- HIV-1 Integrase
- HIV-2 Integrase
- HIV Integrase
HIV-1-Integrase Selective Inhibitors
|Catalog No.||Product Name||Information||Selective / Pan||IC50 / Ki|
BMS-707035 is a specific HIV-I integrase (IN) inhibitor with IC50 of 15 nM. Phase 2.
|Selective||HIV-I integrase, IC50: 15 nM|
Bictegravir (GS-9883) is a novel, potent, once-daily, unboosted inhibitor of HIV-1 integrase.
Lavendustin B inhibits HIV-1 integrase (IN) interaction with its cognate cellular cofactor lens epithelium-derived growth factor (LEDGF/p75). Lavendustin B is an inhibitor of Tyrosine Kinase and also a competitive inhibitor of glucose transporter 1 (Glut1).
Elvitegravir (GS-9137, JTK-303) is an HIV integrase inhibitor for HIV-1 IIIB, HIV-2 EHO and HIV-2 ROD with IC50 of 0.7 nM, 2.8 nM and 1.4 nM in cell-free assays, respectively.
|Pan||HIV-1 IIIB, IC50: 0.7 nM|
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