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CYN154806

Cat.No.P1236

CYN154806, a cyclic octapeptide, is a potent and selective somatostatin SST2 receptor antagonist, with pIC50 values of 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant SST2, SST1, SST3, SST4 and SST5 receptors respectively.
CYN154806 Chemical Structure

Chemical Structure

CAS No. 183658-72-2

Quality Control

Batch: P123601 DMSO] 100 mg/mL] false] Ethanol] 100 mg/mL] false] Water] 50 mg/mL] false Purity: 98.21%
98.21

Chemical Information & Solubility

Storage (From the date of receipt) 3 years-20°C powder

In vitro
Batch:

DMSO : 100 mg/mL (83.51 mM)；
(Moisture-contaminated DMSO may reduce solubility. Use fresh, anhydrous DMSO.)

Ethanol : 100 mg/mL

Water : 50 mg/mL


Molecular Weight Calculator

In vivo
Batch:

Add solvents to the product individually and in order.


In vivo Formulation Calculator

Biological Activity

Description CYN154806, a cyclic octapeptide, is a potent and selective somatostatin SST2 receptor antagonist, with pIC50 values of 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant SST2, SST1, SST3, SST4 and SST5 receptors respectively.
Targets/IC50/Ki
SST2
SST3
SST4
SST1

References
  • https://pubmed.ncbi.nlm.nih.gov/10818260/

Product Information

Molecular Formula

C56H68N12O14S2
Molecular Weight 1197.34
CAS No. 183658-72-2
Appearance White Powder
Peptide Content (by %N) ≥80%
Single Impurity (by HPLC) ≤1.0%
Assay (By Anhydrous, Acetic Acid-free) 95.0~105.0%
MS Consistent
Packing plastic vial(dedicated for peptide packing) or glass vial, quantity according to customer's detail requirement.
Storage
(From the date of receipt)		 3 years-20°C powder
Shipping Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)

Read more about CAS number molecular weight storage stability stock solution SMILES