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GLUT

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Isoform-selective Products

Cat.No. Product Name Information Product Use Citations Product Validations
S8452 BAY-876 BAY-876 is a potent and selective GLUT1 inhibitor (IC50=0.002 μM) with a selectivity factor of >100 against GLUT2, GLUT3, and GLUT4.
BMC Cancer, 2025, 25(1):716
Am J Pathol, 2024, S0002-9440(24)00116-0
Cancer Cell Int, 2024, 24(1):19
S7927 WZB117 WZB117 is an inhibitor of Glucose Transporter 1 (GLUT1). It inhibited cell proliferation in lung cancer A549 cells and breast cancer MCF7 cells with an IC50 of approximately 10 μM.
Nat Commun, 2025, 16(1):4929
Nat Commun, 2024, 15(1):4363
Am J Pathol, 2024, S0002-9440(24)00116-0
S7931 STF-31 STF-31 is a selective glucose transporter GLUT1 inhibitor.
Cancer Cell Int, 2025, 25(1):199
Immunity, 2022, 55(1):159-173.e9
J Control Release, 2022, 352:540-555
Verified customer review of STF-31
S9636 DRB18 DRB18 is a pan-GLUT (glucose transporters) inhibitor that inhibits growth and proliferation in several different cancer types with IC50 high nM range.
Cancer Cell, 2022, 40(10):1207-1222.e10
Cancers (Basel), 2022, 14(13)3225
E0805 KL-11743 KL-11743 is a potent glucose-competitive inhibitor of the class I glucose transporters with IC50s of 115, 137 and 90 nM for GLUT1, GLUT2, and GLUT3.
Sci Rep, 2024, 14(1):15340
S5748 4′-Deoxyphlorizin 4'-Deoxyphlorizin is an inhibitor of the glucose transport system.
S0235 Lavendustin B Lavendustin B inhibits HIV-1 integrase (IN) interaction with its cognate cellular cofactor lens epithelium-derived growth factor (LEDGF/p75). This compound is an inhibitor of Tyrosine Kinase and also a competitive inhibitor of glucose transporter 1 (Glut1).