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GSK-2879552 LSD1 inhibitor

Cat.No.E4596

GSK-2879552 is a selective and potent inhibitor of Lysine-specific demethylase 1 (LSD1, KDM1A), with the potential to treat Small cell lung cancer (SCLC). It induces the expression of putative KDM1A target genes and demonstrates potent, predominantly cytostatic, antiproliferative activity in SCLC cell lines and tumor xenograft models.
GSK-2879552 LSD1 inhibitor Chemical Structure

Chemical Structure

Molecular Weight: 364.48

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Chemical Information, Storage & Stability

Molecular Weight 364.48 Formula

C23H28N2O2

 Storage (From the date of receipt)
CAS No. 1401966-69-5 Download SDF Storage of Stock Solutions

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Method for preparing in vivo formulation: Take μL DMSO master liquid, next add μL Corn oil, mix and clarify.

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Mechanism of Action

Targets/IC50/Ki
LSD1/KDM1A [1]
References

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