(+)-JQ1 is a potent BRD4 inhibitor. It affects MYC signaling pathway, by blocking BRD4 binding, inhibiting tumor growth.
Comprehensive IC50 Values for (+)-JQ1 Across Cell-free Enzyme Inhibitory Profiles and Cell-based Functional Assays.
(+)-JQ1 is a potent BRD4 inhibitor. It affects MYC signaling pathway, by blocking BRD4 binding, inhibiting tumor growth.