Tersolisib is a mutant-specific PI3Kα inhibitor. It affects PI3K/AKT/mTOR signaling by allosteric binding, inhibiting cancer.
Comprehensive IC50 Values for Tersolisib (STX-478) Across Cell-free Enzyme Inhibitory Profiles and Cell-based Functional Assays.
Tersolisib is a mutant-specific PI3Kα inhibitor. It affects PI3K/AKT/mTOR signaling by allosteric binding, inhibiting cancer.