Tersolisib (STX-478): Mechanism of Action

Tersolisib (STX-478) MOA:Targeting PI3Kα/PI3K-AKT-mTOR Pathway for Breast Cancer

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Tersolisib is a mutant-specific PI3Kα inhibitor. It affects PI3K/AKT/mTOR signaling by allosteric binding, inhibiting cancer.

Primary Applications and Mechanism of Action