Calcium Channel

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Calcium Channel Inhibitors | Activators | Antagonists (28)

water-soluble

Cat.No. Product Name Information Product Use Citation Customer Product Validation
S1356 Levetiracetam Levetiracetam is an anticonvulsant medication used to treat epilepsy.
S1813 Amlodipine Besylate Amlodipine Besylate is a long-acting calcium channel blocker, used to lower blood pressure and prevent chest pain.
S1293 Cilnidipine Cilnidipine is a unique L-type and N-type calcium channel blocker, used for high blood pressure treatment.
S1425 Ranolazine 2HCl Ranolazine 2HCl is a calcium uptake inhibitor via the sodium/calcium channal, used to treat chronic angina.
S4202 Verapamil HCl Verapamil HCl is an L-type calcium channel blocker that is a class IV anti-arrhythmia agent.
S1799 Ranolazine Ranolazine 2HCl is a calcium uptake inhibitor via the sodium/calcium channal, used to treat chronic angina.
S1662 Isradipine Isradipine is a potent and selective L-type voltage-gated calcium channel blocker, used to treat high blood pressure.
S1885 Felodipine Felodipine is a selective L-type Ca2+ channel blocker with IC50 of 0.15 nM.
S1905 Amlodipine Amlodipine is a long-acting calcium channel blocker, used to lower blood pressure and prevent chest pain.
S2482 Manidipine 2HCl Manidipine 2HCl is a HCl salt form of Manidipine, which is a calcium channel blocker with IC50 of 2.6 nM, used clinically as an antihypertensive. Phase 4.
Cat.No. Product Name Information Product Use Citation Customer Product Validation
S1748 Nisoldipine Nisoldipine (Sular) is a calcium channel blocker belonging to the dihydropyridines class, specific for L-type Cav1.2 with IC50 of 10 nM.
S2481 Manidipine Manidipine is a calcium channel blocker (dihydropyridine type) that is used clinically as an antihypertensive.
S2721 Nilvadipine Nilvadipine is a potent calcium channel blocker with an IC50 of 0.03 nM.
S1747 Nimodipine Nimodipine is a dihydropyridine calcium channel blocker and an autophagy inhibitor, used in the treatment of high blood pressure.
S1994 Lacidipine Lacidipine is a L-type calcium channel blocker.
S2114 Dronedarone HCl Dronedarone HCl is a therapy for the treatment of patients with paroxysmal and persistent atrial fibrillation or atrial flutter.
S2080 Clevidipine Butyrate Clevidipine Butyrate is a dihydropyridine calcium channel blocker, uses as an agent for the reduction of blood pressure.
S4181 Nicardipine HCl Nicardipine is a dihydropyridine calcium-channel blocking agent used for the treatment of vascular disorders.
S2030 Flunarizine 2HCl Flunarizine 2HCl is a dihydrochloride salt form which is a calcium channel blocker with a Ki of 68 nM.
S2017 Benidipine HCl Benidipine HCl is a hydrochloride salt form of benidipine which is a dihydropyridine calcium channel blocker.
Cat.No. Product Name Information Product Use Citation Customer Product Validation
S3053 Azelnidipine Azelnidipine is a dihydropyridine calcium channel blocker.
S2050 Strontium Ranelate Strontium Ranelate is a strontium(II) salt of ranelic acid for (-)-desmethoxyverapamil binding to calcium channel with IC50 of 0.5 mM.
S2573 Tetracaine HCl Tetracaine HCl is a hydrochloride salt form of tetracaine which is a potent local anaesthetic and a channel function allosteric inhibitor.
S2491 Nitrendipine Nitrendipine is a dihydropyridine calcium channel blocker with an IC50 of 95 nM.
S1865 Diltiazem HCl Diltiazem HCl (Tiazac) is a benzothiazepine derivative with vasodilating action due to its antagonism of the actions of the calcium ion in membrane functions.
S3045 Cinepazide maleate Cinepazide maleate is a maleate salt form of cinepazide which is a vasodilator.
S2403 Tetrandrine Tetrandrine, a bis-benzylisoquinoline alkaloid derived from Stephania tetrandra, is a calcium channel blocker.
S4084 Lomerizine HCl Lomerizine dihydrochloride is a relatively new L- and T-type calcium channel blocker used in the treatment of migraine.

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Cat.No. Product Name Solubility (25°C)
Water DMSO Ethanol
S1356 Levetiracetam 34 mg/mL 34 mg/mL 34 mg/mL
S1813 Amlodipine Besylate <1 mg/mL 113 mg/mL 14 mg/mL
S1293 Cilnidipine <1 mg/mL 99 mg/mL 15 mg/mL
S1425 Ranolazine 2HCl 100 mg/mL 100 mg/mL <1 mg/mL
S4202 Verapamil HCl 50 mg/mL 98 mg/mL 12 mg/mL
S1799 Ranolazine <1 mg/mL 86 mg/mL 20 mg/mL
S1662 Isradipine <1 mg/mL 74 mg/mL 74 mg/mL
S1885 Felodipine <1 mg/mL 77 mg/mL 72 mg/mL
S1905 Amlodipine <1 mg/mL 82 mg/mL 82 mg/mL
S2482 Manidipine 2HCl <1 mg/mL 21 mg/mL <1 mg/mL
S1748 Nisoldipine <1 mg/mL 77 mg/mL 60 mg/mL
S2481 Manidipine <1 mg/mL 122 mg/mL 3 mg/mL
S2721 Nilvadipine <1 mg/mL 77 mg/mL 33 mg/mL
S1747 Nimodipine <1 mg/mL 84 mg/mL 84 mg/mL
S1994 Lacidipine <1 mg/mL 91 mg/mL 22 mg/mL
S2114 Dronedarone HCl <1 mg/mL 80 mg/mL 40 mg/mL
S2080 Clevidipine Butyrate <1 mg/mL 91 mg/mL 3 mg/mL
S4181 Nicardipine HCl <1 mg/mL 100 mg/mL <1 mg/mL
S2030 Flunarizine 2HCl <1 mg/mL 5 mg/mL 3 mg/mL
S2017 Benidipine HCl <1 mg/mL 8 mg/mL <1 mg/mL
S3053 Azelnidipine <1 mg/mL 117 mg/mL 7 mg/mL
S2050 Strontium Ranelate <1 mg/mL <1 mg/mL <1 mg/mL
S2573 Tetracaine HCl 60 mg/mL 60 mg/mL 30 mg/mL
S2491 Nitrendipine <1 mg/mL 72 mg/mL <1 mg/mL
S1865 Diltiazem HCl 90 mg/mL 90 mg/mL 4 mg/mL
S3045 Cinepazide maleate 107 mg/mL 107 mg/mL <1 mg/mL
S2403 Tetrandrine <1 mg/mL 4 mg/mL 2 mg/mL
S4084 Lomerizine HCl <1 mg/mL 4 mg/mL <1 mg/mL
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