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Calcium Channel inhibitors/antagonist

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Isoform-selective Products

Cat.No. Product Name Information Product Use Citations Product Validations
S7924 Bay K 8644 Bay K 8644 is a racemate. Bay K 8644 is a potent, selective activator of L-type Ca2+ channel with IC50 of 17.3 nM.
J Neurotrauma, 2025, 10.1177/08977151251374286
EMBO Rep, 2024, 25(11):4777-4802
ACS Nano, 2021, 10.1021/acsnano.1c03517
Verified customer review of Bay K 8644
S7914 ISX-9 (Isoxazole 9) Isoxazole 9 (Isx-9) is a synthetic promotor of adult neurogenesis by triggering neuronal differentiation of adult neural stem/precursor cells (NSPCs). Isoxazole 9 (Isx-9) activates multiple pathways including TGF-β induced epithelial–mesenchymal transition (EMT) signaling, canonical and non-canonical Wnt signaling at different stages of cardiac differentiation.
iScience, 2025, 28(3):112015
Front Cell Dev Biol, 2025, 13:1513163
Cell Regen, 2025, 14(1):18
S4202 Verapamil HCl Verapamil HCl is an L-type calcium channel blocker that is a class IV anti-arrhythmia agent. Verapamil inhibits both permeability-glycoprotein (P-gp) and CYP3A4.
Cancer Cell, 2025, 43(4):776-796.e14
Nat Commun, 2025, 16(1):7115
Blood Sci, 2025, 7(2):e00236
Verified customer review of Verapamil HCl
S1808 Nifedipine Nifedipine is a dihydropyridine calcium channel blocker, used to lower hypertension and to treat angina.
Dis Model Mech, 2025, 18(6)dmm052220
J Immunother Cancer, 2024, 12(11)e009805
Laryngoscope Investig Otolaryngol, 2023, 8(5):1390-1400
Verified customer review of Nifedipine
S2721 Nilvadipine Nilvadipine (ARC029, FR34235,FK235) is a potent calcium channel blocker with an IC50 of 0.03 nM.
Cell Death Differ, 2024, 10.1038/s41418-024-01418-y
J Immunother Cancer, 2024, 12(11)e009805
Nat Commun, 2022, 13-1:6117
S2030 Flunarizine 2HCl Flunarizine 2HCl (KW-3149, R14950) is a dihydrochloride salt form which is a calcium channel blocker with a Ki of 68 nM.
Sci Adv, 2023, 9(15):eadf2695
J Pers Med, 2022, 12(2)258
Hum Cell, 2022, 10.1007/s13577-022-00671-y
S1905 Amlodipine Amlodipine (UK-48340) is a long-acting calcium channel blocker, used to lower blood pressure and prevent chest pain.
J Immunother Cancer, 2024, 12(11)e009805
Cancer Med, 2024, 13(11):e7291
Acta Pharm Sin B, 2023, 13(10):4217-4233
S1293 Cilnidipine Cilnidipine is a unique L-type and N-type calcium channel blocker, used for high blood pressure treatment.
J Immunother Cancer, 2024, 12(11)e009805
Nat Commun, 2021, 12(1):3907
Cell Discov, 2020, 6(1):96
S1748 Nisoldipine Nisoldipine (Sular, BAY K 5552) is a calcium channel blocker belonging to the dihydropyridines class, specific for L-type Cav1.2 with IC50 of 10 nM.
J Immunother Cancer, 2024, 12(11)e009805
Biomed Pharmacother, 2022, 145:112432
iScience, 2022, 25(10):105068
S1356 Levetiracetam (UCB-L059) Levetiracetam (UCB-L059, SIB-S1) is an anticonvulsant medication used to treat epilepsy and an agonist of muscarinic acetylcholine receptors (mAChR). This compound also modulates the presynaptic P/Q-type voltage-dependent calcium (Ca2+) channel.
Front Neurosci, 2023, 17:1336026
bioRxiv, 2023, 2023.11.10.566574
Alzheimers Dement (N Y), 2022, 8(1):e12329
Verified customer review of Levetiracetam (UCB-L059)

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