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ACK

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Isoform-selective Products

Cat.No. Product Name Information Product Use Citations Product Validations
S8272 XMD8-87 XMD8-87 is a novel tyrosine kinase nonreceptor 2(TNK2) inhibitor with IC50s of 38 nmol/L and 113 nmol/L for the D163E and R806Q mutations.
Cancer Cell, 2022, S1535-6108(22)00312-9
Ph.D. Thesis, Technische Universität München, 2017, Page 128 (approx)
S2212 AIM-100 AIM-100 is a potent small molecule inhibitor of Ack1 with IC50 of 24nM.
Frontiers in Immunology, 2022, 864995
Front Immunol, 2022, 13:864995
S8273 XMD16-5 XMD16-5 is a novel tyrosine kinase nonreceptor 2(TNK2) inhibitor with IC50s of 16 nmol/L and 77 nmol/L for the D163E and R806Q mutations.
Cell Rep, 2022, 41(11):111827