Home Transmembrane Transporters MCT MCT4 Selective Inhibitors

MCT4 Selective Inhibitors

  • MCT1
  • MCT4
  • MCT2
Catalog No. Product Name Information Selective / Pan IC50 / Ki
S9929 VB124 VB124, a potent and selective MCT4 inhibitor, specifically inhibits lactate efflux/import in MDA-MB-231 cells expressing MCT4, and is used for the research of cardiac hypertrophy, heart failure, and metabolism.  Selective MCT4, IC50: 8.6 nM; MCT4, IC50: 19 nM
S9907 Syrosingopine Syrosingopine is a dual MCT1 and MCT4 inhibitor with IC50 values of 2500nM and 40 nM in HAP1 cells, respectively. Selective MCT4, IC50: 40 nM