Cholinesterase (ChE) Antagonists

Featured Inhibitors
Inhibitors (35)
Modulator (1)
Chemicals (11)
Agonists (2)
Activator (1)
Antagonists (3)

Cat.No.	Product Name	Information	Product Use Citations
S3809	Imperatorin	Imperatorin (Ammidin, Marmelosin, Pentosalen, 8-Isoamylenoxypsoralen), a naturally occurring psoralen-type furanocoumarin, is a potent myorelaxant agent and acts as a calcium antagonist on vascular smooth muscle.	Frontiers in Cell and Developmental Biology, December 21, 2020, 592433 Pharmaceuticals, 2023, 1595 Pharmaceuticals (Basel), 2023, 10.3390/ph16111595
S1890	Nizatidine	Nizatidine is a histamine H2 receptor antagonist with IC50 of 0.9 nM, also inhibits AChE with IC50 of 6.7 μM.	Anticancer Research, July 2019, 3767-3775 Gastroenterology, 2022, 162(4):1210-1225 Calcif Tissue Int, 2021, 109(6):696-705
S3701	Benactyzine hydrochloride	Benactyzine hydrochloride is a centrally acting muscarinic antagonist. It is used as an antidepressant in the treatment of depression and associated anxiety.	Theranostics, 2024, 593-607

Cat.No.

Product Name

Information

Product Use Citations

Product Validations

S3809

Imperatorin

Imperatorin (Ammidin, Marmelosin, Pentosalen, 8-Isoamylenoxypsoralen), a naturally occurring psoralen-type furanocoumarin, is a potent myorelaxant agent and acts as a calcium antagonist on vascular smooth muscle.

Frontiers in Cell and Developmental Biology, December 21, 2020, 592433

Pharmaceuticals, 2023, 1595

Pharmaceuticals (Basel), 2023, 10.3390/ph16111595

S1890

Nizatidine

Nizatidine is a histamine H2 receptor antagonist with IC50 of 0.9 nM, also inhibits AChE with IC50 of 6.7 μM.

Anticancer Research, July 2019, 3767-3775

Gastroenterology, 2022, 162(4):1210-1225

Calcif Tissue Int, 2021, 109(6):696-705

S3701

Benactyzine hydrochloride

Benactyzine hydrochloride is a centrally acting muscarinic antagonist. It is used as an antidepressant in the treatment of depression and associated anxiety.

Theranostics, 2024, 593-607