GlyT2 Selective Inhibitors

Catalog No. Product Name Information Selective / Pan IC50 / Ki
S4218 Amoxapine

Amoxapine (CL 67772) is a tricyclic dibenzoxazepine (an N-aryl piperazine) which acts similarly to several other tricyclic antidepressants, amoxapine inhibits GLYT2a transport activity with IC50 of 92 μM.

Selective GlyT2a, IC50: 92 μM