PKMYT1

Other Apoptosis Related Inhibitors

Hedgehog/Smoothened CGRP Receptor Endothelin Receptor S1P Receptor Cannabinoid Receptor SGLT Opioid Receptor GPR CCR MT Receptor LPA Receptor

Cat.No.	Product Name	Information	Product Use Citations
E8297^New	Myt1-IN-1	Myt1-IN-1 is a potent and selective inhibitor of membrane-associated tyrosine and threonine-specific cdc2-inhibitory kinase (Myt1)(Gene: PKMYT1) with an IC50 of <10 nM. It exhibits anticancer activity and can be used in research on cancers with CCNE1 amplification or FBXW7 mutations that rely on Myt1 activity.
E0636	GSK-1520489A	GSK-1520489A(EX-A5430) is an active Protein Kinase, Membrane Associated Tyrosine/Threonine 1 (PKMYT1) inhibitor.
E1175	lunresertib (RP-6306)	lunresertib (RP-6306) is a Protein Kinase, Membrane Associated Tyrosine/Threonine 1 (PKMYT1) inhibitor, which can be used for the research of cancer.	Cell Rep, 2025, 44(8):116019 BMC Cancer, 2024, 24(1):1333

Cat.No.

Product Name

Information

Product Use Citations

Product Validations

E8297^New

Myt1-IN-1

Myt1-IN-1 is a potent and selective inhibitor of membrane-associated tyrosine and threonine-specific cdc2-inhibitory kinase (Myt1)(Gene: PKMYT1) with an IC50 of <10 nM. It exhibits anticancer activity and can be used in research on cancers with CCNE1 amplification or FBXW7 mutations that rely on Myt1 activity.

E0636

GSK-1520489A

GSK-1520489A(EX-A5430) is an active Protein Kinase, Membrane Associated Tyrosine/Threonine 1 (PKMYT1) inhibitor.

E1175

lunresertib (RP-6306)

lunresertib (RP-6306) is a Protein Kinase, Membrane Associated Tyrosine/Threonine 1 (PKMYT1) inhibitor, which can be used for the research of cancer.

Cell Rep, 2025, 44(8):116019

BMC Cancer, 2024, 24(1):1333