Melanocortin Receptor
Inhibitory Selectivity
Melanocortin Receptor Products
| Catalog No. | Information | Product Use Citations | Product Validations |
|---|---|---|---|
| S0019 |
JNJ-10229570JNJ-10229570 (UNII-N9IX402L35) is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R). JNJ-10229570 inhibits sebaceous gland differentiation and the production of sebum-specific lipids. JNJ-10229570 inhibits the binding of 125I-NDP-α-MSH to cells expressing human MC1R and MC5R with IC50 of 270 nM and 200 nM, respectively. |
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| S0814New |
THIQTHIQ is a potent and selective agonist of melanocortin-4 receptor (MC4R) with IC50 of 1.2 nM and 0.6 nM for hMC4R and rMC4R, respectively. |
| Catalog No. | Information | Product Use Citations | Product Validations |
|---|---|---|---|
| S0019 |
JNJ-10229570JNJ-10229570 (UNII-N9IX402L35) is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R). JNJ-10229570 inhibits sebaceous gland differentiation and the production of sebum-specific lipids. JNJ-10229570 inhibits the binding of 125I-NDP-α-MSH to cells expressing human MC1R and MC5R with IC50 of 270 nM and 200 nM, respectively. |
| Catalog No. | Information | Product Use Citations | Product Validations |
|---|---|---|---|
| S0814New |
THIQTHIQ is a potent and selective agonist of melanocortin-4 receptor (MC4R) with IC50 of 1.2 nM and 0.6 nM for hMC4R and rMC4R, respectively. |
