DprE1

Cat.No. Product Name Information Product Use Citations Product Validations
E7885 TBA-7371 TBA-7371 is a potent, noncovalent DprE1 inhibitor. TBA-7371 has potent antitubercular activity .
E7076 BTZ043 BTZ043 is an inhibitor of decaprenyl-phosphoribose-epimerase (DprE1), with MICs of of 2.3 nM and 9.2 nM for M. tuberculosis H37Rv and Mycobacterium smegmatis, respectively.
S1097 BTZ043 Racemate BTZ043 racemate is a decaprenylphosphoryl-β-D-ribose 2'-epimerase (DprE1) inhibitor acting as a new antimycobacterial agent that kill Mycobacterium tuberculosis.
Drug Deliv Transl Res, 2021, 11(4):1766-1778
J Med Chem, 2020, 28;63(10):5367-5386
Blood Adv, 2019, 3(5):797-812
S6549 PBTZ169 PBTZ169 (macozinone), an antibiotic with antimycobacterial activity, is an irreversible inhibitor of DprE1.
Cell Death Dis, 2019, 10(4):319