GHSR

Inhibitory Selectivity

GHSR Products

Catalog No. Information Product Use Citations Product Validations
S8673

ONC212

ONC212, a fluorinated-ONC201 analogue, is a selective agonist of GPR132. ONC212 is broadly efficacious across most solid tumors and hematological malignancies in the low nanomolar range and has robust anti-leukemic activity.

S4980

Anamorelin

Anamorelin (ONO-7643, RC-1291, ST-1291) is an orally active, high-affinity, selective agonist of the ghrelin receptor with an EC50 value of 0.74 nM in the HEK293/GRLN FLIPR assay.

S1151

Ibutamoren mesylate

Ibutamoren mesylate (MK-0667, L163191) is a potent, orally active growth hormone (GH) secretagogue. Ibutamoren (Mesylate) is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.

Catalog No. Information Product Use Citations Product Validations
S8673

ONC212

ONC212, a fluorinated-ONC201 analogue, is a selective agonist of GPR132. ONC212 is broadly efficacious across most solid tumors and hematological malignancies in the low nanomolar range and has robust anti-leukemic activity.

S4980

Anamorelin

Anamorelin (ONO-7643, RC-1291, ST-1291) is an orally active, high-affinity, selective agonist of the ghrelin receptor with an EC50 value of 0.74 nM in the HEK293/GRLN FLIPR assay.

S1151

Ibutamoren mesylate

Ibutamoren mesylate (MK-0667, L163191) is a potent, orally active growth hormone (GH) secretagogue. Ibutamoren (Mesylate) is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.