Haspin Kinase

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Haspin Kinase Products

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  • Haspin Kinase Inhibitors (3)
  • New Haspin Kinase Products
Catalog No. Product Name Information Product Use Citations Product Validations
E1132New CHR-6494 CHR-6494 is a potent inhibitor of haspin, with an IC50 of 2 nM, inhibits histone H3T3 phosphorylation, and can be used in the research of cancer.
S2198 SGI-1776 free base SGI-1776 free base is a novel ATP competitive inhibitor of Pim1 with IC50 of 7 nM in a cell-free assay, 50- and 10-fold selective versus Pim2 and Pim3, also potent to Flt3 and haspin. SGI-1776 induces apoptosis and autophagy. Phase 1.
Int J Gynecol Pathol, 2022, 10.1097/PGP.0000000000000882
Cancer Res, 2021, 81(23):6029-6043
Cancer Res, 2021, canres.1023.2021
S3406 LDN-192960 LDN-192960 (Compd 1) is a potent inhibitor of Haspin and Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2) with IC50 of 10 nM and 48 nM, respectively.
Colloids Surf B Biointerfaces, 2022, 209(Pt 1):112182
E1132New CHR-6494 CHR-6494 is a potent inhibitor of haspin, with an IC50 of 2 nM, inhibits histone H3T3 phosphorylation, and can be used in the research of cancer.
S2198 SGI-1776 free base SGI-1776 free base is a novel ATP competitive inhibitor of Pim1 with IC50 of 7 nM in a cell-free assay, 50- and 10-fold selective versus Pim2 and Pim3, also potent to Flt3 and haspin. SGI-1776 induces apoptosis and autophagy. Phase 1.
Int J Gynecol Pathol, 2022, 10.1097/PGP.0000000000000882
Cancer Res, 2021, 81(23):6029-6043
Cancer Res, 2021, canres.1023.2021
S3406 LDN-192960 LDN-192960 (Compd 1) is a potent inhibitor of Haspin and Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2) with IC50 of 10 nM and 48 nM, respectively.
Colloids Surf B Biointerfaces, 2022, 209(Pt 1):112182
E1132New CHR-6494 CHR-6494 is a potent inhibitor of haspin, with an IC50 of 2 nM, inhibits histone H3T3 phosphorylation, and can be used in the research of cancer.
Tags: Haspin Kinase inhibitor|Haspin Kinase agonist|Haspin Kinase activator|Haspin Kinase inducer|Haspin Kinase antagonist|Haspin Kinase signaling pathway|Haspin Kinase assay kit