Melanocortin Receptor

Other GPCR & G Protein Related Inhibitors

Hedgehog/Smoothened PKA CGRP Receptor Endothelin Receptor S1P Receptor Cannabinoid Receptor SGLT Opioid Receptor GPR CCR

Cat.No.	Product Name	Information
E1002	Setmelanotide (RM-493)	Setmelanotide (RM-493, BIM-22493, CAM 4072) is a cyclic peptide full agonist of melanocortin-4 receptor (MC4R) with an EC50 of 0.27 nM and a Ki of 2.1 nM.
S0019	JNJ-10229570	JNJ-10229570 (UNII-N9IX402L35) is a potent MC1R and MC5R antagonist.
E8155	α-MSH	α-MSH (α-Melanocyte-Stimulating Hormone) is an endogenous neuropeptide and an agonist melanocortin-4 receptor (MC4R). It demonstrates anti-inflammatory, antipyretic activities, staphylocidal activity and also exhibits strong and rapid antimicrobial activity.