PREP

PREP Products

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  • PREP Inhibitors (5)
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Catalog No. Product Name Information Product Use Citations Product Validations
S2268 Baicalein Baicalein is a CYP2C9 and prolyl endopeptidase inhibitor.
SLAS Discov, 2024, S2472-5552(24)00007-8
Redox Rep, 2023, 28(1):2152607
Microbiol Spectr, 2023, 11(3):e0470222
S2396 Salidroside Salidroside (Rhodioloside), a phenylpropanoid glycoside isolated from Rhodiola rosea, has been reported to have a broad spectrum of pharmacological properties. Salidroside is a prolyl endopeptidase inhibitor. Salidroside alleviates cachexia symptoms in mouse models of cancer cachexia via activating mTOR signalling. Salidroside protects dopaminergic neurons by enhancing PINK1/Parkin-mediated mitophagy.
Mol Med Rep, 2023, 27(2)37
Research Square, 2023, 10.21203/rs.3.rs-3696850/v1
FASEB J, 2021, 35(12):e22044
S2269 Baicalin Baicalin is an inhibitor of prolyl oligopeptidase and also is an allosteric activator of carnitine palmityl transferase 1 (CPT1). Baicalin reduces the expression of NF-κB.
Chem Biol Interact, 2024, 387:110820
Int J Mol Sci, 2023, 24(11)9435
Molecules, 2021, 26(5)1210
S0842 SP-13786 SP-13786 (UAMC-1110)(compound 60) is a potent and selective inhibitor of fibroblast activation protein (FAP) and prolyl oligopeptidase (PREP) with IC50 of 3.2 nM and 1.8 μM, respectively.
S3249 Corypalmine Corypalmine ((R)-(+)-Corypalmine), an alkaloid isolated from Stephania cepharantha, is an inhibitor of prolyl endopeptidase/oligopeptidase (PREP/POP) with IC50 of 128.0 μM.
S2268 Baicalein Baicalein is a CYP2C9 and prolyl endopeptidase inhibitor.
SLAS Discov, 2024, S2472-5552(24)00007-8
Redox Rep, 2023, 28(1):2152607
Microbiol Spectr, 2023, 11(3):e0470222
S2396 Salidroside Salidroside (Rhodioloside), a phenylpropanoid glycoside isolated from Rhodiola rosea, has been reported to have a broad spectrum of pharmacological properties. Salidroside is a prolyl endopeptidase inhibitor. Salidroside alleviates cachexia symptoms in mouse models of cancer cachexia via activating mTOR signalling. Salidroside protects dopaminergic neurons by enhancing PINK1/Parkin-mediated mitophagy.
Mol Med Rep, 2023, 27(2)37
Research Square, 2023, 10.21203/rs.3.rs-3696850/v1
FASEB J, 2021, 35(12):e22044
S2269 Baicalin Baicalin is an inhibitor of prolyl oligopeptidase and also is an allosteric activator of carnitine palmityl transferase 1 (CPT1). Baicalin reduces the expression of NF-κB.
Chem Biol Interact, 2024, 387:110820
Int J Mol Sci, 2023, 24(11)9435
Molecules, 2021, 26(5)1210
S0842 SP-13786 SP-13786 (UAMC-1110)(compound 60) is a potent and selective inhibitor of fibroblast activation protein (FAP) and prolyl oligopeptidase (PREP) with IC50 of 3.2 nM and 1.8 μM, respectively.
S3249 Corypalmine Corypalmine ((R)-(+)-Corypalmine), an alkaloid isolated from Stephania cepharantha, is an inhibitor of prolyl endopeptidase/oligopeptidase (PREP/POP) with IC50 of 128.0 μM.

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Tags: PREP inhibitor|PREP agonist|PREP activator|PREP inducer|PREP antagonist|PREP signaling pathway|PREP assay kit