Home Peptide Products CYN154806

research use only

CYN154806

Cat.No.P1236

CYN154806, a cyclic octapeptide, is a potent and selective somatostatin SST2 receptor antagonist, with pIC50 values of 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant SST2, SST1, SST3, SST4 and SST5 receptors respectively.

Amino-acid Sequence

CYN154806 Amino-acid Sequence

CAS No. 183658-72-2

Quality Control

Batch: P123601 DMSO] 100 mg/mL] false] Ethanol] 100 mg/mL] false] Water] 50 mg/mL] false Purity: 98.21%
98.21

Chemical Information & Solubility

Storage (From the date of receipt) 3 years-20°C powder

In vitro
Batch:

DMSO : 100 mg/mL (83.51 mM)；
(Moisture-contaminated DMSO may reduce solubility. Use fresh, anhydrous DMSO.)

Ethanol : 100 mg/mL

Water : 50 mg/mL


Molecular Weight Calculator

In vivo
Batch:

Add solvents to the product individually and in order.


In vivo Formulation Calculator

Biological Activity

Description CYN154806, a cyclic octapeptide, is a potent and selective somatostatin SST2 receptor antagonist, with pIC50 values of 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant SST2, SST1, SST3, SST4 and SST5 receptors respectively.
Targets/IC50/Ki
SST2
SST3
SST4
SST1

References
  • https://pubmed.ncbi.nlm.nih.gov/10818260/

Product Information

Molecular Formula

C56H68N12O14S2
Molecular Weight 1197.34
CAS No. 183658-72-2
Appearance White Powder
Peptide Content (by %N) ≥80%
Single Impurity (by HPLC) ≤1.0%
Assay (By Anhydrous, Acetic Acid-free) 95.0~105.0%
MS Consistent
Packing plastic vial(dedicated for peptide packing) or glass vial, quantity according to customer's detail requirement.
Storage
(From the date of receipt)		 3 years-20°C powder
Shipping Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)