AGT Selective Inhibitors

Catalog No. Product Name Information Selective / Pan IC50 / Ki
S8056 Lomeguatrib Lomeguatrib (PaTrin-2) is a potent inhibitor of O6-alkylguanine-DNA-alkyltransferase with IC50 of 5 nM. Selective O6-alkylguanine-DNA-alkyltransferas, IC50: 5 nM
S3658 O6-Benzylguanine O6-Benzylguanine (O6-BG) is a potent O6-alkylguanine DNA alkyltransferase (AGT) inactivator. Selective