Lonafarnib (SCH66336): Mechanism of Action

Lonafarnib (SCH66336) MOA:Targeting Farnesyltransferase/Nuclear Lamin Pathway for Hutchinson-Gilford Progeria Syndrome

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Lonafarnib (SCH66336) is a potent, multi-targeting farnesyltransferase inhibitor. It affects insulin/mTOR/Akt signaling pathways by blocking farnesylation and binding viral proteins, effectively inhibiting tumor growth, viral replication, and promoting apoptosis.

Primary Applications and Mechanism of Action