Valemetostat (DS-3201): Selectivity & Specificity
Valemetostat (DS-3201) is a potent inhibitor of EZH1 (10.0 nM), EZH2 (6.0 nM), MATE1 (0.548 µmol/L). Valemetostat (DS-3201) exhibits the greatest inhibitory potency toward EZH2 (IC50 = 6.0 nM).
Valemetostat (DS-3201) is a potent inhibitor of EZH1 (10.0 nM), EZH2 (6.0 nM), MATE1 (0.548 µmol/L). Valemetostat (DS-3201) exhibits the greatest inhibitory potency toward EZH2 (IC50 = 6.0 nM).