Histamine Receptor Agonists

Cat.No.	Product Name	Information	Product Use Citations
S1357	Lidocaine	Lidocaine (Alphacaine) is a selective inverse peripheral histamine H1-receptor agonist with an IC50 of >32 μM.	J Inflamm Res, 2025, 18:7907-7919 Cell Rep, 2022, 38(10):110468 Exp Ther Med, 2021, 21(5):424
S3968	Histamine	Histamine, an organic nitrogenous compound, is involved in local immune responses regulating physiological function in the gut and acting as a neurotransmitter for the brain, spinal cord, and uterus. It is a potent H1 and H2 receptor agonist. This compound can be used to induce animal models of Gastric and Intestinal Ulcers.	Theranostics, 2024, 14(9):3719-3738 Life Sci, 2019, 227:74-81
S4118	Histamine 2HCl	Histamine(Ceplene) is an organic nitrogen compound, acts on target cells in mammalian brain via stimulation of Histamine 1/2.Histamine 2HCl can be used to induce animal models of Gastric and Intestinal Ulcers.	Front Pharmacol, 2017, 8:667
S4382	Pyrilamine Maleate	Pyrilamine Maleate (Mepyramine)is a histamine H1 receptor inverse agonist, it binds to a G protein-coupled form of the receptor and promotes a G protein-coupled inactive state of the H1 receptor that interferes with the Gq/11-mediated signaling.	J Cell Commun Signal, 2023, 17(1):151-165
S4117	Histamine Phosphate	Histamine(Histamine diphosphate) acts directly on the blood vessels to dilate arteries and capillaries mediated by both H 1- and H 2-receptors. Histamine Phosphate can be used to induce animal models of Gastric and Intestinal Ulcers.
S6612	Betazole Dihydrochloride	Betazole Dihydrochloride (Ametazole, 2-(3-Pyrazolyl)ethanamine) is a histamine H2 agonist used clinically to test gastric secretory function.
S5498	Betahistine mesylate	Betahistine mesylate is the mesylate salt form of Betahistine, a histamine analog and H3 receptor agonist that serves as a vasodilator.
S6569	VUF10460	VUF10460 is a histamine H4 receptor agonist.
S5619	Betahistine	Betahistine is an antivertigo drug that primarily acts as a histamine H1 agonist.