Home Epigenetics PROTAC inhibitor YDR1

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YDR1 PROTAC inhibitor

Cat.No.E8294

YDR1 is a potent, selective and orally bioavailable Cereblon-based PROTAC and a degrader of SMARCA2 with DC50 of 60 nM at 48 hours. It exhibits antitumor activity in SMARCA4-mutant lung cancer xenograft models and can be used in research on non-small cell lung cancer.
YDR1 PROTAC inhibitor Chemical Structure

Chemical Structure

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Chemical Information, Storage & Stability

Molecular Weight Formula Storage (From the date of receipt)
CAS No. 2951015-31-7 -- Storage of Stock Solutions

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