Opioid Receptor Inhibitors

Cat.No.	Product Name	Information	Product Use Citations	Product Validations
S2503	Racecadotril	Racecadotril (Acetorphan) is a peripherally acting enkephalinase inhibitor with an IC50 of 4.5 μM.
S5701	Alvimopan dihydrate (LY246736 dihydrate)	Alvimopan (LY-246736) is a potent, relatively nonselective opioid antagonist with Ki values of 0.77, 4.4, and 40 nM for the μ, δ, and κ opioid receptors, respectively, displaying >100-fold selectivity over other aminergic G-protein-coupled receptors.