ROCK Rho-associated Protein Kinase

  • Compare ROCK Inhibitors
  • Research Area

ROCK Inhibitors (4)

water-soluble

Cat.No. Product Name Information Product Citations Customer Reviews
S1049 Y-27632 2HCl Y-27632 2HCl is a selective ROCK1 (p160ROCK) inhibitor with Ki of 140 nM.
S1573 Fasudil HCl (HA-1077) Fasudil is a potent inhibitor of ROCK-II, PKA, PKG, PKC, and MLCK with Ki of 0.33 μM, 1.6 μM, 1.6 μM, 3.3 μM and 36 μM, respectively.
S1459 Thiazovivin Thiazovivin (Tzv) is a novel ROCK inhibitor with IC50 of ~0.5 μM.
S1474 GSK429286A GSK429286A is a selective inhibitor of ROCK1 and ROCK2 with IC50 of 14 nM and 63 nM, respectively.
Tags: ROCK inhibition | ROCK activity | ROCK activation | Rho kinase inhibition | Rho kinase activation | Rho kinase activity | ROCK phosphorylation | ROCK signaling pathway | Rho kinase assay | Rho kinase signaling pathway | ROCK inhibitors for glaucoma | ROCK inhibitor review