S1PR5 Agonists | Modulators
|Catalog No.||Product Name||Information||Selective / Pan||IC50 / Ki|
BAF312 (Siponimod) is a next-generation S1P receptor agonist, selective for S1P1 and S1P5 receptors with EC50 of 0.39 nM and 0.98 nM, exhibits >1000-fold selectivity over S1P2, S1P3 and S1P4 receptors. Phase 3.
|Pan||S1P5 receptor, EC50: 0.98 nM|
Ozanimod (RPC1063) is a selective oral S1P Receptor 1 modulator. Phase 3.
|Pan||S1P5R, EC50: 11 nM|
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