Home Epigenetics Histone Methyltransferase inhibitor BIX-01294

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BIX-01294 Histone Methyltransferase inhibitor

Cat.No.E4799

BIX-01294 is a potent, reversible and highly selective dual inhibitor of G9a and GLP, with IC₅₀ values of 1.7 μM and 38 μM, respectively. It selectively inhibits recurrent tumor cell growth and represents a targetable dependency in recurrent breast cancer research.
BIX-01294 Histone Methyltransferase inhibitor Chemical Structure

Chemical Structure

Molecular Weight: 490.64

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Chemical Information, Storage & Stability

Molecular Weight 490.64 Formula

C28H38N6O2

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CAS No. 935693-62-2 Download SDF Storage of Stock Solutions

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Method for preparing in vivo formulation: Take μL DMSO master liquid, next add μL Corn oil, mix and clarify.

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