RO4929097 (RG-4733): Selectivity & Specificity

RO4929097 (RG-4733) is a potent inhibitor of NOTCH1 (0.46 nM), NOTCH2, NOTCH3, NOTCH4. RO4929097 (RG-4733) exhibits the greatest inhibitory potency toward NOTCH1 (IC50 = 0.46 nM).