Eltanexor (KPT-8602): Mechanism of Action

Eltanexor (KPT-8602) MOA:Targeting XPO1/Nuclear Export Pathway for Hematological Malignancies

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Eltanexor (KPT-8602) is a selective XPO1 inhibitor. It affects MAPK, STAT3, and p53 signaling pathways by binding to XPO1 and blocking nuclear export, effectively inhibiting cancer cell proliferation and promoting apoptosis.

Primary Applications and Mechanism of Action