Cell-free Assays (IC50/Ki) for Wortmannin (SL-2052)
| Key Target | IC50 (Cell-free) | Description | Reference |
|---|---|---|---|
| class III PI3K | 10 to 50 nM | blocking the class III PI3K pathway | Download PDF |
| PI3K enzyme | 5 nM | Enzyme activity assay | Download PDF |
| p110 catalytic subunit of PI3K | 3 nM | cell-free assay | PMC5406601 |
Cell-based Assay (IC50) for Wortmannin (SL-2052)
| Cell Type | IC50 (Cell-based) | Description | Reference |
|---|---|---|---|
| KB cells | 3.6 ± 1 µM | MTT conversion assay | PMC13092155 |
| MDA-MB-231-TFluc cells | 0.12 μM | Luciferase reporter gene assay | Download PDF |
Check the
Wortmannin (SL-2052)
product page for in-depth specifications, including solubility, stock solutions, MOA, and working concentrations.
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- Wortmannin (SL-2052) Mechanism of Action: PI3K Inhibition in Cancer Cell Research
- Wortmannin (SL-2052) Working Concentration | Cell Culture | Treatment
- Wortmannin (SL-2052) Solubility in DMSO
- Wortmannin (SL-2052) Stock Solution
- Wortmannin (SL-2052) Storage
- Wortmannin (SL-2052) Stability
- Wortmannin (SL-2052) Combination Database
- Wortmannin (SL-2052) Molecular Weight
- Wortmannin (SL-2052) SMILES
- Wortmannin (SL-2052) CAS Number
- Wortmannin (SL-2052) Chemical Structure (2D and 3D)
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- Wortmannin (SL-2052) SDS|MSDS