PREP

Choose Selective PREP Inhibitors

PREP Products

  • All (5)
  • PREP Inhibitors (5)
  • New PREP Products
Catalog No. Product Name Information Product Use Citations Product Validations
S0842 SP-13786 SP-13786 (UAMC-1110)(compound 60) is a potent and selective inhibitor of fibroblast activation protein (FAP) and prolyl oligopeptidase (PREP) with IC50 of 3.2 nM and 1.8 μM, respectively.
S2268 Baicalein Baicalein is a CYP2C9 and prolyl endopeptidase inhibitor.
Cancer Cell, 2022, S1535-6108(22)00312-9
Adv Sci (Weinh), 2021, e2103360
Free Radic Biol Med, 2021, 163:234-242
S2269 Baicalin (NSC-661431) Baicalin (NSC-661431) is a known prolyl endopeptidase inhibitor and affects the GABA receptors.
Molecules, 2021, 26(5)1210
Innate Immun, 2021, 27(7-8):533-542
Reprod Fertil Dev, 2019, 31(5):983-992
S2396 Salidroside Salidroside (Rhodioloside), a phenylpropanoid glycoside isolated from Rhodiola rosea, has been reported to have a broad spectrum of pharmacological properties. Salidroside is a prolyl endopeptidase inhibitor. Salidroside alleviates cachexia symptoms in mouse models of cancer cachexia via activating mTOR signalling. Salidroside protects dopaminergic neurons by enhancing PINK1/Parkin-mediated mitophagy.
FASEB J, 2021, 35(12):e22044
Curr Med Sci, 2021, 10.1007/s11596-021-2374-6
J Med Virol, 2019, 91(8):1440-1447
S3249 Corypalmine Corypalmine ((R)-(+)-Corypalmine), an alkaloid isolated from Stephania cepharantha, is an inhibitor of prolyl endopeptidase/oligopeptidase (PREP/POP) with IC50 of 128.0 μM.
S0842 SP-13786 SP-13786 (UAMC-1110)(compound 60) is a potent and selective inhibitor of fibroblast activation protein (FAP) and prolyl oligopeptidase (PREP) with IC50 of 3.2 nM and 1.8 μM, respectively.
S2268 Baicalein Baicalein is a CYP2C9 and prolyl endopeptidase inhibitor.
Cancer Cell, 2022, S1535-6108(22)00312-9
Adv Sci (Weinh), 2021, e2103360
Free Radic Biol Med, 2021, 163:234-242
S2269 Baicalin (NSC-661431) Baicalin (NSC-661431) is a known prolyl endopeptidase inhibitor and affects the GABA receptors.
Molecules, 2021, 26(5)1210
Innate Immun, 2021, 27(7-8):533-542
Reprod Fertil Dev, 2019, 31(5):983-992
S2396 Salidroside Salidroside (Rhodioloside), a phenylpropanoid glycoside isolated from Rhodiola rosea, has been reported to have a broad spectrum of pharmacological properties. Salidroside is a prolyl endopeptidase inhibitor. Salidroside alleviates cachexia symptoms in mouse models of cancer cachexia via activating mTOR signalling. Salidroside protects dopaminergic neurons by enhancing PINK1/Parkin-mediated mitophagy.
FASEB J, 2021, 35(12):e22044
Curr Med Sci, 2021, 10.1007/s11596-021-2374-6
J Med Virol, 2019, 91(8):1440-1447
S3249 Corypalmine Corypalmine ((R)-(+)-Corypalmine), an alkaloid isolated from Stephania cepharantha, is an inhibitor of prolyl endopeptidase/oligopeptidase (PREP/POP) with IC50 of 128.0 μM.
Tags: PREP inhibitor|PREP agonist|PREP activator|PREP inducer|PREP antagonist|PREP signaling pathway|PREP assay kit