NK1R Selective Antagonists
|Catalog No.||Product Name||Information||Selective / Pan||IC50 / Ki|
L-732138 (L-732,138) is a selective, potent and competitive antagonist of neurokinin-1 (NK-1) receptor/substance P (SP) receptor. L-732138 inhibits the binding of 125I-SP to the human NK-1 receptor stably expressed in CHO cells with IC50 of 2.3 nM.
|Selective||NK-1 receptor, IC50: 2.3 nM|
|S3038||Fosaprepitant dimeglumine salt||
Fosaprepitant dimeglumine salt (MK-0517) is a water-soluble phosphoryl prodrug for Aprepitant which is a NK1 antagonist.
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