ICG-001 is a potent β-catenin/CBP inhibitor. It blocks Wnt/β-catenin signaling by disrupting the protein-protein interaction between β-catenin and CBP, effectively inhibiting cancer cell proliferation, migration, and tissue fibrosis.
ICG-001 MOA:Targeting CBP/Wnt/β-catenin signaling pathway for Oncology
ICG-001 is a potent β-catenin/CBP inhibitor. It blocks Wnt/β-catenin signaling by disrupting the protein-protein interaction between β-catenin and CBP, effectively inhibiting cancer cell proliferation, migration, and tissue fibrosis.