MRP Inhibitors

Cat.No.	Product Name	Information	Product Use Citations
S1679	Flurbiprofen	Flurbiprofen (a member of the phenylalkanoic acid derivative family of non-steroidal anti-inflammatory drugs (NSAIDs)) is a member of the phenylalkanoic acid derivative family of non-steroidal anti-inflammatory drugs (NSAIDs).	bioRxiv, July 13, 2023, nan
S2466	Estriol	Estriol (NSC-12169) is an antagonist of the G-protein coupled estrogen receptor in estrogen receptor-negative breast cancer cells.	Mol Cell, 2019, 75(6):1103-1116.e9
S5789	Propafenone	Propafenone (SA-79) is an orally active sodium channel blocking agent and a beta-adrenoceptor (β-adrenergic receptor) antagonist. This compound offers a broad spectrum of activity in the treatment of cardiac arrhythmias.It can be used to induce animal models of Heart Failure.	Anticancer Research, December 15, 2021, 6179-6190
E4900	Enalapril	Enalapril(Eletriptan, Amprace, Vaseretic) is an inhibitor of angiotensin-converting enzyme (ACE), primarily used to treat hypertension, heart failure, and asymptomatic left ventricular dysfunction. It also attenuates frailty in aging mice.	Biochem Pharmacol, 2025, 240:117098
E2970	Gramicidin	Gramicidin from Bacillus aneurinolyticus (Bacillus brevis) is an antimicrobial peptide that destroys gram-positive bacteria. It inhibits the growth of bacteria by forming pores and channels in the cell wall, which increase its permeability to monovalent cations.
E4812	Fluoxetine	Fluoxetine (LY-110140 free base) is a selective 5-hydroxytryptamine (5-HT) reuptake inhibitor. This compound is used widely in the treatment of depression, anxiety-related symptoms and also displays anticonvulsant activity.
S4210	Benzocaine	Benzocaine(ethyl 4-aminobenzoate) is the ethyl ester of p-aminobenzoic acid (PABA), it is a local anesthetic commonly used as a topical pain reliever or in cough drops.
E6074^New	Reserpine hydrochloride	Reserpine hydrochloride (Serpivite hydrochloride) is a potent inhibitor of the vesicular monoamine transporter 2 (VMAT2) and depletes monoamines from nerve terminals. It exhibits the potential to produce a pharmacological model of depression in animals.
E0209	Cinobufotalin	Cinobufotalin, extracted from the skin secretion of the giant toad, is a novel SREBP1 inhibitor that suppresses proliferation of hepatocellular carcinoma by targeting lipogenesis.