Lipase

  • Inhibitory Selectivity
  • Solubility
Catalog No. Product Name Solubility(25°C)
Water DMSO Alcohol
S1629 Orlistat <1 mg/mL 99 mg/mL 99 mg/mL
S4904 JZL184 <1 mg/mL 100 mg/mL <1 mg/mL
S7364 Atglistatin <1 mg/mL 56 mg/mL 4 mg/mL
S7457 XEN445 <1 mg/mL 80 mg/mL 34 mg/mL
S9234 Schaftoside -1 mg/mL 100 mg/mL -1 mg/mL
S4930 Cetilistat <1 mg/mL 3 mg/mL 8 mg/mL
S2365 Tanshinone IIA <1 mg/mL 5 mg/mL <1 mg/mL
S4825 Pancreatin <1 mg/mL 0.01 mg/mL <1 mg/mL
Catalog No. Information Product Use Citations Product Validations
S1629

Orlistat

Orlistat is a general lipase inhibitor with IC50 of 122 ng/ml for PL from human duodenal juice.
S4904

JZL184

JZL 184 is the first selective inhibitor of monoacylglycerol lipase (MAGL) with IC50 of 8 nM.
S7364

Atglistatin

Atglistatin is a highly potent, and selective inhibitor of adipose triglyceride lipase (ATGL) with IC50 of 0.7 μM, high selectivity over other key metabolic lipases.

S7457

XEN445

XEN445 is a potent and selective endothelial lipase inhibitor with IC50 of 0.237 μM.

S9234New

Schaftoside

Schaftoside, a bioactive compound found in the Herba Desmodii Styracifolii, exhibits pancreatic lipase inhibitory activity.
S4930New

Cetilistat

Cetilistat is a novel highly lipophilic benzoxazinone that inhibits gastrointestinal and pancreatic lipases. It shows a good safety and tolerability profile in vivo
S2365

Tanshinone IIA

Tanshinone IIA(Tanshinone B) is the most abundant diterpene quinone in Danshen, Salviae miltiorrhizae Radix, a widely prescribed traditional herbal medicine that is used to treat cardiovascular and inflammatory diseases; A natural monoacylglycerol lipase inhibitor.
S4825New

Pancreatin

Pancreatic enzymes also known as pancrelipase and pancreatin, are commercial mixtures of amylase, lipase, and protease. They are used to treat malabsorption syndrome due to pancreatic problems.