VVD-214 (VVD-133214, RO7589831): Mechanism of Action

VVD-214 (VVD-133214, RO7589831) MOA:Targeting WRN Helicase for Microsatellite Instability-High Solid Tumors

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VVD-214 (VVD-133214, RO7589831) is a targeted WRN inhibitor. It affects mismatch repair (MMR) and KMT2D-associated signaling, by inhibiting WRN function, effectively suppressing the proliferation of microsatellite instability (MSI) colorectal cancer cells harboring KMT2D loss-of-function mutations.

Primary Applications and Mechanism of Action