BzATP triethylammonium salt

BzATP triethylammonium salt acts as a P2X receptor agonist with pEC50s of 8.74, 5.26, 7.10, 7.50, 6.19, 6.31, 5.33 for P2X1, P2X2, P2X3, P2X2/3, P2X4 and P2X7, respectively, also is potent at P2X7 receptors with EC50s of 3.6 μM and 285 μM for rat P2X7 and mouse P2X7, respectively.

BzATP triethylammonium salt Chemical Structure

BzATP triethylammonium salt Chemical Structure

CAS: 112898-15-4

Purity & Quality Control

Batch: E112801 Water] 100 mg/mL] false] DMSO] 50 mg/mL] false] Ethanol] Insoluble] false Purity: 99.44%
99.44

BzATP triethylammonium salt Related Products

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Biological Activity

Description BzATP triethylammonium salt acts as a P2X receptor agonist with pEC50s of 8.74, 5.26, 7.10, 7.50, 6.19, 6.31, 5.33 for P2X1, P2X2, P2X3, P2X2/3, P2X4 and P2X7, respectively, also is potent at P2X7 receptors with EC50s of 3.6 μM and 285 μM for rat P2X7 and mouse P2X7, respectively.
Targets
P2X1 [1]
(in fluo-3 Ca2+ influx assay)
P2X3 [1]
(in fluo-3 Ca2+ influx assay)
P2X4 [1]
(in fluo-3 Ca2+ influx assay)
P2X2/3 [1]
(in fluo-3 Ca2+ influx assay)
P2X7 [1]
(in fluo-3 Ca2+ influx assay)
Click to View More Targets
8.74(pEC50) 7.1(pEC50) 6.31(pEC50) 6.19(pEC50) 5.33(pEC50)

Chemical Information & Solubility

Molecular Weight 816.58 Formula

C24H24N5O15P3.C6H15N

CAS No. 112898-15-4 SDF --
Storage (From the date of receipt) 3 years -20°C powder

In vitro
Batch:

Water : 100 mg/mL

DMSO : 50 mg/mL ( (61.23 mM); Moisture-absorbing DMSO reduces solubility. Please use fresh DMSO.)

Ethanol : Insoluble


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In vivo
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Method for preparing in vivo formulation: Take μL DMSO master liquid, next add μL Corn oil, mix and clarify.

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