Vasopressin receptor 1 Antagonists

Catalog No. Product Name Information Selective / Pan IC50 / Ki
S2593 Tolvaptan

Tolvaptan is an orally effective nonpeptide arginine vasopressin V2 receptor antagonist with IC50 of 3 nM, used to treat hyponatremia.

Pan vasopressin receptor 1a, IC50: 580 nM
S2920 Mozavaptan

Mozavaptan is a novel competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.

Pan Vasopressin receptor 1, IC50: 1.2 μM
S2116 Conivaptan HCl

Conivaptan HCl is a non-peptide inhibitor of antidiuretic hormone (vasopressin receptor antagonist).

Pan