Valemetostat is a potent dual EZH1/2 inhibitor. It affects p53/p21 signaling by reducing H3K27me3, to inhibit tumor growth.
Comprehensive IC50 Values for Valemetostat (DS-3201) Across Cell-free Enzyme Inhibitory Profiles and Cell-based Functional Assays.
Valemetostat is a potent dual EZH1/2 inhibitor. It affects p53/p21 signaling by reducing H3K27me3, to inhibit tumor growth.