Product Categories

Sodium Channel

Cat.No.	Product Name	Information
S1614	Riluzole (Rilutek)	Riluzole(Rilutek) is a drug used to treat amyotrophic lateral sclerosis.
S1693	Carbamazepine (Carbatrol)	Carbamazepine (Carbatrol) is a sodium channel blocker with IC50 of 131 μM in rat brain synaptosomes.
S2524	Phenytoin sodium (Dilantin)	Phenytoin sodium (Dilantin) is an inactive voltage-gated sodium channel stabilizer.
S2785	A-803467	A-803467 is a selective Na_V1.8 channel blocker with IC50 of 8 nM.
S3024	Lamotrigine	Lamotrigine is a novel anticonvulsant drug for inhibition of 5-HT with IC50 of 240 μM and 474 μM in human platelets and rat brain synaptosomes, respectively.
S4038	Dibucaine (Cinchocaine) HCl	Dibucaine (Cinchocaine) HCl is a local anesthetics.
S4023	Procaine (Novocaine) HCl	Procaine (Novocaine) HCl is an inhibitor of sodium channel, NMDA receptor and nAChR with IC50 of 60 μM, 0.296 mM and 45.5 μM, which is also an inhibitor of 5-HT3 with K_D of 1.7 μM.
S4016	Ouabain	Ouabain is a selective Na+, K+-ATPase inhibitor, binds to α2 subunit and α3 subunit with K_i of 41 nM and 15 nM, respectively.
S1256	Rufinamide (Banzel)	Rufinamide, a triazole derivative, is an anticonvulsant medication.
S1391	Oxcarbazepine	Oxcarbazepine inhibits the binding of [3H]BTX to sodium channels with IC50 of 160 μM and also inhibits the influx of ²²Na⁺ into rat brain synaptosomes with IC50 about 100 μM.

Cat.No.	Product Name	Information
S2500	Propafenone (Rytmonorm) HCl	Propafenone(Rytmonorm) is a classic anti-arrhythmic medication, which treats illnesses associated with rapid heartbeats such as atrial and ventricular arrhythmias.
S2525	Phenytoin (Lepitoin)	Phenytoin (Lepitoin; NSC 8722; Phenytek; Phenytoine; Sodanton; Zentropi) is an inactive voltage-gated sodium channel stabilizer.
S2560	Amiloride HCl dihydrate	Amiloride hydrochloride dihydrate is a potent epithelial sodium channel blocker.
S1828	Proparacaine HCl	Proparacaine HCl is a voltage-gated sodium channels antagonist with ED50 of 3.4 mM.
S2110	Vinpocetine (Cavinton)	Vinpocetine is a selectively inhibitor of voltage-sensitive sodium channel for the treatment of stroke, vascular dementia and Alzheimer's disease.
S2118	Ibutilide fumarate	Ibutilide is a Class III antiarrhythmic agent that is indicated for acute cardioconversion of atrial fibrillation and atrial flutter of a recent onset to sinus rhythm by induction of slow inward sodium current, which prolongs action potential and refractory period of myocardial cells.
S3064	Ambroxol HCl	Ambroxol HCl is a potent inhibitor of the neuronal Na⁺ channels with IC50 of 35.2 μM and 22.5 μM for tonic and phasic block, respectively.