50 of approximately 10 μM.
Oncol Rep, 2022, 47(1)7
Int J Mol Sci, 2021, 22(16)9070
Neurosci Bull, 2021, 10.1007/s12264-020-00624-1
S7931 STF-31 STF-31 is a selective glucose transporter GLUT1 inhibitor.
Immunity, 2022, 55(1):159-173.e9
Mol Oncol, 2022, 16(15):2861-2880
FASEB J, 2022, 36(3):e22229
S8452 BAY-876 BAY-876 is a potent and selective GLUT1 inhibitor (IC50=0.002 μM) with a selectivity factor of >100 against GLUT2, GLUT3, and GLUT4.
Cell Chem Biol, 2021, S2451-9456(21)00441-4
Front Oncol, 2021, 11:783194
SSRN, 2021, 10.2139/ssrn.3862792
S9636 DRB18 DRB18 is a pan-GLUT (glucose transporters) inhibitor that inhibits growth and proliferation in several different cancer types with IC50 high nM range.
Cancers (Basel), 2022, 14(13)3225
E0805New KL-11743 KL-11743 is a potent glucose-competitive inhibitor of the class I glucose transporters with IC50s of 115, 137 and 90 nM for GLUT1, GLUT2, and GLUT3.
S0235 Lavendustin B Lavendustin B inhibits HIV-1 integrase (IN) interaction with its cognate cellular cofactor lens epithelium-derived growth factor (LEDGF/p75). Lavendustin B is an inhibitor of Tyrosine Kinase and also a competitive inhibitor of glucose transporter 1 (Glut1).
S5748 4′-Deoxyphlorizin 4'-Deoxyphlorizin is an inhibitor of the glucose transport system.
S7927 WZB117 WZB117 is an inhibitor of Glucose Transporter 1 (GLUT1). It inhibited cell proliferation in lung cancer A549 cells and breast cancer MCF7 cells with an IC50 of approximately 10 μM.
Oncol Rep, 2022, 47(1)7
Int J Mol Sci, 2021, 22(16)9070
Neurosci Bull, 2021, 10.1007/s12264-020-00624-1
S7931 STF-31 STF-31 is a selective glucose transporter GLUT1 inhibitor.
Immunity, 2022, 55(1):159-173.e9
Mol Oncol, 2022, 16(15):2861-2880
FASEB J, 2022, 36(3):e22229
S8452 BAY-876 BAY-876 is a potent and selective GLUT1 inhibitor (IC50=0.002 μM) with a selectivity factor of >100 against GLUT2, GLUT3, and GLUT4.
Cell Chem Biol, 2021, S2451-9456(21)00441-4
Front Oncol, 2021, 11:783194
SSRN, 2021, 10.2139/ssrn.3862792
S9636 DRB18 DRB18 is a pan-GLUT (glucose transporters) inhibitor that inhibits growth and proliferation in several different cancer types with IC50 high nM range.
Cancers (Basel), 2022, 14(13)3225
E0805New KL-11743 KL-11743 is a potent glucose-competitive inhibitor of the class I glucose transporters with IC50s of 115, 137 and 90 nM for GLUT1, GLUT2, and GLUT3.
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