Cholinesterase (ChE) Antagonists

Featured Inhibitors
Inhibitors (35)
Modulator (1)
Chemicals (11)
Agonists (2)
Activator (1)
Antagonists (3)

Cat.No.	Product Name	Information	Product Use Citations
S3809	Imperatorin	Imperatorin (Ammidin, Marmelosin, Pentosalen, 8-Isoamylenoxypsoralen), a naturally occurring psoralen-type furanocoumarin, is a potent myorelaxant agent and acts as a calcium antagonist on vascular smooth muscle.	Pharmaceuticals (Basel), 2023, 10.3390/ph16111595 Metabolites, 2022, 13(1)3 Adv Sci (Weinh), 2020, 7(16):2000925
S1890	Nizatidine	Nizatidine is a histamine H2 receptor antagonist with IC50 of 0.9 nM, also inhibits AChE with IC50 of 6.7 μM.	Gastroenterology, 2022, 162(4):1210-1225 Calcif Tissue Int, 2021, 109(6):696-705 bioRxiv, 2021, 10.1101/2021.04.29.441931
S3701	Benactyzine hydrochloride	Benactyzine hydrochloride is a centrally acting muscarinic antagonist. It is used as an antidepressant in the treatment of depression and associated anxiety.

Cat.No.

Product Name

Information

Product Use Citations

Product Validations

S3809

Imperatorin

Imperatorin (Ammidin, Marmelosin, Pentosalen, 8-Isoamylenoxypsoralen), a naturally occurring psoralen-type furanocoumarin, is a potent myorelaxant agent and acts as a calcium antagonist on vascular smooth muscle.

Pharmaceuticals (Basel), 2023, 10.3390/ph16111595

Metabolites, 2022, 13(1)3

Adv Sci (Weinh), 2020, 7(16):2000925

S1890

Nizatidine

Nizatidine is a histamine H2 receptor antagonist with IC50 of 0.9 nM, also inhibits AChE with IC50 of 6.7 μM.

Gastroenterology, 2022, 162(4):1210-1225

Calcif Tissue Int, 2021, 109(6):696-705

bioRxiv, 2021, 10.1101/2021.04.29.441931

S3701

Benactyzine hydrochloride

Benactyzine hydrochloride is a centrally acting muscarinic antagonist. It is used as an antidepressant in the treatment of depression and associated anxiety.