Avapritinib is a potent KIT/PDGFRA inhibitor. It affects Akt/Erk signaling by binding kinase domains to inhibit tumor growth.
Comprehensive IC50 Values for Avapritinib (BLU-285) Across Cell-free Enzyme Inhibitory Profiles and Cell-based Functional Assays.
Avapritinib is a potent KIT/PDGFRA inhibitor. It affects Akt/Erk signaling by binding kinase domains to inhibit tumor growth.