Calcium Channel

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Calcium Channel Inhibitors | Activators | Antagonists (33)

water-soluble

Cat.No. Product Name Information Product Use Citation Customer Product Validation
S1356 Levetiracetam Levetiracetam is an anticonvulsant medication used to treat epilepsy.
  • Sci Rep, 2016, 6:25705
S1813 Amlodipine Besylate Amlodipine Besylate is a long-acting calcium channel blocker, used to lower blood pressure and prevent chest pain.
S1293 Cilnidipine Cilnidipine is a unique L-type and N-type calcium channel blocker, used for high blood pressure treatment.
S1425 Ranolazine 2HCl Ranolazine 2HCl is a calcium uptake inhibitor via the sodium/calcium channal, used to treat chronic angina.
S4202 Verapamil HCl Verapamil HCl is an L-type calcium channel blocker that is a class IV anti-arrhythmia agent.
S1799 Ranolazine Ranolazine is a calcium uptake inhibitor via the sodium/calcium channel, used to treat chronic angina.
S1662 Isradipine Isradipine is a potent and selective L-type voltage-gated calcium channel blocker, used to treat high blood pressure.
S1885 Felodipine Felodipine is a selective L-type Ca2+ channel blocker with IC50 of 0.15 nM.
S1905 Amlodipine Amlodipine is a long-acting calcium channel blocker, used to lower blood pressure and prevent chest pain.
S2482 Manidipine 2HCl Manidipine 2HCl is a HCl salt form of Manidipine, which is a calcium channel blocker with IC50 of 2.6 nM, used clinically as an antihypertensive. Phase 4.
Cat.No. Product Name Information Product Use Citation Customer Product Validation
S1748 Nisoldipine Nisoldipine (Sular) is a calcium channel blocker belonging to the dihydropyridines class, specific for L-type Cav1.2 with IC50 of 10 nM.
S2481 Manidipine Manidipine is a calcium channel blocker (dihydropyridine type) that is used clinically as an antihypertensive.
S2535 Econazole nitrate Econazole Nitrate is a Ca2+ channel blocker, used as an antifungal medicine that fights infections caused by fungus.
S2721 Nilvadipine Nilvadipine is a potent calcium channel blocker with an IC50 of 0.03 nM.
S1747 Nimodipine Nimodipine is a dihydropyridine calcium channel blocker and an autophagy inhibitor, used in the treatment of high blood pressure.
  • Antiviral Res, 2016, 132:38-45
S1994 Lacidipine Lacidipine is a L-type calcium channel blocker, used for treating high blood pressure.
S2114 Dronedarone HCl Dronedarone HCl is a multichannel blocker targeting potassium channel, sodium channel and calcium channel, used as an antiarrhythmic drug for treatment of atrial fibrillation (AF).
S2080 Clevidipine Butyrate Clevidipine Butyrate is a dihydropyridine calcium channel blocker, uses as an agent for the reduction of blood pressure.
S4181 Nicardipine HCl Nicardipine is a dihydropyridine calcium-channel blocking agent used for the treatment of vascular disorders.
S1808 Nifedipine Nifedipine is a dihydropyridine calcium channel blocker, used to lower hypertension and to treat angina.
  • Antiviral Res, 2016, 132:38-45
  • Toxicol Appl Pharmacol, 2015, 285(1):51-60
Cat.No. Product Name Information Product Use Citation Customer Product Validation
S2030 Flunarizine 2HCl Flunarizine 2HCl is a dihydrochloride salt form which is a calcium channel blocker with a Ki of 68 nM.
S2017 Benidipine HCl Benidipine HCl is a hydrochloride salt form of benidipine which is a dihydropyridine calcium channel blocker.
S2918 HC-030031 HC-030031 is a selective TRPA1 channel blocker that antagonizes AITC- and formalin-evoked calcium influx with IC50 of 6.2 μM and 5.3 μM respectively.
S3053 Azelnidipine Azelnidipine is a dihydropyridine calcium channel blocker.
S2050 Strontium Ranelate Strontium Ranelate is a strontium(II) salt of ranelic acid for (-)-desmethoxyverapamil binding to calcium channel with IC50 of 0.5 mM.
S2573 Tetracaine HCl Tetracaine HCl is a hydrochloride salt form of tetracaine which is a potent local anaesthetic and a channel function allosteric inhibitor.
S2491 Nitrendipine Nitrendipine is a dihydropyridine calcium channel blocker with an IC50 of 95 nM.
S1865 Diltiazem HCl Diltiazem HCl (Tiazac) is a benzothiazepine derivative with vasodilating action due to its antagonism of the actions of the calcium ion in membrane functions.
S4209 Chlorocresol Chlorocresol is an activator of ryanodine receptor.
S3045 Cinepazide maleate Cinepazide maleate is a maleate salt form of cinepazide which is a vasodilator.
Cat.No. Product Name Information Product Use Citation Customer Product Validation
S2403 Tetrandrine Tetrandrine, a bis-benzylisoquinoline alkaloid derived from Stephania tetrandra, is a calcium channel blocker.
  • Antiviral Res, 2016, 132:38-45
  • Biochem Biophys Res Commun, 2016, 476(4):481-6
S4084 Lomerizine HCl Lomerizine dihydrochloride is a relatively new L- and T-type calcium channel blocker used in the treatment of migraine.
S8073 Optovin Optovin is a reversible photoactivated TRPA1 activator.

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Cat.No. Product Name Solubility (25°C)
Water DMSO Ethanol
S1356 Levetiracetam 34 mg/mL 34 mg/mL 34 mg/mL
S1813 Amlodipine Besylate <1 mg/mL 113 mg/mL 14 mg/mL
S1293 Cilnidipine <1 mg/mL 99 mg/mL 15 mg/mL
S1425 Ranolazine 2HCl 100 mg/mL 100 mg/mL <1 mg/mL
S4202 Verapamil HCl 50 mg/mL 98 mg/mL 12 mg/mL
S1799 Ranolazine <1 mg/mL 86 mg/mL 20 mg/mL
S1662 Isradipine <1 mg/mL 74 mg/mL 74 mg/mL
S1885 Felodipine <1 mg/mL 77 mg/mL 72 mg/mL
S1905 Amlodipine <1 mg/mL 82 mg/mL 82 mg/mL
S2482 Manidipine 2HCl <1 mg/mL 21 mg/mL <1 mg/mL
S1748 Nisoldipine <1 mg/mL 77 mg/mL 60 mg/mL
S2481 Manidipine <1 mg/mL 122 mg/mL 3 mg/mL
S2535 Econazole nitrate <1 mg/mL 89 mg/mL 5 mg/mL
S2721 Nilvadipine <1 mg/mL 77 mg/mL 33 mg/mL
S1747 Nimodipine <1 mg/mL 84 mg/mL 84 mg/mL
S1994 Lacidipine <1 mg/mL 91 mg/mL 22 mg/mL
S2114 Dronedarone HCl <1 mg/mL 80 mg/mL 40 mg/mL
S2080 Clevidipine Butyrate <1 mg/mL 91 mg/mL 3 mg/mL
S4181 Nicardipine HCl <1 mg/mL 100 mg/mL <1 mg/mL
S1808 Nifedipine <1 mg/mL 69 mg/mL 15 mg/mL
S2030 Flunarizine 2HCl <1 mg/mL 5 mg/mL 3 mg/mL
S2017 Benidipine HCl <1 mg/mL 8 mg/mL <1 mg/mL
S2918 HC-030031 <1 mg/mL 32 mg/mL <1 mg/mL
S3053 Azelnidipine <1 mg/mL 117 mg/mL 7 mg/mL
S2050 Strontium Ranelate <1 mg/mL <1 mg/mL <1 mg/mL
S2573 Tetracaine HCl 60 mg/mL 60 mg/mL 30 mg/mL
S2491 Nitrendipine <1 mg/mL 72 mg/mL <1 mg/mL
S1865 Diltiazem HCl 90 mg/mL 90 mg/mL 4 mg/mL
S4209 Chlorocresol <1 mg/mL 29 mg/mL 29 mg/mL
S3045 Cinepazide maleate 107 mg/mL 107 mg/mL <1 mg/mL
S2403 Tetrandrine <1 mg/mL 1 mg/mL <1 mg/mL
S4084 Lomerizine HCl <1 mg/mL 100 mg/mL 52 mg/mL
S8073 Optovin <1 mg/mL 63 mg/mL <1 mg/mL
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