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S4002
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Sitagliptin phosphate monohydrate |
Sitagliptin phosphate (MK-0431) is a potent inhibitor of DPP-IV with IC50 of 19 nM in Caco-2 cell extracts. |
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S1344
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Glimepiride |
Glimepiride is a medium-to-long acting sulfonylurea anti-diabetic compound with an ED50 of 182 μg/kg. |
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S1540
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Saxagliptin (BMS-477118,Onglyza) |
Saxagliptin (BMS-477118, Onglyza) is a selective and reversible DPP4 inhibitor with IC50 of 26 nM. |
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S3031
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Linagliptin (BI-1356) |
Linagliptin is a highly potent, selective DPP-4 inhibitor with IC50 of 1 nM. |
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S3033
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Vildagliptin (LAF-237) |
Vildagliptin (LAF-237) inhibits DPP−4 with IC50 of 2.3 nM. |
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S2868
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Alogliptin (SYR-322) |
Alogliptin(SYR-322) is a potent, selective inhibitor of DPP-4 with IC50 of < 10 nM. |
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