D3-βArr TSH Receptor modulator

D3-βArr(NCGC00379308) is a positive allosteric modulator of thyrotropin receptor (TSHR) that modulates TSH-induced β-Arr 1 translocation.

D3-βArr TSH Receptor modulator Chemical Structure

Chemical Structure

Molecular Weight: 333.43

Purity & Quality Control

Batch: S031901 DMSO]67 mg/mL]false]Ethanol]33 mg/mL]false]Water]Insoluble]false Purity: 99.96%
99.96

Chemical Information

Molecular Weight 333.43 Formula

C20H23N5

CAS No. 662164-09-2 SDF --
Synonyms NCGC00379308
Smiles CC(C1=CC=CC=C1)NC2=NC(=NC3=CC=CC=C32)N4CCNCC4

Storage and Stability

Storage (From the date of receipt) 3 years -20°C powder

In vitro
Batch:

DMSO : 67 mg/mL ( (200.94 mM) Moisture-absorbing DMSO reduces solubility. Please use fresh DMSO.)

Ethanol : 33 mg/mL

Water : Insoluble


Molecular Weight Calculator

In vivo
Batch:

Add solvents to the product individually and in order.


In vivo Formulation Calculator

Mechanism of Action

Targets
TSHR [1]

References

  • https://pubmed.ncbi.nlm.nih.gov/29089368/

Tech Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store inhibitors, and issues that need special attention for cell-based assays and animal experiments.

Handling Instructions

Tel: +1-832-582-8158 Ext:3
If you have any other enquiries, please leave a message.

* Indicates a Required Field

Please enter your name.
Please enter your email. Please enter a valid email address.
Please write something to us.