Carbetapentane

Synonyms: Pentoxyverine, CB

Carbetapentane (Pentoxyverine, CB) is an antitussive anticonvulsant nonselective sigma-1 (σ1) agonist.

Carbetapentane Chemical Structure

Carbetapentane Chemical Structure

CAS: 77-23-6

Purity & Quality Control

Batch: S086901 Purity: 98.61%
98.61

Carbetapentane Related Products

Choose Selective Sigma Receptor Inhibitors

Biological Activity

Description Carbetapentane (Pentoxyverine, CB) is an antitussive anticonvulsant nonselective sigma-1 (σ1) agonist.
Targets
σ1 [1]
NCT Number Recruitment Conditions Sponsor/Collaborators Start Date Phases
NCT05312372 Withdrawn
Esophageal Squamous Cell Carcinoma
Institut de Recherches Internationales Servier|ADIR a Servier Group company|Servier
May 2025 Phase 1|Phase 2
NCT06135064 Not yet recruiting
PTSD
University of Utah
April 2024 Phase 1|Phase 2
NCT05992831 Recruiting
Mild Cognitive Impairment|Depression
Medical University of South Carolina|National Institute on Aging (NIA)
January 11 2024 Not Applicable
NCT06116357 Not yet recruiting
Primary Hypertension
Jing Huang|The Second Affiliated Hospital of Chongqing Medical University
December 1 2023 Not Applicable
NCT05896332 Recruiting
Alcohol Use Disorder|Mild Cognitive Impairment|Transcranial Magnetic Stimulation
Medical University of South Carolina|National Institutes of Health (NIH)|National Institute on Alcohol Abuse and Alcoholism (NIAAA)
November 1 2023 Phase 1

Chemical Information & Solubility

Molecular Weight 333.46 Formula

C20H31NO3

CAS No. 77-23-6 SDF --
Density 1.048 g/mL
Smiles CCN(CC)CCOCCOC(=O)C1(CCCC1)C2=CC=CC=C2
Storage (From the date of receipt) 2 years -20°C liquid

In vitro
Batch:


Molecular Weight Calculator

In vivo
Batch:

Add solvents to the product individually and in order.


In vivo Formulation Calculator

Preparing Stock Solutions

Molarity Calculator

Mass Concentration Volume Molecular Weight

In vivo Formulation Calculator (Clear solution)

Step 1: Enter information below (Recommended: An additional animal making an allowance for loss during the experiment)

mg/kg g μL

Step 2: Enter the in vivo formulation (This is only the calculator, not formulation. Please contact us first if there is no in vivo formulation at the solubility Section.)

% DMSO % % Tween 80 % ddH2O
%DMSO %

Calculation results:

Working concentration: mg/ml;

Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO ( Master liquid concentration mg/mL, Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug. )

Method for preparing in vivo formulation: Take μL DMSO master liquid, next addμL PEG300, mix and clarify, next addμL Tween 80, mix and clarify, next add μL ddH2O, mix and clarify.

Method for preparing in vivo formulation: Take μL DMSO master liquid, next add μL Corn oil, mix and clarify.

Note: 1. Please make sure the liquid is clear before adding the next solvent.
2. Be sure to add the solvent(s) in order. You must ensure that the solution obtained, in the previous addition, is a clear solution before proceeding to add the next solvent. Physical methods such
as vortex, ultrasound or hot water bath can be used to aid dissolving.

Tech Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store inhibitors, and issues that need special attention for cell-based assays and animal experiments.

Handling Instructions

Tel: +1-832-582-8158 Ext:3
If you have any other enquiries, please leave a message.

* Indicates a Required Field

Please enter your name.
Please enter your email. Please enter a valid email address.
Please write something to us.
Tags: buy Carbetapentane | Carbetapentane supplier | purchase Carbetapentane | Carbetapentane cost | Carbetapentane manufacturer | order Carbetapentane | Carbetapentane distributor